_SKIPNAVIGATION
ITA |
ENG
Personale
Recapiti
Pagina Cercachi
Italiano
Curriculum
Pubblicazioni
Insegnamenti
English
Curriculum
Gian Luca BARTOLUCCI
Ruolo attuale:
Professore Associato
SSD:
CHEM-07/A - Chimica farmaceutica
Afferenza organizzativa:
Dipartimento di Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)
Recapiti
0554573734
gianluca.bartolucci(AT)unifi.it
Gian Luca BARTOLUCCI
Curriculum
Il sottoscritto BARTOLUCCI GIAN LUCA nato a Firenze il 03/11/67 e residente nel comune di Sesto Fiorentino in Via U. Bassi 106, dichiara :
- di essersi iscritto all’ I.T.I.S
”Tullio Buzzi” di Prato nell’anno scolastico 1981/82 e di aver conseguito il diploma di perito chimico con la specializzazione in chimica industriale nell’anno 1985/86 con la valutazione di 50/60
- di essersi iscritto alla facoltà di Farmacia dell’Università di Firenze, corso di laurea in farmacia, nell’anno 1986/87 e di aver conseguito la laurea in FARMACIA nell’anno accademico 1993/94 con la valutazione di 110/110 presentando una Tesi di laurea sperimentale con il seguente titolo : ”Sviluppo di un metodo quantitativo mediante Gascromatografia-Spettrometria di Massa in Diluizione Isotopica per il dosaggio plasmatico della Finasteride, un farmaco per la cura dell'Ipertrofia Prostatica Benigna ”
- di aver prestato servizio di supplenza annuale presso l’Istituto Professionale Femminile ”Ginori-Conti” di Firenze dal 18/10/88 al 31/08/89 in qualità di assistente tecnico di laboratorio occupandomi del laboratorio di chimica del suddetto istituto
- di aver prestato servizio di supplenza annuale presso l’I.T.I. ”Galileo Ferraris” di Empoli dal 21/10/89 al 31/03/90 in qualità di assistente tecnico di laboratorio occupandomi del laboratorio di chimica qualitativa di tale istituto (corso di diploma in chimica industriale)
- di essere stato in servizio presso l’attuale laboratorio A.R.P.A.T. (ex PMPA della U.S.L. 10/A) dal 1/10/90
al 31/10/2001 in qualità di Operatore Coordinatore Vigilanza e Ispezione
- di essere in servizio in qualità di RICERCATORE non confermato presso il Dipartimento di Scienze Farmaceutiche dell’Università degli studi di Firenze dal 01/11/2001 al 01/11/2004
- di essere in servizio in qualità di RICERCATORE confermato presso il Dipartimento di Scienze Farmaceutiche dell’Università degli studi di Firenze dal 01/11/2004 a tutt’oggi
Gian Luca BARTOLUCCI
Pubblicazioni
Legenda
Contributo su rivista |
Articolo su libro |
Libro |
Contributo in atti di convegno (proceeding) |
Brevetto |
Curatela |
Altro |
Tesi di Dottorato
Crocetti, Letizia; Catarzi, Francesca; Giovannoni, Maria Paola; Vergelli, Claudia; Bartolucci, Gianluca; Pallecchi, Marco; Paoli, Paola; Rossi, Patrizia; Lippi, Martina; Schepetkin, Igor A.; Quinn, Mark T.; Guerrini, Gabriella (2024). Ebselen analogues with dual human neutrophil elastase (HNE) inhibitory and antiradical activity. RSC MEDICINAL CHEMISTRY, pp. 1-11, ISSN:2632-8682
DOI
Niccolai, Elena; Pedone, Matteo; Martinelli, Ilaria; Nannini, Giulia; Baldi, Simone; Simonini, Cecilia; Di Gloria, Leandro; Zucchi, Elisabetta; Ramazzotti, Matteo; Spezia, Pietro Giorgio; Maggi, Fabrizio; Quaranta, Gianluca; Masucci, Luca; Bartolucci, Gian Luca; Stingo, Francesco Claudio; Mandrioli, Jessica; Amedei, Amedeo (2024). Amyotrophic lateral sclerosis stratification: unveiling patterns with virome, inflammation, and metabolism molecules. JOURNAL OF NEUROLOGY, pp. 0-0, ISSN:0340-5354
DOI
Fosca Errante, Marco Pallecchi, Gian Luca Bartolucci, Elena Frediani, Francesca Margheri, Lisa Giovannelli, Anna M. Papini, Paolo Rovero (2024). Development of a retro-inverso tetrapeptide collagen modulator as anti-aging active principle. In: 37th European Peptide Symposium and 14th International Peptide Symposium, European Peptide Society, pp. 0-0.
Russo, Edda; Bellando-Randone, Silvia; Carboni, Davide; Fioretto, Bianca Saveria; Romano, Eloisa; Baldi, Simone; El Aoufy, Khadija; Ramazzotti, Matteo; Rosa, Irene; Lepri, Gemma; Di Gloria, Leandro; Pallecchi, Marco; Bruni, Cosimo; Melchiorre, Daniela; Guiducci, Serena; Manetti, Mirko; Bartolucci, Gian Luca; Matucci-Cerinic, Marco; Amedei, Amedeo (2024). The differential crosstalk of the skin-gut microbiome axis as a new emerging actor in systemic sclerosis. RHEUMATOLOGY, vol. 63, pp. 226-234, ISSN:1462-0324
DOI
Accesso ONLINE all'editore
Niccolai, Elena; Di Gloria, Leandro; Trolese, Maria Chiara; Fabbrizio, Paola; Baldi, Simone; Nannini, Giulia; Margotta, Cassandra; Nastasi, Claudia; Ramazzotti, Matteo; Bartolucci, Gian Luca; Bendotti, Caterina; Nardo, Giovanni; Amedei, Amedeo (2024). Host genetics and gut microbiota influence lipid metabolism and inflammation: potential implications for ALS pathophysiology in SOD1G93A mice. ACTA NEUROPATHOLOGICA COMMUNICATIONS, vol. 12, pp. 0-0, ISSN:2051-5960
DOI
Maglie, Roberto; Baldi, Simone; Nannini, Giulia; Di Gloria, Leandro; Pallecchi, Marco; Bartolucci, Gianluca; Ramazzotti, Matteo; Niccolai, Elena; Baffa, Maria Efenesia; Camilla, Biagioni; Solimani, Farzan; Antiga, Emiliano; Amedei, Amedeo (2024). Alterations of circulating free fatty acids in patients with pemphigus vulgaris. EXPERIMENTAL DERMATOLOGY, vol. 33, pp. 0-0, ISSN:0906-6705
DOI
Bartolucci, Gian Luca; Pallecchi, Marco; Braconi, Laura; Dei, Silvia; Teodori, Elisabetta; Lapolla, Annunziata; Sartore, Giovanni; Traldi, Pietro (2024). Mass Spectrometry Study about In Vitro and In Vivo Reaction between Metformin and Glucose: A Preliminary Investigation on Alternative Biological Behavior. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 25, pp. 1-13, ISSN:1422-0067
DOI
Accesso ONLINE all'editore
Kaluç, Nur; Bertorello, Sara; Tombul, Oğuz Kaan; Baldi, Simone; Nannini, Giulia; Bartolucci, Gian luca; Niccolai, Elena; Amedei, Amedeo (2024). Gut-lung microbiota dynamics in mice exposed to Nanoplastics. NANOIMPACT, pp. 0-0, ISSN:2452-0748
DOI
Bellando-Randone, Silvia; Russo, Edda; Di Gloria, Leandro; Lepri, Gemma; Baldi, Simone; Fioretto, Bianca Saveria; Romano, Eloisa; Ghezzi, Giulio; Bertorello, Sara; El Aoufy, Khadija; Rosa, Irene; Pallecchi, Marco; Bruni, Cosimo; Cei, Francesco; Nannini, Giulia; Niccolai, Elena; Orlandi, Martina; Bandini, Giulia; Guiducci, Serena; Bartolucci, Gian Luca; Ramazzotti, Matteo; Manetti, Mirko; Matucci-Cerinic, Marco; Amedei, Amedeo (2024). Gut microbiota in very early systemic sclerosis: the first case-control taxonomic and functional characterisation highlighting an altered butyric acid profile. RMD OPEN, vol. 10, pp. e004647-e004647, ISSN:2056-5933
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Accesso ONLINE all'editore
Nocentini A.; Costa A.; Bonardi A.; Ammara A.; Giovannuzzi S.; Petreni A.; Bartolucci G.; Rani B.; Leri M.; Bucciantini M.; Fernandez-Bolanos J.G.; Lopez O.; Passani M.B.; Provensi G.; Gratteri P.; Supuran C.T. (2024). Enhanced Recognition Memory through Dual Modulation of Brain Carbonic Anhydrases and Cholinesterases. JOURNAL OF MEDICINAL CHEMISTRY, vol. 67, pp. 16873-16898, ISSN:1520-4804
DOI
Sofia Chioccioli , Gabriele Rocchetti , Jessica Ruzzolini , Silvia Urciuoli , Francesco Vitali, Gianluca Bartolucci , Marco Pallecchi , Giovanna Caderni, Carlotta De Filippo, Chiara Nediani, Luigi Lucini (2024). Changes in faecal microbiota profile and plasma biomarkers following the administration of an antioxidant oleuropein-rich leaf extract in a rat model mimicking colorectal cancer. ANTIOXIDANTS, vol. 13, pp. 0-0, ISSN:2076-3921
DOI
Maria Bellumori; Marco Pallecchi; Beatrice Zonfrillo; Luigi Lucio; Marta Menicatti; Marzia Innocenti; Nadia Mulinacci; Gian Luca Bartolucci (2024). Study of mono and di-O-caffeoylquinic acid isomers in Acmella oleracea extracts by HPLC-MS/MS and application of Linear Equation of Deconvolution Analysis (LEDA) algorithm for their characterization. In: 4th MS-Mass-NatMedDay, Salerno (Italy), February 15-16, 2024, Scientific Committee of 4th MS-Mass-NatMedDay, February 15-16, 2024 Salerno (Italy), pp. 67-67.
M.Pallecchi; M.Regnacq; A. Maroto; G.Bartolucci; A.Memboeuf; (2024). Thermalisation in CID MS/MS on a QqQ: towards ion trap CID excitation conditions ?. In: 40th INFORMAL MEETING ON MASS SPECTROMETRY, HUN-REN Research Centre for Natural Sciences, Magyar Tudósok krt 2, Budapest, Hungary., 12-15 May 2024, Organising Committee of 40th INFORMAL MEETING ON MASS SPECTROMETRY, HUN-REN Research Centre for Natural Sciences, Magyar Tudósok krt 2, Budapest, Hungary, 12-15 May 2024, pp. 1-1.
Accesso ONLINE all'editore
Braconi L.; Riganti C.; Parenti A.; Cecchi M.; Nocentini A.; Bartolucci G.; Menicatti M.; Contino M.; Colabufo N.A.; Manetti D.; Romanelli M.N.; Supuran C.T.; Teodori E. (2024). Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold. MOLECULES, vol. 29, pp. 1-32, ISSN:1420-3049
DOI
Accesso ONLINE all'editore
Emanuela Berrino; Bastien Michelet; Kassandra Vitse; Alessio Nocentini; Gianluca Bartolucci; Agnès Martin-Mingot; Paola Gratteri; Fabrizio Carta; Claudiu T. Supuran; Sébastien Thibaudeau (2024). Superacid-Synthesized Fluorinated Diamines Act as Selective hCA IV Inhibitors. JOURNAL OF MEDICINAL CHEMISTRY, pp. 0-0, ISSN:0022-2623
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Simone Baldi, Giuditta Pagliai, Leandro Di Gloria, Marco Pallecchi, Francesco Barca, Benedetta Pieri, Gianluca Bartolucci, Matteo Ramazzotti, Amedeo Amedei, Gianna Palendri, Francesco Sofi (2024). Beneficial Effects of Micronutrient Supplementation in Restoring the Altered Microbiota and Gut–Retina Axis in Patients with Neovascular Age-Related Macular Degeneration—A Randomized Clinical Trial. NUTRIENTS, vol. 16, pp. 3971-3985, ISSN:2072-6643
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Nannini, Giulia; Di Gloria, Leandro; Russo, Edda; Sterrantino, Gaetana; Kiros, Seble Tekle; Coppi, Marco; Niccolai, Elena; Baldi, Simone; Ramazzotti, Matteo; Di Pilato, Vincenzo; Lagi, Filippo; Bartolucci, Gian Luca; Rossolini, Gian Maria; Bartoloni, Alessandro; Amedei, Amedeo (2024). Oral microbiota signatures associated with viremia and CD4 recovery in treatment-naïve HIV-1-infected patients. MICROBES AND INFECTION, pp. 0-0, ISSN:1286-4579
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Baldi, Simone; Fabbrizzi, Alessio; Di Gloria, Leandro; Pallecchi, Marco; Nannini, Giulia; D'Ambrosio, Mario; Luceri, Cristina; Bartolucci, Gian luca; Ramazzotti, Matteo; Fontana, Giovanni; Mannini, Claudia; Lavorini, Federico; Amedei, Amedeo (2024). First Exploration of the Altered Microbial Gut-Lung Axis in the Pathogenesis of Human Refractory Chronic Cough. LUNG, vol. 202, pp. 0-0, ISSN:0341-2040
DOI
Errante, Fosca; Pallecchi, Marco; Bartolucci, Gian luca; Frediani, Elena; Margheri, Francesca; Giovannelli, Lisa; Papini, Anna M.; Rovero, Paolo (2024). Retro-inverso collagen modulator peptide derived from Serpin A1 with enhanced stability and activity in vitro. JOURNAL OF MEDICINAL CHEMISTRY, vol. 67, pp. 5053-5063, ISSN:0022-2623
DOI
Accesso ONLINE all'editore
Gitto, Stefano; Vizzutti, Francesco; Baldi, Simone; Campani, Claudia; Navari, Nadia; Falcini, Margherita; Venturi, Giulia; Montanari, Stanislao; Roccarina, Davide; Arena, Umberto; Pallecchi, Marco; Di Bonaventura, Chiara; Bartolucci, Gianluca; Ramazzotti, Matteo; Citone, Michele; Fanelli, Fabrizio; Amedei, Amedeo; Marra, Fabio (2023). Transjugular intrahepatic Porto-systemic shunt positively influences the composition and metabolic functions of the gut microbiota in cirrhotic patients. DIGESTIVE AND LIVER DISEASE, pp. 0-0, ISSN:1878-3562
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Pagliai, Giuditta; Coman, Maria Magdalena; Baldi, Simone; Dinu, Monica; Nannini, Giulia; Russo, Edda; Curini, Lavinia; Colombini, Barbara; Lotti, Sofia; Pallecchi, Marco; Di Gloria, Leandro; Bartolucci, Gianluca; Ramazzotti, Matteo; Verdenelli, Maria Cristina; Sofi, Francesco; Amedei, Amedeo (2023). Effects of the probiotic Lactiplantibacillus plantarum IMC 510® on body composition, biochemical parameters, gut microbiota composition and function, and clinical symptoms of overweight/obese subjects. FRONTIERS IN NUTRITION, vol. 10, pp. 1142527-1142537, ISSN:2296-861X
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Crocetti, Letizia; Giovannoni, Maria Paola; Guerrini, Gabriella; Lamanna, Silvia; Melani, Fabrizio; Bartolucci, Gian Luca; Pallecchi, Marco; Paoli, Paola; Lippi, Martina; Wang, Junjie; Dahl, Gerhard (2023). Design, Synthesis and Pharmacological Evaluation of New Quinoline-Based Panx-1 Channel Blockers. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 24, pp. 1-23, ISSN:1422-0067
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Accesso ONLINE all'editore
Marco Pallecchi; Marta Menicatti; Gian Luca Bartolucci (2023). Tandem mass spectrometry approaches for recognition of isomeric compounds mixtures. In: 2nd MS-SeaDay, Livorno, 11-12 July 2023, Società Chimica Italiana Divisione Spettrometria di Massa, pp. 0-0.
Accesso ONLINE all'editore
Crotti S.; Menicatti M.; Pallecchi M.; Bartolucci G. (2023). Tandem mass spectrometry approaches for recognition of isomeric compounds mixtures. MASS SPECTROMETRY REVIEWS, pp. 0-0, ISSN:0277-7037
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Pallecchi M.; Lucio L.; Braconi L.; Menicatti M.; Dei S.; Teodori E.; Bartolucci G. (2023). Isomers Recognition in HPLC-MS/MS Analysis of Human Plasma Samples by Using an Ion Trap Supported by a Linear Equations-Based Algorithm. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 24, pp. 0-0, ISSN:1422-0067
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Accesso ONLINE all'editore
Castellini G, Cassioli E, Vitali F, Rossi E, Dani C, Melani G, Flaccomio D, D'Andria M, Mejia Monroy M, Galli A, Cavalieri D, Ricca V, Bartolucci GL, De Filippo C (2023). Gut microbiota metabolites mediate the interplay between childhood maltreatment and psychopathology in patients with eating disorders. SCIENTIFIC REPORTS, pp. 0-0, ISSN:2045-2322
Gerace, Elisabetta; Baldi, Simone; Salimova, Maya; Di Gloria, Leandro; Curini, Lavinia; Cimino, Virginia; Nannini, Giulia; Russo, Edda; Pallecchi, Marco; Ramazzotti, Matteo; Bartolucci, Gianluca; Occupati, Brunella; Lanzi, Cecilia; Scarpino, Maenia; Lanzo, Giovanni; Grippo, Antonello; Lolli, Francesco; Mannaioni, Guido; Amedei, Amedeo (2023). Oral and fecal microbiota perturbance in cocaine users: Can rTMS-induced cocaine abstinence support eubiosis restoration?. ISCIENCE, vol. 26, pp. 106627-106627, ISSN:2589-0042
DOI
Bellumori, Maria; Pallecchi, Marco; Zonfrillo, Beatrice; Lucio, Luigi; Menicatti, Marta; Innocenti, Marzia; Mulinacci, Nadia; Bartolucci, Gian Luca (2023). Study of Mono and Di-O-caffeoylquinic Acid Isomers in Acmella oleracea Extracts by HPLC-MS/MS and Application of Linear Equation of Deconvolution Analysis Algorithm for Their Characterization. PHARMACEUTICALS, vol. 16, pp. 0-0, ISSN:1424-8247
DOI
Accesso ONLINE all'editore
Silvano, Angela; Niccolai, Elena; Baldi, Simone; Seravalli, Viola; Strambi, Noemi; Nannini, Giulia; Pallecchi, Marco; Bartolucci, Gianluca; Parenti, Astrid; Amedei, Amedeo; Di Tommaso, Mariarosaria (2023). Exploring Plasma-Level Gut Microbiota Mediators and Pro-Inflammatory Markers in Pregnant Women with Short Cervix and Gestational Diabetes Mellitus. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 24, pp. 13653-13653, ISSN:1422-0067
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Braconi L.; Dei S.; Contino M.; Riganti C.; Bartolucci G.; Manetti D.; Romanelli M.N.; Perrone M.G.; Colabufo N.A.; Guglielmo S.; Teodori E. (2023). Tetrazole and oxadiazole derivatives as bioisosteres of tariquidar and elacridar: New potent P-gp modulators acting as MDR reversers. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 259, pp. 0-0, ISSN:1768-3254
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M. Pallecchi; G. Bartolucci; L. Braconi; S. Dei; E. Teodori; A. Lapolla; G. Sartore; P. Traldi; (2023). Metformin reacts directly with glucose following the Maillard reaction pathway. In: 39th INFORMAL MEETING ON MASS SPECTROMETRY, Sorbonne Université, Paris, France, 15th – 17th May 2023, Organising Committee of 39th INFORMAL MEETING ON MASS SPECTROMETRY, Sorbonne Université, Paris, France 15th – 17th May 2023, pp. 55-55.
M. Pallecchi; L. Braconi; M. Menicatti; S. Giachetti; S. Dei; E. Teodori; Gian Luca Bartolucci (2023). Application of LEDA Algorithm for the characterization of Isomers in Simultaneous Degradation Study in Human Plasma by HPLC-MS/MS. In: 39th INFORMAL MEETING ON MASS SPECTROMETRY, Sorbonne Université, Paris, France, 15th – 17th May 2023, Organising Committee of 39th INFORMAL MEETING ON MASS SPECTROMETRY, Sorbonne Université, Paris, France 15th – 17th May 2023, pp. 49-49.
Accesso ONLINE all'editore
A. Memboeuf; D. Jeanne Dit Fouque; M. Pallecchi; A.Maroto; G.Bartolucci (2023). Collisional cooling in CID tandem MS ion trap experiments. In: 39th INFORMAL MEETING ON MASS SPECTROMETRY, Sorbonne Université, Paris, France, 15th – 17th May 2023, Organising Committee of 39th INFORMAL MEETING ON MASS SPECTROMETRY, Sorbonne Université, Paris, France 15th – 17th May 2023, pp. 63-63.
Accesso ONLINE all'editore
BALDI S; TRISTAN ASENSI M; PALLECCHI M; SOFI F; BARTOLUCCI G; AMEDEI A (2023). Interplay between Lignans and Gut Microbiota: Nutritional, Functional and Methodological Aspects. MOLECULES, vol. 28, pp. 2-14, ISSN:1420-3049
Niccolai, Elena; Bettiol, Alessandra; Baldi, Simone; Silvestri, Elena; Di Gloria, Leandro; Bello, Federica; Nannini, Giulia; Ricci, Federica; Nicastro, Maria; Ramazzotti, Matteo; Vaglio, Augusto; Bartolucci, Gianluca; Emmi, Giacomo; Amedei, Amedeo; Prisco, Domenico (2022). Gut Microbiota and Associated Mucosal Immune Response in Eosinophilic Granulomatosis with Polyangiitis (EGPA). BIOMEDICINES, vol. 10, pp. 1227--, ISSN:2227-9059
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Baldi, Simone; Dinu, Monica; Pagliai, Giuditta; Colombini, Barbara; Di Gloria, Leandro; Curini, Lavinia; Pallecchi, Marco; Ramazzotti, Matteo; Bartolucci, Gianluca; Benedettelli, Stefano; Amedei, Amedeo; Sofi, Francesco (2022). Effect of ancient wheat pasta on gut microbiota composition and bacteria-derived metabolites: A randomized controlled trial. FRONTIERS IN NUTRITION, vol. 9, pp. 971666-971674, ISSN:2296-861X
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Sartiani, Laura; Bartolucci, Gian Luca; Pallecchi, Marco; Spinelli, Valentina; Cerbai, Elisabetta (2022). Pharmacological basis of the antifibrotic effects of pirfenidone: Mechanistic insights from cardiac in-vitro and in-vivo models. FRONTIERS IN CARDIOVASCULAR MEDICINE, vol. 9, pp. 0-0, ISSN:2297-055X
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Braconi L.; Teodori E.; Contino M.; Riganti C.; Bartolucci G.; Manetti D.; Romanelli M.N.; Perrone M.G.; Colabufo N.A.; Guglielmo S.; Dei S. (2022). Overcoming Multidrug Resistance (MDR): Design, Biological Evaluation and Molecular Modelling Studies of 2,4-Substituted Quinazoline Derivatives. CHEMMEDCHEM, pp. e202200027-21, ISSN:1860-7179
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Pallecchi, Marco; Braconi, Laura; Menicatti, Marta; Giachetti, Sara; Dei, Silvia; Teodori, Elisabetta; Bartolucci, Gian Luca (2022). Simultaneous Degradation Study of Isomers in Human Plasma by HPLC-MS/MS and Application of LEDA Algorithm for Their Characterization. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 23, pp. 0-0, ISSN:1422-0067
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Letizia Crocetti, Gabriella Guerrini, Claudia Vergelli, Maria Paola Giovannoni, Gian Luca Bartolucci, Silvia Lamanna, Marco Pallecchi, Paola Paoli, Patrizia Rossi (2022). Molecular manipulation of the 1,5,6,7-tetrahydro-4 H -indazol-4-one scaffold to obtain new human neutrophil elastase (HNE) inhibitors. JOURNAL OF MOLECULAR STRUCTURE, vol. 1263, pp. 133140-133154, ISSN:0022-2860
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Chiaramonte N.; Angeli A.; Sgambellone S.; Bonardi A.; Nocentini A.; Bartolucci G.; Braconi L.; Dei S.; Lucarini L.; Teodori E.; Gratteri P.; Wunsch B.; Supuran C.T.; Romanelli M.N. (2022). 2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 228, pp. 0-0, ISSN:0223-5234
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Russo, Edda; Nannini, Giulia; Sterrantino, Gaetana; Kiros, Seble Tekle; Di Pilato, Vincenzo; Coppi, Marco; Baldi, Simone; Niccolai, Elena; Ricci, Federica; Ramazzotti, Matteo; Pallecchi, Marco; Lagi, Filippo; Rossolini, Gian Maria; Bartoloni, Alessandro; Bartolucci, Gianluca; Amedei, Amedeo (2022). Effects of viremia and CD4 recovery on gut "microbiome-immunity" axis in treatment-naïve HIV-1-infected patients undergoing antiretroviral therapy. WORLD JOURNAL OF GASTROENTEROLOGY, vol. 28, pp. 635-652, ISSN:2219-2840
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Pallecchi, Marco; Menicatti, Marta; Braconi, Laura; Supuran, Claudiu T; Dei, Silvia; Teodori, Elisabetta; Bartolucci, Gian Luca (2022). Application of LEDA algorithm for the recognition of P-glycoprotein and Carbonic Anhydrase hybrid inhibitors and evaluation of their plasma stability by HPLC-MS/MS analysis. JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, vol. 219, pp. 0-0, ISSN:0731-7085
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Chiaramonte N.; Gabellini A.; Angeli A.; Bartolucci G.; Braconi L.; Dei S.; Teodori E.; Supuran C.T.; Romanelli M.N. (2022). New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I Activators. MOLECULES, vol. 27, pp. 0-0, ISSN:1420-3049
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Micheli L.; Lucarini E.; Toti A.; Ferrara V.; Ciampi C.; Parisio C.; Bartolucci G.; Di Cesare Mannelli L.; Ghelardini C. (2022). Effects of Ultramicronized N-Palmitoylethanolamine Supplementation on Tramadol and Oxycodone Analgesia and Tolerance Prevention. PHARMACEUTICS, vol. 14, pp. 403-403, ISSN:1999-4923
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Lucarini E, Di Pilato V, Parisio C, Micheli L, Toti A, Pacini A, Bartolucci G, Baldi S, Niccolai E, Amedei A, Rossolini GM, Nicoletti C, Cryan JF, O'Mahony SM, Ghelardini C, Di Cesare Mannelli L. (2022). Visceral sensitivity modulation by faecal microbiota transplantation: the active role of gut bacteria in pain persistence. PAIN, pp. 1-17, ISSN:1872-6623
Giovannuzzi S.; D'ambrosio M.; Luceri C.; Osman S.M.; Pallecchi M.; Bartolucci G.; Nocentini A.; Supuran C.T. (2022). Aromatic sulfonamides including a sulfonic acid tail: New membrane impermeant carbonic anhydrase inhibitors for targeting selectively the cancer‐associated isoforms. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 23, pp. 0-0, ISSN:1422-0067
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Micheli, Laura; Lucarini, Elena; Nobili, Stefania; Bartolucci, Gianluca; Pallecchi, Marco; Toti, Alessandra; Ferrara, Valentina; Ciampi, Clara; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo (2022). Ultramicronized N-palmitoylethanolamine contributes to morphine efficacy against neuropathic pain: implication of mast cells and glia. CURRENT NEUROPHARMACOLOGY, vol. 21, pp. 0-0, ISSN:1570-159X
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Braconi, Laura; Teodori, Elisabetta; Riganti, Chiara; Coronnello, Marcella; Nocentini, Alessio; Bartolucci, Gian Luca; Pallecchi, Marco; Contino, Marialessandra; Manetti, Dina; Romanelli, Maria Novella; Supuran, Claudiu T; Dei, Silvia (2022). New dual P-Glycoprotein (P-gp) and human carbonic anhydrase XII (hCA XII) inhibitors as Multidrug Resistance (MDR) reversers in cancer cells. JOURNAL OF MEDICINAL CHEMISTRY, vol. 65, pp. 14655-14672, ISSN:0022-2623
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Sofia Chioccioli; Jessica Ruzzolini; Silvia Urciuoli; Gian Luca Bartolucci; Marco Pallecchi; Lido Calorini; Carlotta De Filippo; Francesco Vitali; Chiara Nediani; Francesca Bianchini; Giovanna Caderni (2022). Oleuropein-rich leaf extract affects intestinal microbiota and free fatty acids in Apc-mutant and wt rats. In: 7th MS-Food, Florence (Italy), 5-7 October 2022, Scientific Committee of 7th MS-Food, 5-7 October 2022, Florence (Italy), pp. 68-69.
Russo, Edda; Cinci, Lorenzo; Di Gloria, Leandro; Baldi, Simone; D'Ambrosio, Mario; Nannini, Giulia; Bigagli, Elisabetta; Curini, Lavinia; Pallecchi, Marco; Andrea Arcese, Donato; Scaringi, Stefano; Malentacchi, Cecilia; Bartolucci, Gianluca; Ramazzotti, Matteo; Luceri, Cristina; Amedei, Amedeo; Giudici, Francesco (2022). Crohn's disease recurrence updates: first surgery vs. surgical relapse patients display different profiles of ileal microbiota and systemic microbial-associated inflammatory factors. FRONTIERS IN IMMUNOLOGY, vol. 13, pp. 1-18, ISSN:1664-3224
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Baldi, Simone; Pagliai, Giuditta; Dinu, Monica; Di Gloria, Leandro; Nannini, Giulia; Curini, Lavinia; Pallecchi, Marco; Russo, Edda; Niccolai, Elena; Danza, Giovanna; Benedettelli, Stefano; Ballerini, Giovanna; Colombini, Barbara; Bartolucci, Gianluca; Ramazzotti, Matteo; Sofi, Francesco; Amedei, Amedeo (2022). Effect of ancient Khorasan wheat on gut microbiota, inflammation, and short-chain fatty acid production in patients with fibromyalgia. WORLD JOURNAL OF GASTROENTEROLOGY, vol. 28, pp. 1965-1980, ISSN:1007-9327
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Federica, Ricci; Edda, Russo; Daniela, Renzi; Simone, Baldi; Giulia, Nannini; Gabriele, Lami; Marta, Menicatti; Marco, Pallecchi; Gianluca, Bartolucci; Elena, Niccolai; Matteo, Cerboneschi; Serena, Smeazzetto; Matteo, Ramazzotti; Amedeo, Amedei; Salvatore, Calabrò Antonino (2022). Characterization of the "gut microbiota-immunity axis" and microbial lipid metabolites in atrophic and potential celiac disease. FRONTIERS IN MICROBIOLOGY, vol. 13, pp. 0-0, ISSN:1664-302X
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Vannozzi G.; Vullo D.; Angeli A.; Ferraroni M.; Combs J.; Lomelino C.; Andring J.; Mckenna R.; Bartolucci G.; Pallecchi M.; Lucarini L.; Sgambellone S.; Masini E.; Carta F.; Supuran C.T. (2021). One-Pot Procedure for the Synthesis of Asymmetric Substituted Ureido Benzene Sulfonamides as Effective Inhibitors of Carbonic Anhydrase Enzymes. JOURNAL OF MEDICINAL CHEMISTRY, vol. 65, pp. 824-837, ISSN:0022-2623
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Marco Pallecchi, Marta Menicatti, Gian Luca Bartolucci (2021). Drug Plasma Stability of PG-P and Carbonic Anhydrase hybrids inhibitors by LC-MS/MS and application of LEDA algorithm for their characterization. In: 9th J-Day, i giovani e la spettrometria di massa, on-line, 24-Giugno-2021, Divisione di Spettrometria di Massa della Società Chimica Italiana, pp. 47-47.
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Cantini, Niccolò; Khlebnikov, Andrei I.; Crocetti, Letizia; Schepetkin, Igor A.; Floresta, Giuseppe; Guerrini, Gabriella; Vergelli, Claudia; Bartolucci, Gianluca; Quinn, Mark T.; Paola Giovannoni, Maria (2021). Exploration of Nitrogen Heterocycle Scaffolds for the Development of Potent Human Neutrophil Elastase Inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 29, pp. 1-17, ISSN:0968-0896
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Errante, Fosca; Menicatti, Marta; Pallecchi, Marco; Giovannelli, Lisa; Papini, Anna Maria; Rovero, Paolo; Bartolucci, Gian Luca (2021). Susceptibility of cosmeceutical peptides to proteases activity: Development of dermal stability test by LC-MS/MS analysis. JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, vol. 194, pp. 1-9, ISSN:0731-7085
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Baldi S.; Menicatti M.; Nannini G.; Niccolai E.; Russo E.; Ricci F.; Pallecchi M.; Romano F.; Pedone M.; Poli G.; Renzi D.; Taddei A.; Calabro A.S.; Stingo F.C.; Bartolucci G.; Amedei A. (2021). Free fatty acids signature in human intestinal disorders: Significant association between butyric acid and celiac disease. NUTRIENTS, vol. 13, pp. 1-14, ISSN:2072-6643
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Dugheri S.; Mucci N.; Mini E.; Squillaci D.; Marrubini G.; Bartolucci G.; Bucaletti E.; Cappelli G.; Trevisani L.; Arcangeli G. (2021). Characterization and separation of platinum-based antineoplastic drugs by zwitterionic hydrophilic interaction liquid chromatography (Hilic)–tandem mass spectrometry, and its application in surface wipe sampling. SEPARATIONS, vol. 8, pp. 0-0, ISSN:2297-8739
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Nicolo S.; Tanturli M.; Mattiuz G.; Antonelli A.; Baccani I.; Bonaiuto C.; Baldi S.; Nannini G.; Menicatti M.; Bartolucci G.; Rossolini G.M.; Amedei A.; Torcia M.G. (2021). Vaginal lactobacilli and vaginal dysbiosis-associated bacteria differently affect cervical epithelial and immune homeostasis and anti-viral defenses. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 22, pp. 0-0, ISSN:1661-6596
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Dugheri S.; Mucci N.; Squillaci D.; Marrubini G.; Bartolucci G.; Melzi C.; Bucaletti E.; Cappelli G.; Trevisani L.; Arcangeli G. (2021). Developing a fast ultra-high-performance liquid chromatography–tandem mass spectrometry method for high-throughput surface contamination monitoring of 26 antineoplastic drugs. SEPARATIONS, vol. 8, pp. 0-0, ISSN:2297-8739
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Kucukbay H.; Gonul Z.; Kucukbay F.Z.; Tekin Z.; Angeli A.; Bartolucci G.; Supuran C.T.; Tatlici E.; Apohan E.; Yesilada O. (2021). Synthesis of new 7-amino-3,4-dihydroquinolin-2(1H)-one-peptide derivatives and their carbonic anhydrase enzyme inhibition, antioxidant, and cytotoxic activities. ARCHIV DER PHARMAZIE, vol. 354, pp. 0-0, ISSN:0365-6233
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Kucukbay H.; Parladi F.M.; Kucukbay F.Z.; Angeli A.; Bartolucci G.; Supuran C.T. (2021). Synthesis, antioxidant and carbonic anhydrase inhibitory properties of monopeptide-anthraquinone conjugates. ORGANIC COMMUNICATIONS, vol. 14, pp. 255-269, ISSN:1307-6175
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Niccolai E.; Di Pilato V.; Nannini G.; Baldi S.; Russo E.; Zucchi E.; Martinelli I.; Menicatti M.; Bartolucci G.; Mandrioli J.; Amedei A. (2021). The gut microbiota-immunity axis in als: A role in deciphering disease heterogeneity?. BIOMEDICINES, vol. 9, pp. 0-0, ISSN:2227-9059
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V. Fiorini, Fabio Villanelli, Gian Luca Bartolucci, Giovanna Danza (2021). Development of a method for the quantification of estrone and estradiol in serum by LC-MS/MS. In: 9th J-Day, i giovani e la spettrometria di massa, on-line, 24-Giugno-2021, Divisione di Spettrometria di Massa della Società Chimica Italiana, pp. 28-28.
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Cantini, Niccolo; Crocetti, Letizia; Guerrini, Gabriella; Vergelli, Claudia; Schepetkin, Igor A; Pallecchi, Marco; Bartolucci, Gian Luca; Quinn, Mark T; Teodori, Elisabetta; Paola Giovannoni, Maria (2021). 1,5,6,7-Tetrahydro-4H-indazol-4-ones as human neutrophil elastase (HNE) inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 52, pp. 128380-128386, ISSN:0960-894X
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Braconi L.; Bartolucci G.; Contino M.; Chiaramonte N.; Giampietro R.; Manetti D.; Perrone M.G.; Romanelli M.N.; Colabufo N.A.; Riganti C.; Dei S.; Teodori E. (2020). 6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 974-992, ISSN:1475-6366
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Niccolò Chiaramonte, Soumia Maach, Caterina Biliotti, Andrea Angeli, Gian luca Bartolucci, Laura Braconi, Silvia Dei, Elisabetta Teodori, Claudiu T. Supuran, Maria Novella Romanelli (2020). Synthesis and carbonic anhydrase activating properties of a series of 2-amino-imidazolines structurally related to clonidine. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 1003-1010, ISSN:1475-6366
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Dugheri S.; Marrubini G.; Speltini A.; Mucci N.; Cappelli G.; Bartolucci G.; Arcangeli G. (2020). Fully Automated Determination of Trimellitic Anhydride in Saturated Polyester Resins Using Programmed Temperature Vaporization-Large Volume Injection-Gas Chromatography Previous Aqueous Derivatization with Triethyloxonium Tetrafluoroborate. CHROMATOGRAPHIA, vol. 83, pp. 601-613, ISSN:0009-5893
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Berrino E.; Angeli A.; Zhdanov D.D.; Kiryukhina A.P.; Milaneschi A.; De Luca A.; Bozdag M.; Carradori S.; Selleri S.; Bartolucci G.; Peat T.S.; Ferraroni M.; Supuran C.T.; Carta F. (2020). Azidothymidine "clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors. JOURNAL OF MEDICINAL CHEMISTRY, vol. 63, pp. 7392-7409, ISSN:0022-2623
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Nocentini A.; Alterio V.; Bua S.; Micheli L.; Esposito D.; Buonanno M.; Bartolucci G.; Osman S.M.; Alothman Z.A.; Cirilli R.; Pierini M.; Monti S.M.; Di Cesare Mannelli L.; Gratteri P.; Ghelardini C.; De Simone G.; Supuran C.T. (2020). Phenyl(thio)phosphon(amid)ate Benzenesulfonamides as Potent and Selective Inhibitors of Human Carbonic Anhydrases II and VII Counteract Allodynia in a Mouse Model of Oxaliplatin-Induced Neuropathy. JOURNAL OF MEDICINAL CHEMISTRY, vol. 63, pp. 5185-5200, ISSN:0022-2623
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Pagliai, Giuditta; Russo, Edda; Niccolai, Elena; Dinu, Monica; Di Pilato, Vincenzo; Magrini, Alessandro; Bartolucci, Gianluca; Baldi, Simone; Menicatti, Marta; Giusti, Betti; Marcucci, Rossella; Rossolini, Gian Maria; Casini, Alessandro; Sofi, Francesco; Amedei, Amedeo (2020). Influence of a 3-month low-calorie Mediterranean diet compared to the vegetarian diet on human gut microbiota and SCFA: The CARDIVEG study. EUROPEAN JOURNAL OF NUTRITION, vol. 59, pp. 2011-2024, ISSN:1436-6207
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Teodori E.; Braconi L.; Bua S.; Lapucci A.; Bartolucci G.; Manetti D.; Romanelli M.N.; Dei S.; Supuran C.T.; Coronnello M. (2020). Dual P-glycoprotein and CA XII inhibitors: A new strategy to reverse the P-gp Mediated Multidrug Resistance (MDR) in cancer cells y. MOLECULES, vol. 25, pp. 1-26, ISSN:1420-3049
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Menicatti M.; Pallecchi M.; Ricciutelli M.; Galarini R.; Moretti S.; Sagratini G.; Vittori S.; Lucarini S.; Caprioli G.; Bartolucci G. (2020). Determination of coeluted isomers in wine samples by application of MS/MS deconvolution analysis. JOURNAL OF MASS SPECTROMETRY, vol. 55, pp. e4607-e4615, ISSN:1076-5174
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Ricciutelli M.; Bartolucci G.; Campana R.; Salucci S.; Benedetti S.; Caprioli G.; Maggi F.; Sagratini G.; Vittori S.; Lucarini S. (2020). Quantification of 2- and 3-isopropylmalic acids in forty Italian wines by UHPLC-MS/MS triple quadrupole and evaluation of their antimicrobial, antioxidant activities and biocompatibility. FOOD CHEMISTRY, vol. 321, pp. 126726-126734, ISSN:0308-8146
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Kucukbay H.; Gonul Z.; Kucukbay F.Z.; Angeli A.; Bartolucci G.; Supuran C.T. (2020). Preparation, carbonic anhydrase enzyme inhibition and antioxidant activity of novel 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives incorporating mono or dipeptide moiety. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 1021-1026, ISSN:1475-6366
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Marco Pallecchi, Marta Menicatti, Gian Luca Bartolucci (2020). Development of a HPLC-MS/MS method for the pharmacokinetic studies of Pirfenidone in pig plasma. In: Massa 2020-VIP (Virtual International Pre-congress), on-line, 2020, Divisione di Spettrometria di Massa della Società Chimica Italiana, pp. 129-130.
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Bua S.; Lucarini L.; Micheli L.; Menicatti M.; Bartolucci G.; Selleri S.; Di Cesare Mannelli L.; Ghelardini C.; Masini E.; Carta F.; Gratteri P.; Nocentini A.; Supuran C.T. (2020). Bioisosteric Development of Multitarget Nonsteroidal Anti-Inflammatory Drug-Carbonic Anhydrases Inhibitor Hybrids for the Management of Rheumatoid Arthritis. JOURNAL OF MEDICINAL CHEMISTRY, vol. 63, pp. 2325-2342, ISSN:0022-2623
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Kucukbay H.; Bugday N.; Kucukbay F.Z.; Ageli A.; Bartolucci G.; Supuran C.T. (2020). Synthesis and human carbonic anhydrase I, II, VA, and XII inhibition with novel amino acid–sulphonamide conjugates. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 489-497, ISSN:1475-6366
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Aimo A.; Cerbai E.; Bartolucci G.; Adamo L.; Barison A.; Lo Surdo G.; Biagini S.; Passino C.; Emdin M. (2020). Pirfenidone is a cardioprotective drug: Mechanisms of action and preclinical evidence. PHARMACOLOGICAL RESEARCH, vol. 155, pp. 104694-104694, ISSN:1043-6618
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Silvia Dei, Laura Braconi, Alfonso Trezza, Marta Menicatti, Marialessandra Contino, Marcella Coronnello, Niccolò Chiaramonte, Dina Manetti, Maria Grazia Perrone, Maria Novella Romanelli, Chatchanok Udomtanakunchai, Nicola Antonio Colabufo, Gian luca Bartolucci, Ottavia Spiga, Milena Salerno, Elisabetta Teodori (2019). Modulation of the spacer in N,N-bis(alkanol)amine aryl ester heterodimers led to the discovery of a series of highly potent P-glycoprotein-based multidrug-resistance (MDR) modulators. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 172, pp. 71-94, ISSN:1768-3254, Elsevier Masson SAS:
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Betti, Marco; Catarzi, Daniela; Varano, Flavia; Falsini, Matteo; Varani, Katia; Vincenzi, Fabrizio; Pasquini, Silvia; di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Lucarini, Elena; Dal Ben, Diego; Spinaci, Andrea; Bartolucci, Gian Luca; Menicatti, Marta; Colotta, Vittoria (2019). Modifications on the Amino-3,5-dicyanopyridine Core To Obtain Multifaceted Adenosine Receptor Ligands with Antineuropathic Activity. JOURNAL OF MEDICINAL CHEMISTRY, vol. 62, pp. 6894-6912, ISSN:0022-2623
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Dugheri S.; Mucci N.; Cappelli G.; Bonari A.; Campagna M.; Arcangeli G.; Bartolucci G. (2019). New fully automated gas chromatographic analysis of urinary S-phenylmercapturic acid in isotopic dilution using negative chemical ionization with isobutane as reagent gas. JOURNAL OF MASS SPECTROMETRY, pp. 0-0, ISSN:1076-5174
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Stefano Dugheri, Nicola Mucci, Giovanni Cappelli, Alessandro Bonari, Marcello Campagna, Giulio Arcangeli, Gian Luca Bartolucci (2019). New fully automated gas-cromatographic analysis of urinary s-phenylmercapturic acid using negative chemical ionization with isobutane as reagent gas. In: 37th Informal Meeting on Mass Spectrometry, Fiera di Primiero (TN), 05-08 Maggio 2019, 37th Informal Meeting on Mass Spectrometry organizing committee, pp. 93-93, ISBN:978-88-93495-59-2
Küçükbay, Hasan*; Buğday, Nesrin; Küçükbay, F. Zehra; Berrino, Emanuela; Bartolucci, Gian Luca; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T. (2019). Synthesis and carbonic anhydrase inhibitory properties of novel 4-(2-aminoethyl)benzenesulfonamide-dipeptide conjugates. BIOORGANIC CHEMISTRY, vol. 83, pp. 414-423, ISSN:0045-2068
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Morelli A, Filippi S, Comeglio P, Sarchielli E, Cellai I, Pallecchi M, Bartolucci G, Danza G, Rastrelli G, Corno C, Guarnieri G, Fuochi E, Vignozzi L, Maggi M (2019). Physical activity counteracts metabolic syndrome-induced hypogonadotropic hypogonadism and erectile dysfunction in the rabbit.. AMERICAN JOURNAL OF PHYSIOLOGY: ENDOCRINOLOGY AND METABOLISM, vol. 316, pp. 519-535, ISSN:0193-1849
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Maria Novella Romanelli, Martina Del Lungo, Luca Guandalini,Mehrnoush Zobeiri, Andras Gyokeres, TAmas Arpadffy-Lovas, Istvan Koncz, Laura Sartiani, Gian Luca Bartolucci, Silvia Dei, Dina Manetti, Elisabetta Teodori, Thomas Budde, Elisabetta Cerbai (2019). EC18 as a Tool To Understand the Role of HCN4 Channels in Mediating Hyperpolarization-Activated Current in Tissues. ACS MEDICINAL CHEMISTRY LETTERS, vol. 10, pp. 584-589, ISSN:1948-5875
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Angeli A.; Di Cesare Mannelli L.; Ghelardini C.; Peat T.S.; Bartolucci G.; Menicatti M.; Carta F.; Supuran C.T. (2019). Benzensulfonamides bearing spyrohydantoin moieties act as potent inhibitors of human carbonic anhydrases II and VII and show neuropathic pain attenuating effects. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 177, pp. 188-197, ISSN:1768-3254
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Dina Manetti*† , Alexandra Garifulina‡, Gian Luca Bartolucci , Carla Bazzicalupi§ , Cristina Bellucci†, Niccolò Chiaramonte†, Silvia Dei†, Lorenzo Di Cesare Mannelli∥, Carla Ghelardini∥, Paola Gratteri⊥ , Ekaterina Spirova‡, Irina Shelukhina‡, Elisabetta Teodori†, Katia Varani#, Victor Tsetlin‡, Maria Novella Romanelli† (2019). New Rigid Nicotine Analogues, Carrying a Norbornane Moiety, Are Potent Agonists of α7 and α3∗ Nicotinic Receptors. JOURNAL OF MEDICINAL CHEMISTRY, vol. 62, pp. 1887-1901, ISSN:0022-2623
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Berrino E.; Milazzo L.; Micheli L.; Vullo D.; Angeli A.; Bozdag M.; Nocentini A.; Menicatti M.; Bartolucci G.; Di Cesare Mannelli L.; Ghelardini C.; Supuran C.T.; Carta F. (2019). Synthesis and evaluation of carbonic anhydrase inhibitors with carbon monoxide releasing properties for the management of rheumatoid arthritis. JOURNAL OF MEDICINAL CHEMISTRY, vol. 62, pp. 7233-7249, ISSN:1520-4804
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Braconi L., Bartolucci G., Manetti D., Romanelli M.N., Dei S., Teodori E. (2019). Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers. In: XXVI National Meeting in Medicinal Chemistry, Milano, 16-19 luglio 2019, Società Chimica Italiana, pp. P79-P79.
Teodori E.; Contino M.; Riganti C.; Bartolucci G.; Braconi L.; Manetti D.; Romanelli M.N.; Trezza A.; Athanasios A.; Spiga O.; Perrone M.G.; Giampietro R.; Gazzano E.; Salerno M.; Colabufo N.A.; Dei S. (2019). Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 182, pp. 1-25, ISSN:0223-5234
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De Almeida, Carolina Vieira; Lulli, Matteo; di Pilato, Vincenzo; Schiavone, Nicola; Russo, Edda; Nannini, Giulia; Baldi, Simone; Borrelli, Rossella; Bartolucci, Gian Luca; Menicatti, Marta; Taddei, Antonio; Ringressi, Maria Novella; Niccolai, Elena; Prisco, Domenico; Rossolini, Gian Maria; Amedei, Amedeo (2019). Differential Responses of Colorectal Cancer Cell Lines to Enterococcus faecalis' Strains Isolated from Healthy Donors and Colorectal Cancer Patients. JOURNAL OF CLINICAL MEDICINE, vol. 8, pp. 388-403, ISSN:2077-0383
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Dugheri S.; Mucci N.; Cappelli G.; Bonari A.; Garzaro G.; Marrubini G.; Bartolucci G.; Campagna M.; Arcangeli G. (2019). Monitoring of air-dispersed formaldehyde and carbonyl compounds as vapors and adsorbed on particulate matter by denuder-filter sampling and gas chromatographic analysis. INTERNATIONAL JOURNAL OF ENVIRONMENTAL RESEARCH AND PUBLIC HEALTH, vol. 16, pp. 1969-1986, ISSN:1660-4601
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Martina Focardi, Antonella Bosco, Francesca Castiglione, Gian Luca Bartolucci, Barbara Gualco, Valentina Bugelli (2019). Abortion caused by intravaginal self-administration of misoprostol: a case report. REVISTA DE MEDICINA LEGALA, vol. 27, pp. 340-342, ISSN:1221-8618
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Marta Menicatti, Laura Moracci, Laura Braconi, Silvia Dei, Elisabetta Teodori, Gian Luca Bartolucci (2019). Tandem mass spectrometry with ion trap in the isomers resolution. In: 3rd MS NatMedDay-Massa 2019, Divisione di Spettrometria di Massa della Società Chimica Italiana, pp. 31-32.
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Marco Pallecchi, Gian Luca Bartolucci, Mario Maggi, Giovanna Danza (2019). A new method for the simultaneous quantification of different classes of steroid hormones and its application to the clinical routine. In: 37th Informal Meeting on Mass Spectrometry, Fiera di Primiero (TN), 05-08 Maggio 2019, 37th Informal Meeting on Mass Spectrometry organizing committee, pp. 84-84, ISBN:978-88-93495-59-2
Laura Moracci, Marta Menicatti, Silvia Dei, Elisabetta Teodori, Gian luca Bartolucci (2019). Isomers resolution of mult idrug resistence (MDR) inhibitors by LEDA algorithm: application in ion trap mass spectrometry. In: 37th Informal Meeting on Mass Spectrometry, Fiera di Primiero (TN), 05-08 Maggio 2019, 37th Informal Meeting on Mass Spectrometry organizing committee, pp. 80-80, ISBN:978-88-93495-59-2
Andrea Angeli; Lorenzo Di Cesare Mannelli; Carla Ghelardini; Thomas S. Peat; Gianluca Bartolucci; Marta Menicatti; Fabrizio Carta; Claudiu T. Supuran (2019). Benzensulfonamides bearing spyrohydantoin moieties act as potent inhibitors of human carbonic anhydrases {II} and {VII} and show neuropathic pain attenuating effects. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 177, pp. 188-197, ISSN:1768-3254
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Niccolò Chiaramontea, Silvia Bua, Andrea Angeli, Marta Ferraroni, Ilaria Picchioni, Gianluca Bartolucci, Laura Braconi, Silvia Dei, Elisabetta Teodori, Claudiu T. Supuran, Maria Novella Romanelli (2019). Sulfonamides incorporating piperazine bioisosteres as potent human carbonic anhydrase I, II, IV and IX inhibitors. BIOORGANIC CHEMISTRY, vol. 91, pp. 1-11, ISSN:0045-2068
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Falsini M.; Catarzi D.; Varano F.; Ceni C.; Dal Ben D.; Marucci G.; Buccioni M.; Volpini R.; Di Cesare Mannelli L.; Lucarini E.; Ghelardini C.; Bartolucci G.; Menicatti M.; Colotta V. (2019). Antioxidant-Conjugated 1,2,4-Triazolo[4,3-a]pyrazin-3-one Derivatives: Highly Potent and Selective Human A2A Adenosine Receptor Antagonists Possessing Protective Efficacy in Neuropathic Pain. JOURNAL OF MEDICINAL CHEMISTRY, vol. 62, pp. 8511-8531, ISSN:1520-4804
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Niccolai E.; Baldi S.; Ricci F.; Russo E.; Nannini G.; Menicatti M.; Poli G.; Taddei A.; Bartolucci G.; Calabro A.S.; Stingo F.C.; Amedei A. (2019). Evaluation and comparison of short chain fatty acids composition in gut diseases. WORLD JOURNAL OF GASTROENTEROLOGY, vol. 25, pp. 5543-5558, ISSN:1007-9327
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Marta Menicatti, Matilde Maggini, Francesco Caponi, Donato Squillaci, Laura Braconi, Silvia Dei , Elisabetta Teodori, Gian Luca Bartolucci (2018). Drug plasma stability study of multidrug resistance inhibitors by LC-MS/MS analysis. In: Divisione di Spettrometria di Massa della Società Chimica Italiana, Bologna, 11-12-2018, Divisione di Spettrometria di Massa della Società Chimica Italiana, pp. 22-22.
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Giovannoni, Maria Paola; Schepetkin, Igor A.; Quinn, Mark T.; Cantini, Niccolò; Crocetti, Letizia*; Guerrini, Gabriella; Iacovone, Antonella; Paoli, Paola; Rossi, Patrizia; Bartolucci, Gian Luca; Menicatti, Marta; Vergelli, Claudia (2018). Synthesis, biological evaluation, and molecular modelling studies of potent human neutrophil elastase (HNE) inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 1108-1124, ISSN:1475-6366
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Flamini, Riccardo; Menicatti, Marta; De Rosso, Mirko; Gardiman, Massimo; Mayr, Christine; Pallecchi, Marco; Danza, Giovanna; Bartolucci, Gian Luca* (2018). Combining liquid chromatography and tandem mass spectrometry approaches to the study of monoterpene glycosides (Aroma precursors) in wine grape. JOURNAL OF MASS SPECTROMETRY, vol. 53, pp. 792-800, ISSN:1076-5174
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Buğday, Nesrin; Küçükbay, F. Zehra; Küçükbay, Hasan*; Bua, Silvia; Bartolucci, Gian Luca; Leitans, Janis; Kazaks, Andris; Tars, Kaspars; Supuran, Claudiu T. (2018). Synthesis of novel dipeptide sulfonamide conjugates with effective carbonic anhydrase I, II, IX, and XII inhibitory properties. BIOORGANIC CHEMISTRY, vol. 81, pp. 311-318, ISSN:0045-2068
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Laura Braconi; Marta Menicatti; Silvia Dei; Elisabetta Teodori; Gian Luca Bartolucci (2018). ERMS EXPERIMENTS FOR RESOLUTION OF ISOBARIC COMPOUNDS: A CASE OF CIS/TRANS ISOMERISM. In: XXII International Mass Spectrometry Conference, Florence (Italy), August 26-31, 2018, 22nd IMSC SCIENTIFIC COMMITTEE, pp. 840-841, ISBN:9788890738852
Nocentini A, Trallori E, Singh S, Lomelino CL, Bartolucci G, Di Cesare Mannelli L, Ghelardini C, McKenna R, Gratteri P, Supuran CT (2018). 4-Hydroxy-3-nitro-5-ureido-benzenesulfonamides selectively target the tumor-associated carbonic anhydrase isoforms IX and XII showing hypoxia-enhanced anti-proliferative profiles.. JOURNAL OF MEDICINAL CHEMISTRY, vol. 61, pp. 10860-10874, ISSN:0022-2623
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Buonvicino, Daniela; Mazzola, Francesca; Zamporlini, Federica; Resta, Francesco; Ranieri, Giuseppe; Camaioni, Emidio; Muzzi, Mirko; Zecchi, Riccardo; Pieraccini, Giuseppe; Dölle, Christian; Calamante, Massimo; Bartolucci, Gianluca; Ziegler, Mathias; Stecca, Barbara; Raffaelli, Nadia; Chiarugi, Alberto* (2018). Identification of the Nicotinamide Salvage Pathway as a New Toxification Route for Antimetabolites. CELL CHEMICAL BIOLOGY, pp. 0-0, ISSN:2451-9456
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Menicatti, Marta; Pallecchi, Marco; Bua, Silvia; Vullo, Daniela; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Carta, Fabrizio; Supuran, Claudiu T.; Bartolucci, Gianluca* (2018). Resolution of co-eluting isomers of anti-inflammatory drugs conjugated to carbonic anhydrase inhibitors from plasma in liquid chromatography by energy-resolved tandem mass spectrometry. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 671-679, ISSN:1475-6366
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Akgul, Ozlem; Di Cesare Mannelli, Lorenzo; Vullo, Daniela; Angeli, Andrea; Ghelardini, Carla; Bartolucci, Gianluca; Altamimi, Abdulmalik Saleh Alfawaz; Scozzafava, Andrea; Supuran, Claudiu T; Carta, Fabrizio (2018). Discovery of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Management of Rheumatoid Arthritis. JOURNAL OF MEDICINAL CHEMISTRY, pp. 1-60, ISSN:0022-2623
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Menicatti Marta; Bartolucci Gian Luca (2018). Energy Resolved Tandem Mass Spectrometry experiments to resolve coeluting isomers. In: 36th Informal Meeting on Mass Spectrometry, Koszeg (Hungary), 6-9 May 2018, Organizing Committee of 36th Informal Meeting on Mass Spectrometry, pp. 52-52.
Gian Luca Bartolucci; Marco Pallecchi; Sebastiano Gozzo; Giovanna Danza (2018). SET UP OF A SIMPLE, FAST AND FLEXIBLE LC-MS/MS ID METHOD FOR THE SIMULTANEOUS DETERMINATION OF STEROIDS IN DIFFERENT BIOLOGICAL SAMPLES. In: XXII International Mass Spectrometry Conference, Florence, 26-31 Agosto 2018, 22nd IMSC SCIENTIFIC COMMITTEE, pp. 395-395, ISBN:9788890738852
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Silvia Bua; Marta Menicatti; Paola Gratteri; Alessio Nocentini; Claudiu T. Supuran; Gian Luca Bartolucci (2018). STABILITY STUDY IN PLASMA OF NOVEL ESTER-LINKED NSAID - CARBONIC ANHYDRASE INHIBITOR HYBRIDS. In: XXII International Mass Spectrometry Conference, Florence (Italy), August 26-31, 2018, 22nd IMSC SCIENTIFIC COMMITTEE, pp. 841-842, ISBN:9788890738852
Donato Squillaci; Marta Menicatti; Silvia Bua; Claudiu T. Supuran; Gian Luca Bartolucci (2018). APPLICATION OF LINEAR EQUATIONS DECONVOLUTION ANALYSIS (LEDA) ALGORITHM IN ION TRAP MASS SPECTROMETRY: RESOLUTION OF ISOMERIC PAIRS OF CARBONIC ANHYDRASE AND CYCLOOXYGENASE HYBRIDS INHIBITORS. In: XXII International Mass Spectrometry Conference, Florence (Italy), August 26-31, 2018, 22nd IMSC SCIENTIFIC COMMITTEE, pp. 846-847, ISBN:9788890738852
Silvia, Dei; Marcella, Coronnello; Gian Luca Bartolucci, ; Dina, Manetti; Maria Novella Romanelli, ; Chatchanok, Udomtanakunchai; Milena, Salerno; Elisabetta, Teodori (2018). Design and synthesis of new potent N,N-bis(arylalkyl)piperazine derivatives as multidrug resistance (MDR) reversing agents. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 147, pp. 7-20, ISSN:0223-5234
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Niccolò Chiaramonte, Silvia Bua, Marta Ferraroni, Alessio Nocentini, Alessandro Bonardi, Gian Luca Bartolucci, Maria Concetta Durante, Laura Lucarini, Donata Chiapponi, Silvia Dei, Dina Manetti, Elisabetta Teodori, Paola Gratteri, Emanuela Masini, Claudiu T. Supuran, Maria Novella Romanelli (2018). 2-Benzylpiperazine: a new scaffold for potent human Carbonic Anhydrase inhibitors. Synthesis, enzyme inhibition, enantioselectivity, computational and crystallographic studies and in vivo activity for a new class of intraocular pressure lowering agents.. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 151, pp. 363-375, ISSN:1768-3254
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Martino, Maria Vittoria; Guandalini, Luca; Di Cesare Mannelli, Lorenzo; Menicatti, Marta; Bartolucci, Gianluca; Dei, Silvia; Manetti, Dina; Teodori, Elisabetta; Ghelardini, Carla; Romanelli, Maria Novella (2017). Piperazines as nootropic agents: New derivatives of the potent cognition-enhancer DM235 carrying hydrophilic substituents. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 25, pp. 1795-1803, ISSN:0968-0896
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Bua, Silvia; Di Cesare Mannelli, Lorenzo; Vullo, Daniela; Ghelardini, Carla; Bartolucci, Gianluca; Scozzafava, Andrea; Supuran, Claudiu T; Carta, Fabrizio (2017). Design and Synthesis of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Treatment of Rheumatoid Arthritis. JOURNAL OF MEDICINAL CHEMISTRY, vol. 60, pp. 1159-1170, ISSN:0022-2623
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Angeli, Andrea; Carta, Fabrizio; Bartolucci, Gian Luca; Supuran, Claudiu T.* (2017). Synthesis of novel acyl selenoureido benzensulfonamides as carbonic anhydrase I, II, VII and IX inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 25, pp. 3567-3573, ISSN:0968-0896
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Teodori, Elisabetta; Dei, Silvia; Bartolucci, Gianluca; Perrone, Maria Grazia; Manetti, Dina; Romanelli, Maria Novella; Contino, Marialessandra; Colabufo, Nicola Antonio (2017). Structure-Activity Relationship Studies on 6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline Derivatives as Multidrug Resistance Reversers. CHEMMEDCHEM, vol. 12, pp. 1369-1379, ISSN:1860-7179
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Flamini, Riccardo; De Rosso, Mirko; Gardiman, Massimo; Mayr, Christine; Danza, Giovanna; Menicatti, Marta; Bartolucci, Gian Luca (2017). New LC-MS/MS approaches to study monoterpene glycosides (aroma precursors) in grape. In: 5th MS Food Day, Bologna, 11-13 Ottobre 2017, 9788890738838, pp. 249-251, ISBN:9788890738838
Berrino, Emanuela; Bua, Silvia; Mori, Mattia; Botta, Maurizio; Murthy, Vallabhaneni S.; Vijayakumar, Vijayaparthasarathi; Tamboli, Yasinalli; Bartolucci, Gianluca; Mugelli, Alessandro; Cerbai, Elisabetta; Supuran, Claudiu T.; Carta, Fabrizio (2017). Novel sulfamide-containing compounds as selective carbonic anhydrase i inhibitors. MOLECULES, vol. 22, pp. 1049-1065, ISSN:1420-3049
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Angeli, Andrea; Tanini, Damiano; Peat, Thomas S. ; Di Cesare Mannelli,Lorenzo; Bartolucci, Gian Luca; Capperucci, Antonella; Ghelardini, Carla; Supuran, Claudiu T.; and Carta, Fabrizio (2017). Discovery of New Selenoureido Analogues of 4-(4-Fluorophenylureido)benzenesulfonamide as Carbonic Anhydrase Inhibitors. ACS MEDICINAL CHEMISTRY LETTERS, vol. 8, pp. 963-968, ISSN:1948-5875
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Crocetti, Letizia; Bartolucci Gian Luca, ; Cilibrizzi, Agostino; Giovannoni, Maria Paola; Guerrini, Gabriella; Iacovone, Antonella; Menicatti, Marta; Schepetkin, Igor A; Khlebnikov, Andrei I; Quinn, Mark T; Vergelli, Claudia (2017). Synthesis and analytical characterization of new thiazol-2-(3H)-ones as human neutrophil elastase (HNE) inhibitors. CHEMISTRY CENTRAL JOURNAL, vol. 11, pp. 127-141, ISSN:1752-153X
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Nocentini, Alessio; Bua, Silvia; Lomelino, Carrie L.; Mckenna, Robert; Menicatti, Marta; Bartolucci, Gianluca; Tenci, Barbara; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Gratteri, Paola; Supuran, Claudiu T. (2017). Discovery of New Sulfonamide Carbonic Anhydrase IX Inhibitors Incorporating Nitrogenous Bases. ACS MEDICINAL CHEMISTRY LETTERS, vol. 8, pp. 1314-1319, ISSN:1948-5875
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Coppini, Raffaele; Mazzoni, Luca; Ferrantini, Cecilia; Gentile, Francesca; Pioner, Josè Manuel; Laurino, Annunziatina; Santini, Lorenzo; Bargelli, Valentina; Rotellini, Matteo; Bartolucci, Gian Luca; Crocini, Claudia; Sacconi, Leonardo; Tesi, Chiara; Belardinelli, Luiz; Tardiff, Jil; Mugelli, Alessandro; Olivotto, Iacopo; Cerbai, Elisabetta; Poggesi, Corrado (2017). Ranolazine prevents phenotype development in a mouse model of hypertrophic cardiomyopathy. CIRCULATION. HEART FAILURE, vol. 10, pp. 10:e003565-10:e003565, ISSN:1941-3289
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Teodori, Elisabetta; Dei, Silvia; Coronnello, Marcella; Floriddia, Elisa; Bartolucci, Gianluca; Manetti, Dina; Romanelli, Maria Novella; Santo Domingo Porqueras, Diego; Salerno, Milena (2017). N-alkanol-N-cyclohexanol amine aryl esters: Multidrug resistance (MDR) reversing agents with high potency and efficacy. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 127, pp. 586-598, ISSN:0223-5234
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Menicatti, Marta; Guandalini, Luca; Dei, Silvia; Floriddia, Elisa; Teodori, Elisabetta; Traldi, Piero; Bartolucci Gian Luca, (2017). LEDA TOOL: A POST-PROCESSING ALGORITHM TO RESOLVE ISOBARIC COMPOUDS MIXTURES. In: 35th Informal Meeting on Mass spectrometry, Aussois (France), 7-11 Maggio 2017, CNRS, pp. 52-53.
Paoli, Paola ; Rossi, Patrizia; Macedi, Eleonora; Ienco, Andrea; Chelazzi, Laura; Bartolucci, Gian Luca; Bruni, Bruno (2016). Similar but Different: The Case of Metoprolol Tartrate and Succinate Salts. CRYSTAL GROWTH & DESIGN, vol. 16, pp. 789-799, ISSN:1528-7483
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Bartolucci, G.; Menicatti, M.; Guandalini, L.; S, . DEI; Floriddia, E.; Teodori, E. (2016). Linear deconvolution of LC-MS/MS analysis for resolution of isobaric compounds: a case of cis/trans isomerism. In: XXIV National Meeting in Medicinal Chemistry, Perugia, 11-14 settembre 2016, Scoietà Chimica Italiana, pp. PC-157-PC-157.
Menicatti, M.; Guandalini, L.; S, . DEI; Floriddia, E.; Teodori, E.; Traldi, P.; Bartolucci, G. (2016). Resolving mixtures of isobaric compounds using Energy resolved MS/MS experiments and LEDA post-processing algorithm tool. In: International Conference MASSA 2016, Roma, 6-8 settembre 2016, Istituto Superiore di Sanità, vol. 16 C4, pp. 98-98.
Menicatti, M.; Guandalini, L.; Dei, S.; Floriddia, E.; Teodori, E.; Traldi, P.; Bartolucci, G. (2016). Energy resolved MS/MS experiments for resolution of isobaric compounds: a case of cis/trans isomerism. In: 34th IMMS 2016 - 34th Informal Meeting on Mass Spectrometry, Fiera di Primiero (TN), 15-18 maggio 2016, SGEditoriali, pp. 78-79, ISBN:978-88-89884-31-7
Betti, M.; Colotta, V.; Varano, F.; Falsini, M.; Varani, K.; Vincenzi, F.; Dal Ben, D.; Di Cesare Mannelli, L.; Zanardelli, M.; Bartolucci, G.; Menicatti, M.; Catarzi, D. (2016). Aminopyridine-3,5-carbonitrile core for the design of new adenosine receptor agonists: structural exploration to target the A1 subtype. In: XXIV National Meeting on Medicinal Chemistry, 10th Young Medicinal Chemists’ Symposium, 11-14 settembre 2016, Perugia., d, pp. 108-108.
Menicatti, Marta; Guandalini, Luca; Dei, Silvia; Floriddia, Elisa; Teodori, Elisabetta; Traldi, Piero; Bartolucci, Gian Luca (2016). Resolving mixtures of isobaric compounds using energy resolved MS/MS experiments and the LEDA post processing algorithm tool. In: 3th MS ENVI-Day, Livorno, 26-28 Settembre 2016, 9788894173123, pp. 45-45, ISBN:9788894173123
Angeli, A; Peat, T.S.; Bartolucci, G.; Nocentini, A.; Supuran, C.T.; Carta, F. (2016). Intramolecular oxidative deselenization of acylselenoureas: a facile synthesis of benzoxazole amides and carbonic anhydrase inhibitors. ORGANIC & BIOMOLECULAR CHEMISTRY, vol. 14, pp. 11353-11356, ISSN:1477-0520
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Menicatti, Marta; Guandalini, Luca; Dei, Silvia; Floriddia, Elisa; Teodori, Elisabetta; Traldi, Pietro; Bartolucci, Gianluca (2016). The power of energy-resolved tandem mass spectrometry experiments for resolution of isomers: the case of drug plasma stability investigation of multidrug resistance inhibitors. RAPID COMMUNICATIONS IN MASS SPECTROMETRY, vol. 30, pp. 423-432, ISSN:0951-4198
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Nocentini, Alessio; Vullo, Daniela; Bartolucci, Gianluca; Supuran, Claudiu T (2016). N-Nitrosulfonamides: A new chemotype for carbonic anhydrase inhibition. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 24, pp. 3612-3617, ISSN:0968-0896
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Menicatti, Marta; Guandalini, Luca; Dei, Silvia; Floriddia, Elisa; Teodori, Elisabetta; Traldi, Pietro; Bartolucci, Gianluca (2016). Energy resolved tandem mass spectrometry experiments for resolution of isobaric compounds: a case of cis/trans isomerism. EUROPEAN JOURNAL OF MASS SPECTROMETRY, vol. 22, pp. 235-243, ISSN:1469-0667
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Teodori, Elisabetta; Dei, Silvia; Floriddia, Elisa; Coronnello, Marcella; Bartolucci, Gianluca; Manetti, Dina; Maria Novella Romanelli, Salerno, Milena (2015). Aminoarylesters as multidrug resistance (MDR) reverting agents endowed with high potency and efficacy. In: IXth Joint Meeting in Medicinal Chemistry, Atene, 7-10 giugno 2015, Hellenic Society of Medicinal Chemistry, pp. O11-O11.
Guandalini, Luca; Martino, Maria Vittoria; Di Cesare Mannelli, Lorenzo; Bartolucci, Gianluca; Melani, Fabrizio; Malik, Ruchi; Dei, Silvia; Floriddia, Elisa; Manetti, Dina; Orlandi, Francesca; Teodori, Elisabetta; Ghelardini, Carla; Romanelli, Maria Novella (2015). Substituted piperazines as nootropic agents: 2- or 3-phenyl derivatives structurally related to the cognition-enhancer DM235. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 25, pp. 1700-1704, ISSN:0960-894X
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Menicatti, M.; Guandalini, L.; Dei, S.; Floriddia, E.; Teodori, E.; Traldi, P.; Bartolucci, G. (2015). Multidrug resistance inhibitors in plasma samples: the power of LC-energy resolved MS/MS methods for stability investigation. In: Bioanalitica 2015: Nuovi approcci bioanalitici per la determinazione di sostanze ad attività biologica, farmaceutica e nutraceutica, Firenze, 26 giugno 2015, Società Chimica Italiana Divisione di Chimica Analitica, pp. 16-16.
Nocentini, Alessio; Carta, Fabrizio; Ceruso, Mariangela; Bartolucci, Gianluca; Supuran, Claudiu T. (2015). Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 23, pp. 6955-6966, ISSN:0968-0896
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Martino, M. V.; DI CESARE MANNELLI, L. ; Bartolucci, G.; S, . DEI; Manetti, D.; Ghelardini, C.; Teodori, E.; Romanelli, M. N. (2015). 2- or 3-Substituted piperazines as nootropic agents: carbethoxy and hydroxymethyl analogues of the cognition-enhancer DM235. In: XXIII National Meeting on Medicinal Chemistry and 9th Young Medicinal Chemists Symposium (XXIII NMMC – 9th NPCF), Salerno, 6-9 settembre 2015, Edizioni Ziino, pp. 136-136.
Menicatti, Marta; Bartolucci, Gian Luca (2015). CHINESE ASTRAGALUS ROOT EXTRACTS: A CASE STUDY. In: 1st MS-NatMed-Day Natural Molecules and Molecular Complexes: characterization and biomedical effects, Sansepolcro (AR), 21-22 Settembre 2015, Aboca, pp. 28-28.
Sara Marchiani; Linda Vignozzi; Sandra Filippi; Bruna Gurrieri; Paolo Comeglio; Annamaria Morelli; Giovanna Danza; Gianluca Bartolucci; Mario Maggi; Elisabetta Baldi (2015). METABOLIC SYNDROME-ASSOCIATED SPERM ALTERATIONS IN AN EXPERIMENTAL RABBIT MODEL: RELATION WITH METABOLIC PROFILE, TESTIS AND EPIDIDYMIS GENE EXPRESSION AND EFFECT OF TAMOXIFEN TREATMENT. MOLECULAR AND CELLULAR ENDOCRINOLOGY, vol. 401, pp. 12-24, ISSN:0303-7207
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Di Cesare Mannelli, Lorenzo; Zanardelli, Matteo; Bartolucci, Gianluca; Karioti, Anastasia; Bilia, Anna Rita; Vannacci, Alfredo; Mugelli, Alessandro; Ghelardini, Carla (2015). In Vitro Evidence for the Use of Astragali Radix Extracts as Adjuvant against Oxaliplatin-Induced Neurotoxicity. PLANTA MEDICA, vol. 81, pp. 1045-1055, ISSN:0032-0943
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Guandalini, Luca; Soldani, Giacomo; Rosi, Luca; Calamai, Luca; Bartolucci, Gianluca (2015). A methodological approach to the selection of liquid reagents for chemical ionization ion trap-gas chromatography mass spectrometry: A case study of GBL and 1,4-BD. INTERNATIONAL JOURNAL OF MASS SPECTROMETRY, vol. 388, pp. 34-39, ISSN:1387-3806
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Marta Menicatti; Luca Guandalini; Silvia Dei; Elisa Floriddia; Elisabetta Teodori; Gian Luca Bartolucci (2014). Stability in biological fluids by LC-MS/MS analysis of multidrug resistance inhibitors. In: 8° MS-Pharmaday, Sansepolcro (AR), 11-13 giugno 2014, Società Chimica Italiana Divisioni di Chimica Farmaceutica e di Spettrometria di Massa, pp. 36-37.
Silvia Dei; Marcella Coronnello; Elisa Floriddia; Gianluca Bartolucci; Cristina Bellucci; Luca Guandalini; Dina Manetti; Maria Novella Romanelli; Milena Salerno; Ivan Bello; Enrico Mini; Elisabetta Teodori (2014). Multidrug resistance (MDR) reversers: High activity and efficacy in a series of asymmetrical N,N-bis(alkanol)amine aryl esters. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 87, pp. 398-412, ISSN:0223-5234
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I. Maida; M. Fondi; M.C. Papaleo; E. Perrin; V. Orlandini; G. Emiliani; D. de Pascale; E. Parrilli; M.L. Tutino; L. Michaud; A. Lo Giudice; R. Romoli; G. Bartolucci; R. Fani (2014). Phenotypic and genomic characterization of the Antarctic bacterium Gillisia sp. CAL575, a producer of antimicrobial compounds. EXTREMOPHILES, vol. 18, pp. 35-49, ISSN:1431-0651
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Menicatti, Marta; Bartolucci, Gian Luca (2014). Oli essenziali: analisi e caratterizzazione mediante GC-MS e GC-MS/MS. In: Il Congresso Nazionale per la ricerca sugli oli essenziali, Terni, 14-16 Novembre 2014, Istituto Superiore di Sanità, pp. 18-18.
R. Romoli; M.C. Papaleo; D. De Pascale; M.L. Tutino; L. Michaud; A. LoGiudice; R. Fani; G. Bartolucci (2014). GC-MS Volatolomic Approach to Study the Antimicrobial Activity of the Antarctic Bacterium Pseudoalteromonas sp. TB41. METABOLOMICS, vol. 10, pp. 42-51, ISSN:1573-3882
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L. Rosi; P. Frediani; G. Bartolucci (2013). Determination of GHB and its precursors (GBL and 1,4-BD) in dietary supplements through the synthesis of their isotopologues and analysis by GC-MS method. JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, vol. 74, pp. 31-38, ISSN:0731-7085
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Gustavo Ayala;Matteo Morello;Anna Frolov;Sungyong You;Rile Li;Fabiana Rosati;Gianluca Bartolucci;Giovanna Danza;Rosalyn M Adam;Timothy C Thompson;Michael P Lisanti;Michael R Freeman;Dolores Di Vizio (2013). Loss of caveolin-1 in prostate cancer stroma correlates with reduced relapse-free survival and is functionally relevant to tumour progression. JOURNAL OF PATHOLOGY, vol. 231, pp. 77-87, ISSN:0022-3417
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A. Cilibrizzi; L. Crocetti; M.P. Giovannoni; A. Graziano; C. Vergelli; G. Bartolucci; G. Soldani; M.T. Quinn; I.A. Schepetkin; C. Faggi. (2013). Synthesis, HPLC enantioresolution and X-ray analysis of a new series of C5-methyl pyridazines as N-formyl peptide receptor (FPR) agonists. CHIRALITY, vol. 25, pp. 400-408, ISSN:0899-0042
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Enrica Droghetti; Francesco P. Nicoletti; Luca Guandalini; Gianluca Bartolucci; Giulietta Smulevich (2013). SERS detection of benzophenones on viologen functionalized Ag nanoparticles: application to breakfast cereals. JOURNAL OF RAMAN SPECTROSCOPY, vol. 44, pp. 1428-1434, ISSN:0377-0486
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M.C. Papaleo; R. Romoli; G. Bartolucci; I. Maida; E. Perrin; M. Fondi; V. Orlandini; A. Mengoni; G. Emiliani; M. L. Tutino; E. Parrilli; D. de Pascale; L. Michaud; A. Lo Giudice; R. Fani (2013). Bioactive volatile organic compounds from Antarctic (sponges) bacteria. NEW BIOTECHNOLOGY, vol. 30, pp. 824-838, ISSN:1871-6784
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I. Maida; M.C. Papaleo; E. Perrin; M. Fondi; V. Orlandini; G. Emiliani; R. Romoli; G. Bartolucci; M.L. Tutino; G. Parrilli; D. De Pascale; L. Michaud; A. Lo Giudice; R. Fani (2013). Antarctic bacteria as producers of antibiotic volatile compounds inhibiting cystic fibrosis pathogens. JOURNAL OF CYSTIC FIBROSIS, pp. 573-573, ISSN:1569-1993
S. Benemei;E. Gallo;E. Giocaliere;G. Bartolucci;F. Menniti-Ippolito;F. Firenzuoli;A. Mugelli;A. Vannacci (2013). It's time for new rules on vitamin D food supplements. BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, vol. 76, pp. 825-826, ISSN:0306-5251
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L. Guandalini; M. Balliu; C. Cellai; M.V. Martino; A. Nebbioso; C. Mercurio; V. Carafa; G. Bartolucci; S. Dei; D. Manetti; E. Teodori; S. Scapecchi; L. Altucci; F. Paoletti; M.N. Romanelli (2013). Design, synthesis and preliminary evaluation of a series of histone deacetylase inhibitors carrying a benzodiazepine ring. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 66, pp. 56-68, ISSN:0223-5234
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M.C. Papaleo; M. Fondi; I. Maida; E. Perrin; A. Lo Giudice; L. Michaud; S. Mangano; G. Bartolucci; R. Romoli; R. Fani (2012). Sponge-associated microbial Antarctic communities exhibiting antimicrobial activity against Burkholderia cepacia complex bacteria. BIOTECHNOLOGY ADVANCES, vol. 30, pp. 272-293, ISSN:0734-9750
M.C. Papaleo; I. Maida; E. Perrin; M. Fondi; G. Emiliani; R. Romoli; G. Bartolucci; M.L. Tutino; D. de Pascale; L. Michaud; A. Lo Giudice; R. Fani (2012). Antarctic sponge bacteria: a new potential source of natural antibiotic compounds. In: Marine Microbiology and Biotechnology 2012 - Biodiscovery, Biodiversity & Bioremediation, Cork (Ireland), 14-16 novembre, pp. 13-13.
M.C. Papaleo; I. Maida; E. Perrin; M. Fondi; D. Conti; R. Romoli; G. Bartolucci; M.L. Tutino; G. Parrilli; D. de Pascale; L. Michaud; A. Lo Giudice; R. Fani (2012). Volatile organic compounds (VOCs) from Antarctic sponges-associated bacteria inhibiting Cystic Fibrosis pathogens. In: 12th FISV Congress, Roma, 24-27 settembre, pp. 70-70.
Calamai, L.; Villanelli, F.; Bartolucci, G.; Pieraccini, G.; Moneti, G.; (2012). Sample Preparation for Direct MS Analysis of Food. In: Pawliszyn, J.; Mondello, L.; Dugo, P.. Comprehensive Sampling and Sample Preparation, pp. 535-557, OXFORD: Elsevier Science Limited, ISBN:9780123813732.
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A. Cilibrizzi; I.A. Schepetkin; G. Bartolucci; L. Crocetti; V. Dal Piaz; M.P. Giovannoni; A. Graziano; L. N. Kirpotina; M.T. Quinn; C. Vergelli (2012). Synthesis, enantioresolution and activity profile of chiral 6-methyl-2,4-disubstituted pyridazin-3(2H)-ones as potent N-formyl peptide receptor agonists.. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 20, pp. 3781-3792, ISSN:0968-0896
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Rosi, Luca; Frediani, Piero; Soldani, Giacomo; Bartolucci, Gianluca (2012). GHB in dietary supplements. In: 7th MS-PharmaDay, Santa Palomba (Roma), 22-24 Ottobre 2012, Edizioni Nuova Cultura, pp. 39-39, ISBN:9788861348905
Raffaelli, Andrea; Giorgi, Gianluca; Moneti, Gloriano; Bartolucci, Gianluca; Pieraccini, Giuseppe (2012). Corso di formazione specialistica. L'accoppiamento cromatografia liquida ad alte prestazioni-spettrometria di massa (HPLC-MS): principi e applicazioni. In: Raffaelli, Andrea; Giorgi, Gianluca; Moneti, Gloriano; Bartolucci, Gianluca; Pieraccini, Giuseppe. L'accoppiamento cromatografia liquida ad alte prestazioni-spettrometria di massa (HPLC-MS): principi e applicazioni, pp. 1-179, Roma: Edizioni Nuova Cultura, ISBN:9788861349711.
M.C. Papaleo; I. Maida; E. Perrin; M. Fondi; A. LoGiudice; L. Michaud; M.L. Tutino; D. de Pascale; R. Romoli; G. Bartolucci; R. Fani (2011). Production of VOCs by Antarctic bacteria: new potential antibiotic compounds vs Burkholderia cepacia. In: Bageco 2011, Corfù (Grecia), 29 maggio - 2 giugno, pp. 222-222.
L. Calamai; F. Villanelli; G. Bartolucci (2011). L'analisi dei contaminanti organici nelle acque. In: M. Gennari, M Trevisan. Gestione e qualità delle acque. Origini, dinamiche, previsioni, mutamenti sociali, pp. 87-119, Ozzano dell'Emilia (BO): Alberto Perdisa, ISBN:9788883724947.
G. Bartolucci; E. Giocaliere; F. Boscaro; A. Vannacci; E. Gallo; G. Pieraccini; G. Moneti (2011). Vitamin D3 quantification in a cod liver oil-based supplement. JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, vol. 55, pp. 64-70, ISSN:0731-7085
Enrica Droghetti; Gian Luca Bartolucci; Claudia Focardi; Massimo Bambagiotti-Alberti; Mila Nocentini; Giulietta Smulevich (2011). Development and validation of a quantitative spectrophotometric method to detect the amount of carbon monoxide in treated tuna fish.. FOOD CHEMISTRY, vol. 128, pp. 1143-1151, ISSN:0308-8146
DOI
Romoli, Riccardo; Bartolucci, Gianluca; Papaleo, Maria Cristiana; Fani, Renato (2011). Characterization of volatile profile in antartic bacteria using SPME-GC-MS. In: 29th Informal Meeting on Mass Spectrometry, Fiera di Primiero (TN), 15-19 Maggio 2011, SGEditoriali Padova, pp. 57-57, ISBN:9788889884195
M.C. Papaleo; I. Maida; E. Perrin; M. Fondi; A. Lo Giudice; L. Michaud; M.L. Tutino; D. de Pascale; R. Romoli; G. Bartolucci; R. Fani (2011). Volatile compounds (VCs) by Antarctic bacteria: new potential antibiotics vs Burkholderia cepacia. In: 29th National Meeting SIMGBM, Pisa (Italy), 21-23 Settembre, pp. 155-155.
F. Rosati;N. Sturli;M. C. Cungi;M. Morello;F. Villanelli;G. Bartolucci;C. Finocchi;A. Peri;M. Serio;G. Danza (2011). Gonadotropin-releasing hormone modulates cholesterol synthesis and steroidogenesis in SH-SY5Y cells.. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, vol. 124, pp. 77-83, ISSN:0960-0760
DOI
Accesso ONLINE all'editore
Villanelli, Fabio; Calamai, Luca; Bartolucci, Gian Luca (2011). A new fast method for GC-MS/MS analysis of organotin compounds on micro samples of whole blood. In: 29th Informal meeting on mass spectrometry, Fiera di Primiero (TN), 15-19 Maggio 2011, SGEditoriali, pp. 62-62, ISBN:9788889884195
R. Romoli; M.C. Papaleo; D. de Pascale; M.L. Tutino; L. Michaud; A. LoGiudice; R. Fani; G.L. Bartolucci (2011). Characterization of the volatile profile of Antarctic bacteria by using solid-phase microextraction-gas chromatography-mass spectrometry. JOURNAL OF MASS SPECTROMETRY, vol. 46, pp. 1051-1059, ISSN:1076-5174
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E. Martini; L. Di Cesare Mannelli; G. Bartolucci; C. Bertucci; S. Dei; C. Ghelardini; L. Guandalini; D. Manetti; S. Scapecchi; E. Teodori; M. N. Romanelli (2011). Synthesis and Biological Evaluation of 3,7-Diazabicyclo[4.3.0]2 nonan-8-ones as Potential Nootropic and Analgesic Drugs. JOURNAL OF MEDICINAL CHEMISTRY, vol. 54, pp. 2512-2516, ISSN:0022-2623
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Accesso ONLINE all'editore
M.C. Papaleo; I. Maida; E. Perrin; M. Fondi; A. Lo Giudice; S. Mangano; L. Michaud; M.L. Tutino; D. de Pascale; G. Bartolucci; R. Fani (2011). New potential antibiotic sources for Burkholderia cepacia. In: 15th Annual Meeting - International Burkholderia cepacia Working Group, Prague - Repubblica Ceca, Aprile, pp. A32-A32.
M.C. Papaleo; I. Maida; E. Perrin; M. Fondi; A. Lo Giudice; S. Mangano; L. Michaud; M. L. Tutino; D. de Pascale; G. Bartolucci ; R. Fani (2011). New potential antibiotic sources for Burkholderia cepacia. JOURNAL OF CYSTIC FIBROSIS, vol. 10, Supplement 1, pp. S25-S25, ISSN:1569-1993
S.A.Coran; G.Bartolucci;M.Bambagiotti-Alberti (2011). Selective determination of aloin in different matrices by HPTLC densitometry in fluorescence mode. JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, vol. 54, pp. 422-425, ISSN:0731-7085
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B. Bruni; S. A. Coran; G. Bartolucci; M. Di Vaira (2010). 4-Amino-N-(3-methoxypyrazin-2-yl)benzenesulfonamide. ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, vol. 66, pp. o2663-o2663, ISSN:1600-5368
DOI
G. Bartolucci; E. Droghetti; C. Focardi; M. Bambagiotti-Alberti; M. Nocentini; G. Smulevich (2010). High throughput headspace GC-MS quantitative method to measure the amount of carbon monoxide treated tuna fish.. JOURNAL OF MASS SPECTROMETRY, vol. 45, pp. 1041-1045, ISSN:1076-5174
Bartolucci, Gian Luca; Droghetti, Enrica; Focardi, Claudia; Bambagiotti Alberti, Massimo; Nocentini, Mila; Smulevich, Giulietta (2009). Routinary and automated HS-GC-MS quantitative method to measure the amount of carbon monoxide in fraudulently treated tuna fish. In: 1° MS Food-Day, Parma, 2-3 Dicembre 2009, Società Chimica Italiana Divisione Spettrometria di Massa, pp. 41-41.
G.Bartolucci; B.Bruni; S.A.Coran; M.Di Vaira (2009). 4-(3-Methylanilino)-N-[N-(1-methylethyl)carbamoyl]pyridinium-3-sulfonamidate (torasemide T-N): a low temperature redetermination. ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, vol. E65, pp. o972-o973, ISSN:1600-5368
DOI
L.CALAMAI; F.VILLANELLI; G. BARTOLUCCI (2009). Metodi multiresiduali di analisi dei pesticidi. In: Convegno GRIFA, Firenze, Italy, 26 27-novembre, pp. 1-1.
G. Bartolucci; B. Bruni; S. A. Coran; M. Di Vaira (2009). {2-Hydroxy-3-[4-(2-methoxyethyl)-phenoxy]propyl}isopropylammonium hemisuccinate. ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, vol. E65, pp. 1364-1365, ISSN:1600-5368
DOI
Massimo Bambagiotti-Alberti; Gianluca Bartolucci; Bruno Bruni; Silvia A. Coran; Massimo Di Vaira (2009). Physico-chemical and structural characterization of diacerhein. JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, vol. 49, pp. 1065-1069, ISSN:0731-7085
DOI
G.Bartolucci; B.Bruni; S.A.Coran; M.Di Vaira (2009). 4-(3-Methylanilino)-N-[N-(1-methylethyl)carbamoyl]pyridinium-3-sulfonamidate (torasemide) methanol 0.25-solvate 0.25-hydrate. ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, vol. E65, pp. o970-o971, ISSN:1600-5368
DOI
M. BAMBAGIOTTI ALBERTI; G. BARTOLUCCI; B. BRUNI; S. CORAN; M. DI VAIRA (2008). 3-Methyl-1,4-dioxo-1,4-dihydronaphthalen-2-yl 4-aminobenzoate. ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, vol. E64, pp. o718-0718, ISSN:1600-5368
DOI
G. Pieraccini; S. Furlanetto; S. Orlandini; G. Bartolucci; I. Giannini; S. Pinzauti; G. Moneti (2008). Identification and determination of mainstream and sidestream smoke components in different brands and types of cigarettes by means of solid-phase microextraction-gas cromatography-mass spectrometry.. JOURNAL OF CHROMATOGRAPHY A, vol. 1180, pp. 138-150, ISSN:0021-9673
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M.PACENTI; S. DUGHERI; F. VILLANELLI; G. BARTOLUCCI; L. CALAMAI; P. BOCCALON; G. ARCANGELI; F. VECCHIONE; P.ALESSI; I. KIKIC; V. CUPELLI (2008). Determination of organic acids in urine by solid phase microextraction and gas chromatography-ion trap tandem mass spectrometry previous "in sample" derivatisation with trimethyloxonium tetrafluoroborate. BIOMEDICAL CHROMATOGRAPHY, vol. 22, pp. 1155-1163, ISSN:0269-3879
DOI
Silvia A Coran; Gianluca Bartolucci; Massimo Bambagiotti-Alberti (2008). Validation of a reversed phase high performance thin layer chromatographic-densitometric method for secoisolariciresinol diglucoside determination in flaxseed.. JOURNAL OF CHROMATOGRAPHY A, vol. 1207, pp. 155-159, ISSN:0021-9673
DOI
Manzini, Barbara; Parenti, Gabriele; Bartolucci, Gian Luca; Danza, Giovanna; Moneti, Gloriano; Pieraccini, Giuseppe; Leone, Ilenia; Serio, Mario; Mannelli, Massimo (2008). Measurement of Cortisol to Cortisone ratio in human urine and saliva by LC-MS/MS. In: 1st French-Italian Conference on Mass Spectrometry. Fundamentals and applications of mass spectrometry, Siena, 30 Giugno-4 Luglio 2008, Tipografia Senese, pp. 115-115.
M. Bambagiotti Alberti; G. Bartolucci; B. Bruni; S. A. Coran; M. Di Vaira (2008). Diisopropyl[2-[2-(2-oxopyrrolidin-1-yl)acetamido]ethyl]ammonium hydrogen sulfate. ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, vol. 64, pp. o1160-o1160, ISSN:1600-5368
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P.Frediani; L.Rosi; M.Frediani; G.Bartolucci; M. Bambagiotti Alberti (2007). A CONVENIENT ROUTE TO THE SYNTHESIS OF ISOTOPOMERIC DIHYDRO-2(3H)FURANONES. JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, vol. 55, pp. 3877-3883, ISSN:0021-8561
DOI
G. BARTOLUCCI; B. BRUNI; M. DI VAIRA; V. GIANNELLINI (2007). 2-Butyl-4-oxo-3-([2'-(1H-tetrazol-5-yl)biphenyl-4-yl]methyl)-3-aza-1-azoniaspiro[4.4]non-1-ene chloride 1.69-hydrate (irbesartan hydrochloride 1.69-hydrate). ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, vol. 63, pp. o1529-o1531, ISSN:1600-5368
DOI
R. RECENTI; G. LEONE; L. SIMI; M. ORFEI; P. PINZANI; G. PIERACCINI; G. MONETI; CAROSSINO A.M.; A. FRANCHI; BARTOLUCCI G; CARBONELL SALA S; GINANNESCHI M. ; TANINI A.; BRANDI M.L (2007). Clodronate acts on human osteoclastic cell proliferation, differentiation and function in a bioreversible manner. CLINICAL CASES IN MINERAL AND BONE METABOLISM, vol. 4, pp. 146-155, ISSN:1724-8914
M. BAMBAGIOTTI ALBERTI; G. BARTOLUCCI; B. BRUNI; M. DI VAIRA; M. PASSAPONTI (2007). Disodium 2,2'-dithiobis(ethanesulfonate) trihydrate (dimesna trihydrate). ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, vol. 63, pp. m1948-m1948, ISSN:1600-5368
DOI
Bartolucci Gian Luca, Del Fante, Daniele; Mascelloni, Elena; Bambagiotti Alberti, Massimo (2006). Determinazione in matrici vegetali del Secoisolariciresinolo diglucoside, precursore in vivo dei lignani ad azione estrogenica. In: SCI2006 XXII Congresso nazionale della Società Chimica Italiana, Firenze, 10-15 Settembre 2006, Società Chimica Italiana, pp. 413-413.
Pesamosca Facco, Elizete Maria; Pieraccini, Giuseppe; Bartolucci, Gian Luca; Teixeira Godoy, Helena (2006). Determination of phenolic compounds in Brazilian and Italian wines. In: SCI2006: XXII Congresso nazionale della Società Chimica Italiana, Firenze, 10-15 Settembre 2006, Società Chimica Italiana, pp. 420-420.
Turillazzi S; Mastrobuoni G; Dani FR; Moneti G; Pieraccini G; la Marca G; Bartolucci G; Perito B; Lambardi D; Cavallini V; Dapporto L. (2006). Dominulin A and B: two new antibacterial peptides identified on the cuticle and in the venom of the social paper wasp Polistes dominulus using MALDI-TOF, MALDI-TOF/TOF, and ESI-ion trap.. JOURNAL OF THE AMERICAN SOCIETY FOR MASS SPECTROMETRY, vol. Mar;17(3), pp. 376-383, ISSN:1044-0305
DOI
G.Bartolucci; G.Mastrobuoni (2005). Trace analysis in mass spectrometry. In: E.Marcantoni; G.Renzi. Seminars in organic synthesis. «A. Corbella» Summer School 2005, pp. 93-114, Roma: Società Chimica Italiana, ISBN:9788886208307.
V. Giannellini;M. Bambagiotti-Alberti;G. Bartolucci;B. Bruni;S.A. Coran;F. Costantino;M. Di Vaira (2005). Solid-state study of mepivacaine hydrochloride. JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, vol. 39, pp. 444-454, ISSN:0731-7085
DOI
Valerio Giannellini;Francesco Salvatore;Gianluca Bartolucci;Silvia A. Coran;Massimo Bambagiotti-Alberti (2005). A validated HPLC stability-indicating method for the determination of diacerhein in bulk drug substance. JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, vol. 39, pp. 776-780, ISSN:0731-7085
DOI
Innocenti, Marzia; Bartolucci, Gian Luca; Vincieri, Franco Francesco; Mulinacci, Nadia (2005). Identification of carotenoids pigments from Rosa Canina L. and Rhodutorula by HPLC-DAD and HPLC coupled to APCI mass spectrometric detection. In: Massa2005: An international symposium on mass spectrometry, Roma, 28 Giugno-01 Luglio 2005, Società Chimica Italiana Divisione Spettrometria di Massa, pp. 98-98.
Villanelli, Fabio; Pieraccini, Giuseppe; Bartolucci, Gian Luca; Davoli, Enrico; Moneti, Gloriano (2005). New technology on ion trap instrument to improve sensitivity. In: Massa2005: An international Symposium on Mass Spectrometry, Roma, 28 Giugno-01 Luglio 2005, Società Chimica Italiana Divisione Spettrometria di Massa, pp. 17-17.
Mastrobuoni, Guido; Dani; Francesca Romana, ; Pansolli, C.; Dapporto, L.; Gofer, S.; Turbanti, Luca; Bartolucci, Gian Luca; Pieraccini, G.; Mastroianni, D.; De Angelis, F.; Moneti, G.; Turillazzi, S. (2004). Characterization of epicuticolar peptides from social wasps by MS/MS. In: Massa2004: An international symposium on mass spectrometry, Bari, 26-30 Settembre 2004, Società Chimica Italiana Divisione Spettrometria di Massa, pp. 15-15.
Bartolucci, Gian Luca; Gori, A; Abbate, R.; La Marca, Giancarlo; Villanelli, Fabio; Pieraccini, Giuseppe; Moneti, Gloriano (2004). A rapid and sensitive method for simultaneous quantitation of homocysteine, choline, betaine and dimethylglycine in human serum and plasma by HPLC-ESI-MS/MS. In: Massa2004: An international symposium on mass spectrometry, Bari, 26-30 Settembre 2004, Società Chimica Italiana Divisione Spettrometria di Massa, pp. 45-45.
Pieraccini, Giuseppe; Bartolucci, Gian Luca; Moneti, Gloriano (2004). Doping vs Antidoping: a never ending match. In: PBA2004 15th International symposium on pharmaceutical and biomedical analysis, Firenze, 2-6 Maggio 2004, Centro stampa 2P s.r.l., pp. 29-29.
F. Boscaro; G. Pieraccini; G. la Marca; G. Bartolucci; C. Luceri; F. Luceri; G. Moneti (2002). Rapid quantitation of globotriaosylceramide in human plasma and urine: a potential application for monitoring enzyme replacement therapy in Anderson-Fabry disease. RAPID COMMUNICATIONS IN MASS SPECTROMETRY, vol. 16, pp. 1507-1514, ISSN:0951-4198, John Wiley & Sons Limited:1 Oldlands Way, Bognor Regis, P022 9SA United Kingdom:011 44 1243 779777, EMAIL: cs-journals@wiley.co.uk, INTERNET: http://www.wiley.co.uk, Fax: 011 44 1243 843232:
G. Pieraccini; G. Bartolucci; M. Pacenti; S. Dugheri; P. Boccalon; L. Focardi (2002). Gas chromatographic determination of glutaraldehyde in the workplace atmosphere after derivatization with 0-(2,3,4,5,6-pentafluorobenzyl)hydroxylamine on a solid-phase microextraction fibre.. JOURNAL OF CHROMATOGRAPHY A, vol. 955, pp. 117-124, ISSN:0021-9673
P. Crabbe; G. Pieraccini; G. Bartolucci; G. Moneti; C. Van Peteghem (2002). Influence of Helix pomatia enzyme preparations on the oxidative conversion of some clostebol acetate metabolites in urine.. JOURNAL OF ANALYTICAL TOXICOLOGY, vol. 26, pp. 73-80, ISSN:0146-4760
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G. Moneti; G. Pieraccini; G. Bartolucci; G. Guida; R. Seraglia; P. Traldi (2001). Direct coupling of a nano-high-performance liquid chromatography column to an ion trap designed for a gas chromatography/mass spectrometry system. RAPID COMMUNICATIONS IN MASS SPECTROMETRY, vol. 15, pp. 1607-1617, ISSN:0951-4198
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M. Peruzzi; G. Bartolucci; F. Cioni (2000). Determination of phenoxyalkanoic acids and other herbicides at the ng/ml level in water by solid-phase extraction with poly(divinylbenzene-co-N-vinylpyrrolidone) sorbent and high-performance liquid chromatography--diode-array detection.. JOURNAL OF CHROMATOGRAPHY A, vol. 867, pp. 169-175, ISSN:0021-9673
F.Mantelli; G.Caldini; P. Bucci; F. Cioni; G. Bartolucci (2000). Quality control of surface waters for drinking water production in the Province of Florence according to law n. 152/99 of May 1, 1999. BOLLETTINO DEI CHIMICI IGIENISTI. PARTE SCIENTIFICA, vol. 51, pp. 139-152, ISSN:1722-2079
G. Bartolucci; G. Pieraccini; F. Villanelli; G. Moneti; A. Triolo (2000). Liquid chromatography tandem mass spectrometric quantitation of sulfamethazine and its metabolites: direct analysis of swine urine by triple quadrupole and by ion trap mass spectrometry.. RAPID COMMUNICATIONS IN MASS SPECTROMETRY, vol. 14, pp. 967-973, ISSN:0951-4198
DOI
F. Cioni; G. Bartolucci; G. Pieraccini; S. Meloni; G. Moneti (1999). Development of a solid phase microextraction method for detection of the use of banned azo dyes in coloured textiles and leather. RAPID COMMUNICATIONS IN MASS SPECTROMETRY, vol. 13, pp. 1833-1837, ISSN:0951-4198
DOI
R. Ferrari; T. Nilsson; R. Arena; P. Arlati; G. Bartolucci; R. Basla; F. Cioni; G. Del Carlo; P. Dellavedova; E. Fattore; M. Fungi; C. Grote; M. Guidotti; S. Morgillo; L. Müller; M. Volante (1998). Inter-laboratory validation of solid-phase microextraction for the determination of triazine herbicides and their degradation products at ng/l level in water samples.. JOURNAL OF CHROMATOGRAPHY A, vol. 795, pp. 371-376, ISSN:0021-9673
G. Danza; S. Dini; G. Bartolucci; G. Lentini; A. Becorpi; G. Massi; A. Guarna; M. Serio (1996). Isotopic dilution GC-MS measurement of 4-Hydroxyandrostendione in postmenopausal breast cancer. ENDOCRINE-RELATED CANCER, vol. 3, pp. 137-143, ISSN:1351-0088
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G.Bartolucci; A. Guarna; G. Danza; A. Marrucci; S. Dini; M. Serio (1996). Quantitative determination of Finasteride in human plasma at picogram level by an isotopic-dilution mass-spectrometry method. INTERNATIONAL JOURNAL OF ANDROLOGY, vol. 19 (suppl. 1), pp. 1-52, ISSN:0105-6263
DOI
A. Guarna; G. Danza; G. Bartolucci; A. Marrucci; S. Dini; M. Serio (1995). Synthesis of 5,6,6-[2H3]finasteride and quantitative determination of finasteride in human plasma at picogram level by an isotope-dilution mass spectrometric method.. JOURNAL OF CHROMATOGRAPHY B. BIOMEDICAL APPLICATIONS, vol. 674, pp. 197-204, ISSN:0378-4347
F. Cioni; G. Bartolucci (1994). Multiresidue method for the determination of pesticides in aromatic herbs and teas. BOLLETTINO DEI CHIMICI IGIENISTI. PARTE SCIENTIFICA, vol. 45, pp. 51-63, ISSN:1722-2079
F.Cioni; G. Bartolucci (1993). Methods of analysis for natural products with insecticidal activity. BOLLETTINO DEI CHIMICI IGIENISTI. PARTE SCIENTIFICA, vol. 44, pp. 293-303, ISSN:1722-2079
C. Domini; F. Ninci; G. Bartolucci (1992). Integrated pest management and pesticide residues in wine. BOLLETTINO DEI CHIMICI IGIENISTI. PARTE SCIENTIFICA, vol. 43, pp. 97-101, ISSN:1722-2079
Gian Luca BARTOLUCCI
Curriculum
- 11.03.1967: born in Florence, Italy.
- 1995: undergraduate degree in Pharmacy 110/110, University of Florence, advisor Prof. Antonio Guarna.
- 11.01.2001: Researcher in the Department of Pharmaceutical Science of University of Florence
via U.Schiff 6, 50019 Sesto Fiorentino (FI) Italy
- 01.01.2003 since 31-12-2008 member of the Mass Spectrometry Center
as expert in mass spectrometry
- 01.01.2009
member of the Mass Spectrometry Center board
Main research fields:
R&D of Gas and Liquid
Chromatographyc methods for qualification pharmaceutical products. Mass Spectrometric applications in the same field