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Fabrizio MACHETTI

Ruolo attuale:: Docente a Contratto

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fabrizio.machetti(AT)unifi.it

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	Stanza 97 c/o dipartimento di chimica 'Ugo Schiff', via della lastruccia 3-13 Sesto Fiorentino
	055 4573501
	fabrizio.machetti(AT)unifi.it

Fabrizio MACHETTI

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Tesi di Dottorato

Cosimo Antonini, Franca Maria Cordero, Fabrizio Machetti (2024). 5-(Benzoyloxymethyl)isoxazole-3-carboxylic Acid Ethyl Ester. MOLBANK, vol. 2024, pp. 1-5, ISSN:1422-8599 DOI Accesso ONLINE all'editore

Cordero, Franca M.; Giomi, Donatella; Machetti, Fabrizio (2024). 36.9-Five-membered ring systems with O and N atoms. In: R. Alan Aitken, Justin M. Lopchuk. Progress in Heterocyclic Chemistry, pp. 275-308 Elsevier Ltd, ISBN:9780443334948., vol. 36: DOI Accesso ONLINE all'editore

Cordero, Franca Maria; Giomi, Donatella; Machetti, Fabrizio (2024). Synthesis of 2-Azetidinones via Cycloaddition Approaches: An Update. REACTIONS, vol. 5, pp. 492-566, ISSN:2624-781X DOI Accesso ONLINE all'editore

Franca M. Cordero, Donatella Giomi, Fabrizio Machetti (2023). 35.5.7 - Five-membered ring systems with O and N atoms. In: Gordon W. Gribble, R. Alan Aitken. Progress in Heterocyclic Chemistry_Volume 35, pp. 351-382, Oxford: Elsevier Ltd, ISBN:9780443219368. DOI Accesso ONLINE all'editore

Cordero, Franca M.; Lascialfari, Luisa; Machetti, Fabrizio (2023). 34.5.7 - Five-membered ring systems with O and N atoms. In: Gordon W. Gribble, R. Alan Aitken. Progress in Heterocyclic Chemistry_Volume 34, pp. 355-386, Oxford: Elsevier Ltd, ISBN:9780443189395. DOI Accesso ONLINE all'editore

Cordero, Franca M.; Giomi, Donatella; Machetti, Fabrizio (2022). 4.03 - Isoxazoles. In: Franca M. Cordero, Donatella Giomi, Fabrizio Machetti. Comprehensive Heterocyclic Chemistry IV, pp. 308-434 Elsevier Inc., ISBN:9780124095472. DOI Accesso ONLINE all'editore

Cordero Franca Maria, Lascialfari Luisa, Machetti Fabrizio (2021). 33.5.7 - Five-Membered Ring Systems: With O and N Atoms. In: Gordon W. Gribble, John A. Joule. Progress in Heterocyclic Chemistry_Volume 33, pp. 311-340, Oxford: Elsevier Ltd, ISBN:978-0-323-98410-2. DOI Accesso ONLINE all'editore

Cordero, Franca M.; Lascialfari, Luisa; Machetti, Fabrizio (2021). 32.5.7 - Five-Membered Ring Systems: With O and N Atoms. In: Gordon W. Gribble, John A. Joule. Progress in Heterocyclic Chemistry_Volume 32, pp. 365-395, Oxford: Elsevier Ltd, ISBN:978-0-323-89812-6. DOI Accesso ONLINE all'editore

Cordero, Franca M.; Lascialfari, Luisa; Machetti, Fabrizio (2020). 31.5.7 - Five-Membered Ring Systems: With O and N Atoms. In: GORDON W. GRIBBLE, JOHN A. JOULE. Progress in Heterocyclic Chemistry, Volume 31, pp. 399-429 Elsevier Ltd, ISBN:978-0-12-819962-6. DOI Accesso ONLINE all'editore

Biagiotti, Giacomo; Pisaneschi, Federica; Gammon, Seth T.; Machetti, Fabrizio; Ligi, Maria Cristina; Giambastiani, Giuliano; Tuci, Giulia; Powell, Emily; Piwnica-Worms, Helen; Pranzini, Erica; Paoli, Paolo; Cicchi, Stefano; Piwnica-Worms, David (2019). Multiwalled carbon nanotubes for combination therapy: a biodistribution and efficacy pilot study. JOURNAL OF MATERIALS CHEMISTRY. B, vol. -, pp. 1-10, ISSN:2050-750X DOI

Baglieri, Ausilia; Meschisi, Luca; De Sarlo, Francesco; Machetti, Fabrizio (2016). Competitive Copper Catalysis in the Condensation of Primary Nitro Compounds with Terminal Alkynes: Synthesis of Isoxazoles. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. 2016, pp. 4643-4655, ISSN:1434-193X DOI Accesso ONLINE all'editore

Giacomo Biagiotti; Stefano Cicchi; Francesco De Sarlo; Fabrizio Machetti (2014). Reactivity of [60]Fullerene with Primary Nitro Compounds: Addition or Catalysed Condensation to Isoxazolo[60]fullerenes. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, pp. 7906-7915, ISSN:1099-0690 DOI Accesso ONLINE all'editore

Goti, A.; Machetti, F. (2012). XIV Convegno nazionale sulle reazioni pericicliche e sintesi di etero e carbocicli. LA CHIMICA E L'INDUSTRIA, vol. 2012, pp. 70-73, ISSN:0009-4315

E. Trogu; C. Vinattieri; F. De Sarlo; F. Machetti (2012). Acid–Base-Catalysed Condensation Reaction in Water: Isoxazolines andIsoxazoles from Nitroacetates and Dipolarophiles. CHEMISTRY-A EUROPEAN JOURNAL, vol. 18, pp. 2081-2093, ISSN:0947-6539 DOI Accesso ONLINE all'editore

J. Revuelta; F. Machetti; S. Cicchi (2011). Five membered heterocycles: 1,3 azoles. In: J. Alvarez_Builla, J. J. Vaquero, J. barluenga. Modern Heterocyclic Chemistry, pp. 809-924, Weinheim: Wiley-VCH, ISBN:9783527332014.

Trabocchi, Andrea; Mannino, Claudia; Machetti, Fabrizio; De Bernardis, F.; Arancia, S.; Cauda, R.; Cassone, A.; Guarna, Antonio (2010). Identification of Inhibitors of Drug-Resistant Candida albicans Strains from a Library of Bicyclic Peptidomimetic Compounds. JOURNAL OF MEDICINAL CHEMISTRY, vol. 53, pp. 2502-2509, ISSN:0022-2623 DOI Accesso ONLINE all'editore

E. Trogu; F. De Sarlo; F. Machetti (2009). Michael Addition versus Cycloaddition-Condensation of Ethyl Nitroacetate with Electron-deficient Olefins. CHEMISTRY-A EUROPEAN JOURNAL, vol. 15, pp. 7940-7948, ISSN:0947-6539

E. Trogu; L. Cecchi; F. De Sarlo; L. Guideri; F. Ponticelli; F. Machetti (2009). Base- and Copper-Catalysed Condensation of Primary Activated Nitro Compounds with Enolisable Compounds. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. --, pp. 5971-5978, ISSN:1434-193X

P. Quadrelli; B. Bovio; A. Piccinini; P. Caramella; F. De Sarlo; F. Machetti (2009). Conversion of a nitrosocarbonyl hetero Diels-Alder cycloadduct to useful isoxazoline-carbocyclic aminols. TETRAHEDRON, vol. 65, pp. 10679-10684, ISSN:0040-4020

D. GIOMI; F. M. CORDERO; F. MACHETTI (2008). Isoxazoles. In: J. JOULE. Comprehensive Heterocyclic Chemistry - IIIA REVIEW OF THE LITERATURE 1995 – 2007, pp. 365-486, OXFORD: Elsevier Ltd, ISBN:9780080449913. DOI Accesso ONLINE all'editore

L. Cecchi; F. De Sarlo; F. Machetti (2008). Synthesis of 4,5-dihydroisoxazoles by condensation of primary nitro compounds with alkenes by using a copper/base catalytic system.. CHEMISTRY-A EUROPEAN JOURNAL, vol. 14, pp. 7903-7912, ISSN:0947-6539 DOI Accesso ONLINE all'editore

L. Cecchi; F. De Sarlo; F. Machetti (2007). 4,5-Dihydroisoxazoles by copper(II)-catalysed condensation of primary nitroalkanes with dipolarophiles. SYNLETT, vol. --, pp. 2451-2453, ISSN:0936-5214 DOI Accesso ONLINE all'editore

Fabrizio MACHETTI; L. Cecchi; E. Trogu; F. De Sarlo (2007). Isoxazoles and Isoxazolines by 1,3-dipolar Cycloaddition (1,3-DC). Base-Catalyzed Condensation of Primary Nitro compounds with Dipolarophiles to Isoxazole Derivatives.. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. --, pp. 4352-4359, ISSN:1434-193X DOI Accesso ONLINE all'editore

F.Machetti; I.Bucelli; G.Indiani; O.Kappe; A.Guarna (2007). Parallel Synthesis of an Amide Library Based on the 6,8-Dioxa-3-azabicyclo[3.2.1]octane Scaffold by Direct Aminolysis of Methyl Esters.. JOURNAL OF COMBINATORIAL CHEMISTRY, vol. 9, pp. 454-461, ISSN:1520-4766 DOI Accesso ONLINE all'editore

MACHETTI F; BUCELLI I; INDIANI G; KAPPE C. O; A. GUARNA (2007). Synthesis of an Amide Library Based on the 6,8-Dioxa-3-azabicyclo[3.2.1]octane Scaffold by Direct Aminolysis of Methyl Esters. JOURNAL OF COMBINATORIAL CHEMISTRY, vol. 9, pp. 454-461, ISSN:1520-4766, American Chemical Society:1155 Sixteenth Street Northwest:Washington, DC 20036:(800)227-5558, EMAIL: service@acs.org, INTERNET: http://www.pubs.acs.org, Fax: (614)447-3671:

C. Mannino; M. Nievo; F. Machetti; A.Papakyriakou; V. Calderone; M. Fragai; A. Guarna (2006). Synthesis of Bicyclic Molecular Scaffolds (BTAa) for the Development of New Matrix Metalloproteinases Inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 14, pp. 7392-7403, ISSN:1464-3391 DOI Accesso ONLINE all'editore

L. Cecchi; F. De Sarlo; C. Faggi; Fabrizio MACHETTI (2006). 1,2,5-Oxadiazole (Furazan) derivatives from benzoylnitromethane and dipolarophiles in the presence of DABCO: structure and intermediates.. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. --, pp. 3016-3020, ISSN:1434-193X DOI Accesso ONLINE all'editore

A. Meucci; F. Machetti; M. De Santis (2006). STUDIO DELLE CARATTERISTICHE ANALITICHE ED APPLICATIVE DI ALCUNI TANNINI VEGETALI E SINTETICI PER LA CONCIA DEL CUOIO.. TECNOLOGIE CONCIARIE, vol. 201, pp. 105-119

L. Cecchi; F. De Sarlo; Fabrizio MACHETTI (2006). 1,4-Diazabicyclo[2.2.2]octane (DABCO) as an efficient reagent for the synthesis of isoxazole derivatives from primary nitro compounds and dipolarophiles: The role of the base. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. --, pp. 4852-4860, ISSN:1434-193X DOI Accesso ONLINE all'editore

F. M. Cordero; S. Bonollo; F. Machetti; A. Brandi (2006). The Synthesis of 4-Hydroxypipecolic Acids by Stereoselective Cycloaddition of Configurationally Stable Nitrones. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. 2006, pp. 3235-3241, ISSN:1434-193X DOI

TRABOCCHI A.; MENCHI G.; GUARNA F.; MACHETTI F.; SCARPI D.; A. GUARNA (2006). Design, Synthesis and Applications of 3-Aza-6,8-Dioxa-Bicyclo[3.2.1]Octane-Based Scaffolds for peptidominetic Chemistry. SYNLETT, vol. ..., pp. 331-353, ISSN:0936-5214, Georg Thieme Verlag Stuttgart:Postfach 301120, D-70451 Stuttgart Germany:011 49 711 8931321, EMAIL: aboservice@thieme.de, INTERNET: http://www.thieme.de, Fax: 011 49 711 8931422: DOI

L. Ricci; M. Frosini; N. Gaggelli; G. Valensin; F. Machetti; G. Sgaragli; M. Valoti. (2006). Inhibition of rabbit brain 4-aminobutyrate transaminase by some taurine analogues: a kinetic analysis.. BIOCHEMICAL PHARMACOLOGY, vol. 70, pp. 1510-1519, ISSN:0006-2952 DOI Accesso ONLINE all'editore

A.Guarna; F.Machetti; E.G.Occhiato (2005). Synthesis of benzo[c]quinolizin-3-ones: discovery and development of novel inhibitors of human steroid 5alpha-reductase. In: O.Attanasi, D.Spinelli. Targets in heterocyclic systems - chemistry and properties, pp. 428-455, Roma: Società Chimica Italiana.

L. Cecchi; F. De Sarlo; Fabrizio MACHETTI (2005). Isoxazoline derivatives from activated primary nitro compounds and tertiary diamines. TETRAHEDRON LETTERS, vol. 46, pp. 7877-7879, ISSN:0040-4039 DOI Accesso ONLINE all'editore

F. M. CORDERO; F. PISANESCHI; K. MESCHINI BATISTA; S. VALENZA; F. MACHETTI; A. BRANDI (2005). A New Bicyclic Dipeptide Isostere with Pyrrolizidinone Skeleton. JOURNAL OF ORGANIC CHEMISTRY, vol. 70, pp. 856-867, ISSN:0022-3263 DOI Accesso ONLINE all'editore

F. M. CORDERO; F. PISANESCHI; M. SALVATI; F. MACHETTI; A. BRANDI (2004). PYRROLIZINONE DERIVATIVES AS NEW BICYCLIC GLY-PRO DIPEPTIDE ISOSTERS. In: TWELFTH FECHEM CONFERENCE ON HETEROCYCLES IN BIO-ORGANIC CHEMISTRY, SIENA, 20-24 June 2004, pp. 31-31.

F. Machetti; F. M. Cordero; F. De Sarlo; A.M. Papini; M.C. Alcaro; A. Brandi (2004). Synthesis of free and Nalpha-Fmoc/Ngamma-Boc protected (2S, 4S)- and (2S, 4R)-4-aminopipecolic acids. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. 13, pp. 2928-2935, ISSN:1434-193X DOI

A. TRABOCCHI; G. MENCHI; M. ROLLA; F. MACHETTI; I. BUCELLI; A. GUARNA (2003). Enantiospecific synthesis of 3-aza-6,8-dioxa-bicyclo[3.2.1]octane carboxylic acids from erythrose. TETRAHEDRON, vol. 59, pp. 5251-5258, ISSN:0040-4020

F.Machetti; I.Bucelli; G.Indiani; A.Guarna (2003). Neat reaction of carboxylic acid methyl esters and amines for efficient parallel synthesis of scaffold amide libraries.. COMPTES RENDUS CHIMIE, vol. 6, pp. 631-633, ISSN:1631-0748 DOI Accesso ONLINE all'editore

S. VALENZA; F. M. CORDERO; F. MACHETTI; A. BRANDI (2002). DETERMINATION OF ABSOLUTE CONFIGURATION OF BICYCLIC LACTAMIC PROLINES USING THEIR MTPA ESTERS. In: 23RD IUPAC INTERNATIONAL SYMPOSIUM ON THE CHEMISTRY OF NATURAL PRODUCTS, FIRENZE, 28 luglio-2 agosto 2002, pp. 364-364.

F. M. CORDERO; M. CACCIARINI; F. MACHETTI; F. DE SARLO (2002). Synthesis of Taurine Analogues, Part 2. Amino-Sulfonation of Alkenes by a Three Component Reaction. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. 2002, pp. 1407-1411, ISSN:1434-193X

A. Brandi; A. M. Papini; F. De Sarlo; F. M. Cordero; F. Machetti (2002). Studies Towards the Synthesis of Enantiopure 4-Substituted Pipecolic Acids. In: 23RD IUPAC INTERNATIONAL SYMPOSIUM ON THE CHEMISTRY OF NATURAL PRODUCTS, FIRENZE, vol. Atti convegno, pp. 265-265.

CINI N; MACHETTI F; MENCHI G; OCCHIATO E G; A. GUARNA (2002). Bicyclic compounds derived from Tartaric Acid and α-Amino acids (BTAas): Synthesis of New Molecular Scaffolds derived from the Combination of (R,R)-Tartaric Acid and L-Serine. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. ..., pp. 873-880, ISSN:1434-193X

A.GUARNA; I.BUCELLI; F.MACHETTI; G. MENCHI; E.G.OCCHIATO; D.SCARPI; A.TRABOCCHI (2002). Synthesis of New Enantiopure Bicycles gamma/delta-Amino Acid (BTKa), Derived from Tartaric Acid and alfa-Aminoacetophenone. TETRAHEDRON, vol. 58, pp. 9865-9870, ISSN:0040-4020 DOI

N. CINI; F. MACHETTI; G. MENCHI; E. G. OCCHIATO; A. GUARNA (2002). Bicyclic Compounds Derived from Tartaric Acid and -Amino Acids (BTAas): Synthesis of New Molecular Scaffolds Derived from the Combination of (R,R)-Tartaric Acid and L-Serine. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. ., pp. 873-880, ISSN:1434-193X, Wiley-VCH Verlag GmBH:PO Box 101161, D 69451 Weinheim Germany:011 49 6201 606147, EMAIL: service@wiley-vch.de, INTERNET: http://www.wiley-vch.de, Fax: 011 49 6201 606328:

A. GUARNA; E.G. OCCHIATO; F. MACHETTI; A. TRABOCCHI; D. SCARPI; G. DANZA; R. MANCINA; A. COMERCI; M. SERIO (2001). Effect of C-Ring Modifications in Benzo[c]quinolizin-3-ones, New Selective Inhibitors of Human 5a-Reductase 1. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 9, pp. 1385-1393, ISSN:0968-0896 DOI

F. M. Cordero; S. Valenza; F. Machetti; A. Brandi (2001). Design and Synthesis of a New Bicyclic Dipeptide Isostere. CHEMICAL COMMUNICATIONS, vol. 2001, pp. 1590-1591, ISSN:1359-7345 DOI

F. MACHETTI; F. M. CORDERO; F. DE SARLO; A. BRANDI (2001). Practical synthesis of both enantiomers of protected 4-oxopipecolic acid.. TETRAHEDRON, vol. 57, pp. 4995-4998, ISSN:0040-4020

GUARNA A; E. OCCHIATO; SCARPI D; MENCHI G; MACHETTI F (2000). 3-Aza-6,8-dioxabicyclo (3,2,1) octanes and analogues and combinatorial libraries. Numero: PCT WO 01/64686 A1 Università di Firenze

A. GUARNA; F. MACHETTI; E. OCCHIATO; D. SCARPI; A. COMERCI; G. DANZA; R. MANCINA; M. SERIO; K. HARDY (2000). Benzo[c]quinolizin-3-ones: a novel class of potent and selective nonsteroidal inhibitors of human steroid 5alpha-reductase 1. JOURNAL OF MEDICINAL CHEMISTRY, vol. 43, pp. 3718-3735, ISSN:0022-2623

F. M. CORDERO; A. BRANDI; S. VALENZA; F. MACHETTI (2000). BICYCLIC DIPEPTIDE ISOSTERES, THEIR PREPARATION AND USE AS BETA-TURN MIMICS. Numero: EP 1 205 487 A1 F. M. CORDERO, A. BRANDI, S. VALENZA, F. MACHETTI

F. MACHETTI; M. CACCIARINI; F. CATRAMBONE; F. M. CORDERO; M. FROSINI; F. DE SARLO (2000). Synthesis of Taurine Analogues from Alkenes. In: Fabrizio Machetti, Martina Cacciarini, Ferdinando Catrambone, Franca Maria Cordero, Maria Frosini, Franceaco De Sarlo. ADVANCES IN EXPERIMENTAL MEDICINE AND BIOLOGY , pp. 399-401, New York: Plenum Press:Book Customer Service, 233 Spring Street:New York, NY 10013:(212)620-8471, (212)620-8000, EMAIL: info@plenum.com, INTERNET: http://www.plenum.com, Fax: (212)807-1047, ISBN:0-306-46447-0.

F. MACHETTI; M. CACCIARINI; F. CATRAMBONE; F. M. CORDERO; S. ROMOLI; F. DE SARLO; (2000). SYNTHESIS OF TAURINE ANALOGUES. PART 1: 2-AMINOSULFONIC ACIDS FROM ALKENE-SULFUR MONOCHLORIDE ADDUCTS. JOURNAL OF CHEMICAL RESEARCH. SYNOPSES, vol. 2000, pp. 120-121, ISSN:0308-2342

A. GUARNA; F. MACHETTI; E. OCCHIATO; D. SCARPI; E. LOMBARDI (2000). MODIFICATION OF THE AZA-ROBINSON ANNULATION FOR THE SYNTHESIS OF 4-METHYL-BENZO[C]QUINOLIZIN-3-ONES, POTENT INHIBITORS OF STEROID 5A-REDUCTASE 1. JOURNAL OF ORGANIC CHEMISTRY, vol. 65, pp. 8093-8095, ISSN:0022-3263

MACHETTI F.; FERRALI A.; MENCHI G.; OCCHIATO E.G.; A. GUARNA (2000). Oligomers of enantiopure bicyclic g/d-amino acids (BTAa). 1. Synthesis and conformational analysis of 3-Aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic acid oligomers (PolyBTG). ORGANIC LETTERS, vol. 2, pp. 3987-3990, ISSN:1523-7060

A.Guarna; E.G.Occhiato; F.Machetti; G.Danza; M.Serio (2000). Emerging drugs for the third millenium. Discovery and development of the inhibitors of steroids 5alpha-reductase as drugs for the androgen-dependant diaseas. In: XXV Summer school A. Corbella, Gargnano, 12-16/6/2000, Società Chimica Italiana, pp. 47-68, ISBN:88-86208-15-4

A. GUARNA; A. GUIDI; F. MACHETTI; G. MENCHI; E. OCCHIATO; D. SCARPI; S. SISI; A. TRABOCCHI (1999). Synthesis and reactivity of bicycles derived from tartaric acids and alfa-amino acids: a novel class of conformationally constrained dipeptide isosteres based upon enantiopure 3-aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic acid. JOURNAL OF ORGANIC CHEMISTRY, vol. 64, pp. 7347-7364, ISSN:0022-3263

A. GUARNA; E. OCCHIATO; F. MACHETTI; V. GIACOMELLI (1999). 19-NOR-10-AZASTEROIDS. 5.1 A SYNTHETIC STRATEGY FOR THE PREPARATION OF (+)-17-(3-PYRIDYL)-(5B)-10-AZAESTRA-1,16-DIEN-3-ONE, A NOVEL POTENTIAL INHIBITOR FOR HUMAN CYTOCHROME P45017A (17A-HYDROXYLASE/C17,20-LYASE). JOURNAL OF ORGANIC CHEMISTRY, vol. 64, pp. 4985-4989, ISSN:0022-3263

A. GUARNA; E. OCCHIATO; F. MACHETTI; D. SCARPI (1998). A CONCISE ROUTE TO 19-NOR-10-AZASTEROIDS, A NEW CLASS OF STEROID 5-REDUCTASE INHIBITORS. 3.1 SYNTHESIS OF (+)-19-NOR-10-AZATESTOSTERONE AND (+)-17B-ACETYLOXY-(5B)-10-AZAESTR-1-EN-3-ONE. JOURNAL OF ORGANIC CHEMISTRY, vol. 63, pp. 4111-4115, ISSN:0022-3263

E. OCCHIATO; D. SCARPI; F. MACHETTI; A. GUARNA (1998). STEREOSELECTIVITY IN THE TICL4-CATALYSED REEACTION OF DANISHEFSKY'S DIENE WITH A N-(ACYLOXY)IMINIUM ION: SYNTHESIS OF 5A VERSUS 5B D1(2)-19-NOR-10-AZASTEROIDS. PART 4. TETRAHEDRON, vol. 54, pp. 11589-11596, ISSN:0040-4020

A. GUARNA; C. BELLE; F. MACHETTI; E. OCCHIATO; A. H. PAYNE; C. CASSIANI; A; COMERCI; G. DANZA; A. DE BELLIS; S. DINI; A. MARRUCCI; M. SERIO (1997). 19-nor-10-azasteroids: a novel class of inhibitors for human steroid 5alpha-reductases 1 and 2. JOURNAL OF MEDICINAL CHEMISTRY, vol. 40, pp. 1112-1129, ISSN:0022-2623

F. M. Cordero; F. Machetti; F. De Sarlo; A. Brandi (1997). New Synthesis of (Methoxycarbonyl)-indolizidine-7-one and -quinolizidine-2-one: an Access to β-Aminoacids with Indolizidine and Quinolizidine Backbone. GAZZETTA CHIMICA ITALIANA, vol. 127, pp. 25-29, ISSN:0016-5603

A. GUARNA; Fabrizio MACHETTI; A. MARRUCCI; G. DANZA; M. SERIO. (1997). Synthesis and Structure-Activity Relationship of 19-Nor-10-azasteroids, a New Class of 5α -Reductase Inhibitors in Human Prostate.. PHARMACOLOGICAL RESEARCH, vol. 35, pp. 226-227, ISSN:1043-6618

A. GUARNA; E. OCCHIATO; F. MACHETTI; G. DANZA; M. SERIO; P. PAOLI; A. MARRUCCI (1997). 19-nor-10-azasteroids, a new class of steroid 5a-reductase inhibitors. 2. X-ray structure, molecular modeling, conformational analysis of 19-nor-10-azasteroids and comparison with 4-azasteroids and 6-azasteroids. JOURNAL OF MEDICINAL CHEMISTRY, vol. 40, pp. 3466-3477, ISSN:0022-2623

F. Machetti; F. M. Cordero; F. De Sarlo; A. Guarna; A. Brandi (1996). A New Synthesis of (2S)-4-Oxopipecolic Acid by Thermal Rearrangement ofEnantiopure Spirocyclopropaneisoxazolidine. TETRAHEDRON LETTERS, vol. 37, pp. 4205-4208, ISSN:0040-4039

F. Machetti; B. Anichini; S. Cicchi; A. Brandi; W. Wieczoreck; K. M. Pietrusiewicz; J.-C. Gehret (1996). Synthesis and X-ray study of hexahydro- and tetrahydrophospholo[2,3-d]isoxazoles, a new class of heterocycles of potential fungicidal activity. JOURNAL OF HETEROCYCLIC CHEMISTRY, vol. 33, pp. 1091-1098, ISSN:0022-152X