Tondo AR; Fantacuzzi M; Carradori S; D'Agostino I; Angeli A; Supuran CT; Capasso C; Gambacorta N; Piemontese L; Laghezza A; Nicolotti O; Agamennone M (2026). Targeting microbial β-CAs: bridging in silico screening with in vitro validation. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 134, pp. 0-0, ISSN:1464-3391 DOI  

  Gioele Renzi; Lorenzo Masoni; Fabrizio Carta; Marta Ferraroni; Maria Luisa Massardi; Nicolas Tassone; Roberto Ronca; Claudiu T. Supuran; Andrea Angeli (2026). Expanding the Inhibitory Potential of the Benzoxaborinine Scaffold against Carbonic Anhydrases: Synthesis, Structural Characterization, and In Vitro Antitumor Activity. JOURNAL OF MEDICINAL CHEMISTRY, pp. 0-0, ISSN:0022-2623 DOI  

  Costa A.; Provensi G.; Titi C.; Leri M.; Bucciantini M.; Ferraroni M.; Keeton A.B.; Moore A.M.; Piazza G.A.; Abadi A.H.; Angeli A.; Supuran C.T. (2026). Exploring dual inhibitors Carbonic Anhydrases and Phosphodiesterase 5 as potential agents for treatment Alzheimer's disease. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 303, pp. 0-0, ISSN:0223-5234 DOI  

  Venkatesan Saravanan; Andrea Angeli; Francesco Melfi; Nicola Amodio; Ilenia Valentino; Massimo Gentile; Ilaria D'Agostino; Kathiravan Muthukumaradoss; Gokhan Zengin; Davide Moi; Rahime Simsek; Claudiu T. Supuran; Simone Carradori (2026). Coumarin– and Dipicolylamine–Terpenoid Hybrids as Selective Carbonic Anhydrases IX and XII Inhibitors: Mechanistic Insights and Selective Anti-Cancer Potential. Pharmaceuticals , pp. 0-0 DOI  

  Sequeira L.; Distinto S.; Fernandes C.; Sanna E.; Meleddu R.; Gaspari M.; Cottiglia F.; Onali A.; Angeli A.; Borges F.; Uriarte E.; Alcaro S.; Supuran C.T.; Maccioni E. (2026). Chromones as Nonclassical Inhibitors of Carbonic Anhydrase IX and XII Isoforms: Probing Chromone-Based Derivatives. ARCHIV DER PHARMAZIE, vol. 359, pp. 0-0, ISSN:0365-6233 DOI  

  Iacovozzi D.; Carradori S.; Osmanovic A.; Supuran C.T.; Capasso C.; Angeli A. (2026). Managing Malassezia species and related infections: new insights into recent natural and synthetic antifungal compounds and their mechanism of action. MOLECULAR DIVERSITY, pp. 0-0, ISSN:1381-1991 DOI  

  Alberto Deplano; Davide Moi; Serena Vittorio; Andrea Angeli; Claudiu T. Supuran; Valentina Onnis (2026). Synthesis of Hydrazidoureidobenzensulfonamides Incorporating a Nicotinoyl Tail and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity. PHARMACEUTICALS, vol. 19, pp. 0-0, ISSN:1424-8247 DOI  

  Angeli A.; Petrou A.; Kartcev V.; Prezent M.; Sirakanyan S.; Geronikaki A.; Supuran C.T. (2026). p-Aminobenzene-Sulfonamide Derivatives of Substituted Pyrimidines as Human Carbonic Anhydrase Inhibitors. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 27, pp. 0-0, ISSN:1422-0067 DOI  

  Alessandro Bonardi; Marta Ferraroni; Paola Gratteri; Claudiu T. Supuran; Andrea Angeli (2026). Structural and Pharmacological Characterization of AT-121 Reveals Carbonic Anhydrase Inhibition as a Complementary Mechanism to Dual MOR/NOR Agonism. ACS MEDICINAL CHEMISTRY LETTERS, pp. 0-0, ISSN:1948-5875 DOI  

  Bonardi, Alessandro; Carradori, Simone; Paoletti, Niccolò; Angeli, Andrea; Ferraroni, Marta; Iacovozzi, Damiano; Gallorini, Marialucia; D'Agostino, Ilaria; De Luca, Viviana; Gratteri, Paola; Cataldi, Amelia; Supuran, Claudiu T.; Capasso, Clemente (2026). Production, crystallographic studies, and functional profiling of γ-carbonic anhydrase from the probiotic Limosilactobacillus reuteri: In vitro and cell-based insights. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 302, pp. 0-0, ISSN:0223-5234 DOI  

  Yitong Wang; Alessio Nocentini; Marta Ferraroni; Andrea Angeli; Xin Wang; Zhongyu Liu; Mengbi Guo; Cheng Peng; Bin Lin; Zhuang Hou; Yang Liu; Claudiu T. Supuran; Chun Guo (2026). Discovery of Subnanomolar and Highly Selective Carbonic Anhydrase II Inhibitors Featuring L-Shaped Scaffolds via Active-Site-Matched Fragment Growing. JOURNAL OF MEDICINAL CHEMISTRY, vol. 69, pp. 14461-14491, ISSN:0022-2623 DOI  

  Gioele Renzi; Alessandro Tubita; Lorenzo Antonuzzo; Serena Pillozzi; Marta Ferraroni; Andrea Angeli; Claudiu T. Supuran (2026). Design and Synthesis of Bendamustine-Carbonic Anhydrase Inhibitors with Antiproliferative Effects in Clear Cell Renal Cell Carcinoma. JOURNAL OF MEDICINAL CHEMISTRY, pp. 0-0, ISSN:0022-2623 DOI  

  Baroni C.; Ferraroni M.; Supuran C.T.; Angeli A. (2026). Beyond Neddylation Inhibition: X-ray Structures Reveal Carbonic Anhydrase Isoform Selectivity of Pevonedistat. ACS MEDICINAL CHEMISTRY LETTERS, vol. 17, pp. 1393-1397, ISSN:1948-5875 DOI  

  Elena Andreucci , Alessio Biagioni , Sara Peri , Nunzia Di Menna , Michela Pinto , Serena Martinelli , Laura Papucci , Lucia Magnelli , Gioele Renzi , Silvia Selleri , Andrea Angeli , Clemente Capasso , Fabrizio Carta , Claudiu T Supuran (2026). Ketoconazole-carbonic anhydrase inhibitors as potential anticancer agents. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 304, pp. 0-0, ISSN:0223-5234 DOI   Accesso ONLINE all'editore

  Bhowmik R.; D'Agostino I.; Angeli A.; Aspatwar A. (2026). Integrated in silico and in vitro screening approaches for the discovery of small-molecule inhibitors of β-carbonic anhydrases. EXPERT OPINION ON DRUG DISCOVERY, vol. 21, pp. 319-337, ISSN:1746-0441 DOI  

  El-Attar M.A.Z.; Afifi O.S.; Ismail A.; Kamel Y.N.; Yassin H.A.; Nomeir H.M.; Nematalla H.A.; Angeli A.; Labib H.F.; Eldehna W.M.; Supuran C.T.; Belal A.S.F.; Elzahhar P.A.; Hassan N.W. (2026). Click-modifiable isatin hydrazones as COX-2, VEGFR-2, and carbonic anhydrase inhibitors: A multi-target approach to cancer therapy. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 302, pp. 0-0, ISSN:0223-5234 DOI  

  Melfi F.; Mencarelli N.; Carradori S.; Gallorini M.; Angeli A.; Poli G.; Cataldi A.; D'Agostino I.; Di Credico A.; Di Baldassarre A.; Tuccinardi T.; Supuran C.T. (2026). Hybridization Approach Applied to Umbelliferon and Vanilloids toward New Inhibitors of Carbonic Anhydrases IX and XII with In Vitro Antiproliferative and Anti-inflammatory Activities. JOURNAL OF MEDICINAL CHEMISTRY, vol. 69, pp. 1454-1472, ISSN:0022-2623 DOI  

  Abdoli M.; Angeli A.; Bonardi A.; Gratteri P.; Jackevica L.; Sizovs A.; Supuran C.T.; Zalubovskis R. (2026). Investigation on N-Aryl-2-(4-sulfamoylphenyl)hydrazine-1-carbothioamide as Human Carbonic Anhydrases Inhibitors. PHARMACEUTICALS, vol. 19, pp. 0-0, ISSN:1424-8247 DOI  

  Alessia Costa; Murat Bozdag; Gioele Renzi; Barbara Rani; Maria Beatrice Passani; Andrea Angeli; Gustavo Provensi; Fabrizio Carta; Claudiu T. Supuran (2025). Hitting Two Birds With One Stone: Dual Modulation of Brain Carbonic Anhydrases and Histone Deacetylases Boosts Memory Consolidation. ARCHIV DER PHARMAZIE, vol. 358, pp. 0-0, ISSN:1521-4184 DOI  

  Anastasija Balašova; Aleksandrs Pustenko; Andrea Angeli; Elena Andreucci; Alessio Biagioni; Alessio Nocentini; Fabrizio Carta; Claudiu T. Supuran; Raivis Žalubovskis (2025). Unraveling the Potential of Amino-, Acylamino-, and Ureido-Substituted 3H-1,2-Benzoxaphosphepine 2-Oxides toward Nanomolar Inhibitors of Tumor-Associated Carbonic Anhydrases IX and XII. ACS MEDICINAL CHEMISTRY LETTERS, pp. 0-0, ISSN:1948-5875 DOI  

  Berrino E.; Guglielmi P.; Carta F.; Carradori S.; Campestre C.; Angeli A.; Arrighi F.; Pontecorvi V.; Chimenti P.; Secci D.; Supuran C.T.; Gallorini M. (2025). In Vitro CO-Releasing and Antioxidant Properties of Sulfonamide-Based CAI-CORMs in a H2O2-Stimulated Human Achilles Tendon-Derived Cell Model. MOLECULES, vol. 30, pp. 0-0, ISSN:1420-3049 DOI  

  Gioele Renzi; Andrea Angeli; Silvia Selleri; Costanza Spadini; Nicolo' Mezzasalma; Marcus T. Hull; Steven L. Kelly; Clemente Capasso; Clotilde S. Cabassi; Fabrizio Carta; Claudiu T. Supuran (2025). Design and Synthesis of Ketoconazole Derivatives as Innovative Anti‐Infective Agents. ARCHIV DER PHARMAZIE, vol. 358, pp. 0-0, ISSN:1521-4184 DOI  

  Serena Filiberti; Gioele Renzi; Fabrizio Carta; Marialuigia Fantacuzzi; Ilaria D'Agostino; German Benito; Andrea Angeli; Maria Luisa Massardi; Rahime Simsek; Clemente Capasso; Simone Carradori; Roberto Ronca; Claudiu T. Supuran (2025). Pegylation approach applied to erlotinib–carbonic anhydrase inhibitors hybrids towards anticancer agents. RSC MEDICINAL CHEMISTRY, pp. 0-0, ISSN:2632-8682 DOI  

  Angeli A.; Ferraroni M.; Supuran C.T. (2025). Unveiling the Carbonic Anhydrase Inhibitory Profile of Aprocitentan: Kinetic and Structural Characterization. ACS MEDICINAL CHEMISTRY LETTERS, vol. 16, pp. 1682-1686, ISSN:1948-5875 DOI  

  Singh P.; Nerella S.G.; Swain B.; Angeli A.; Kausar S.; Ullah Q.; Supuran C.T.; Arifuddin M. (2025). Synthesis of Chromene-linked Bis-indole Derivatives as Selective Tumor-associated Carbonic Anhydrase IX Inhibitors. ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, vol. 25, pp. 399-410, ISSN:1871-5206 DOI  

  Anakok D.A.; Angeli A.; D'Agostino I.; Renzi G.; Massardi M.L.; Tavani C.; Cete S.; Carradori S.; Ronca R.; Capasso C.; Carta F.; Supuran C.T. (2025). A Journey Around Boronic Acids: Sulfonyl Hydrazone-Containing Derivatives as Carbonic Anhydrase Inhibitors. CHEMICAL BIOLOGY & DRUG DESIGN, vol. 105, pp. 0-0, ISSN:1747-0277 DOI  

  Angeli A.; Petrou A.; Kartsev V.; De Luca V.; Capasso C.; Geronikaki A.; Supuran C.T. (2025). Coumarin-Containing Aromatic Sulfonamides With Carbonic Anhydrase Inhibitory Properties Against Human and Fungal Isoforms. CHEMICAL BIOLOGY & DRUG DESIGN, vol. 106, pp. 0-0, ISSN:1747-0277 DOI  

  Debora Pratesi , Francesco Brenzini Biagioni , Camilla Matassini , Francesca Cardona , Andrea Angeli, Alessandro Bonardi, Paola Gratteri, Claudiu T. Supuran , Andrea Goti (2025). Studies on Azasugar-based sulfonamides: a new class of Carbonic Anhydrase inhibitors. BIOORGANIC CHEMISTRY, vol. 164, pp. 108857-108866, ISSN:0045-2068 DOI  

  Micheli L.; Angeli A.; Di Cesare Mannelli L.; Ghelardini C.; Ferraroni M.; Barons R.; Zalubovskis R.; Zara S.; Carradori S.; Supuran C.T. (2025). Targeting Human Carbonic Anhydrases with Novel Piperazine and Homopiperazine Benzenesulfonamides to Alleviate Paclitaxel-Induced Peripheral Neuropathy. JOURNAL OF MEDICINAL CHEMISTRY, vol. 68, pp. 25485-25504, ISSN:1520-4804 DOI  

  Giovannuzzi S.; Angeli A.; Begines P.; Ferraroni M.; Nocentini A.; Supuran C.T. (2025). Tetrazole Is a Novel Zinc Binder Chemotype for Carbonic Anhydrase Inhibition. ACS MEDICINAL CHEMISTRY LETTERS, vol. 16, pp. 163-166, ISSN:1948-5875 DOI  

  El-Damasy A.K.; Kim H.J.; Faisal M.; Angeli A.; Elsawi A.E.; Eldehna W.M.; Supuran C.T.; Keum G. (2025). Novel N-(3-(1-(4-sulfamoylphenyl)triazol-4-yl)phenyl)benzamide Derivatives as Potent Carbonic Anhydrase Inhibitors with Broad-Spectrum Anticancer Activity: Leveraging Tail and Dual-Tail Approaches. JOURNAL OF MEDICINAL CHEMISTRY, vol. 68, pp. 3764-3781, ISSN:0022-2623 DOI  

  Pontecorvi V.; Angeli A.; Cutarella L.; Mori M.; Secci D.; Coluccia M.; Carradori S.; Troiani A.; Pepi F.; Salvitti C.; Di Noi A.; Spano M.; Arrighi F.; De Falco E.; Bordin A.; Berrino E.; Granese A.; Chimenti P.; Guglielmi P.; Supuran C.T. (2025). Design, synthesis, molecular modelling investigation and biological studies of novel human carbonic anhydrase inhibitors based on coumalic acid. RSC MEDICINAL CHEMISTRY, vol. 16, pp. 3603-3621, ISSN:2632-8682 DOI  

  Paciotti R.; Carradori S.; Angeli A.; D'Agostino I.; Ferraroni M.; Coletti C.; Supuran C.T. (2025). Unprecedented carbonic anhydrase inhibition mechanism: Targeting histidine 64 side chain through a halogen bond. ARCHIV DER PHARMAZIE, vol. 358, pp. 0-0, ISSN:0365-6233 DOI  

  Onali A.; Sanna E.; Lupia A.; Secci D.; Atzeni G.; Demuru L.; Angeli A.; Cottiglia F.; Meleddu R.; Emmolo R.; Corona A.; Maccioni E.; Supuran C.T.; Distinto S. (2025). Synthesis and Evaluation of Thiazolidinone-Isatin Hybrids for Selective Inhibition of Cancer-Related Carbonic Anhydrases. ACS MEDICINAL CHEMISTRY LETTERS, vol. 16, pp. 560-566, ISSN:1948-5875 DOI  

  Poggetti V.; Angeloni E.; Germelli L.; Natale B.; Waqas M.; Sarno G.; Angeli A.; Daniele S.; Salerno S.; Barresi E.; Cosconati S.; Castellano S.; Da Pozzo E.; Costa B.; Supuran C.T.; Da Settimo F.; Taliani S. (2025). Discovery of the First-in-Class Dual TSPO/Carbonic Anhydrase Modulators with Promising Neurotrophic Activity. ACS CHEMICAL NEUROSCIENCE, vol. 16, pp. 1-15, ISSN:1948-7193 DOI  

  Moi D.; Carradori S.; Gallorini M.; Mencarelli N.; Deplano A.; Angeli A.; Vittorio S.; Supuran C.T.; Onnis V. (2025). Investigation on Human Carbonic Anhydrase IX and XII Inhibitory Activity and A549 Antiproliferative Activity of a New Class of Coumarinamides. PHARMACEUTICALS, vol. 18, pp. 0-0, ISSN:1424-8247 DOI  

  Renzi G.; McDonald P.C.; Awrey S.; Tavakoli H.; Bokhari Z.; Lyle M.; Zhang Z.; Ferraroni M.; Dedhar S.; Supuran C.T.; Angeli A. (2025). Dual inhibition of carbonic anhydrase IX and glutathione peroxidase 4 as a novel strategy for ferroptosis-induced tumor cell death. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 300, pp. 0-0, ISSN:0223-5234 DOI  

  Ferraroni M.; Angeli A.; De Luca V.; Capasso C.; Supuran C.T. (2025). Kinetic and structural studies of gamma-carbonic anhydrase from the oral pathogen Porphyromonas gingivalis. JOURNAL OF STRUCTURAL BIOLOGY, vol. 217, pp. 0-0, ISSN:1047-8477 DOI  

  Elena Lucarini; Vanessa D'Antongiovanni; Luca Antonioli; Carla Ghelardini; Lorenzo Di Cesare Mannelli; Marta Ferraroni; Maria Locuoco; Antonella Capperucci; Damiano Tanini; Andrea Angeli; Claudiu T Supuran (2025). Correction: Study of Chalcogen Aspirin Derivatives with Carbonic Anhydrase Inhibitory Properties for Treating Inflammatory Pain (ACS Medicinal Chemistry Letters (2024) 15:9 (1559-1565) DOI: 10.1021/acsmedchemlett.4c00284). ACS MEDICINAL CHEMISTRY LETTERS, vol. 16, pp. 347-347, ISSN:1948-5875 DOI  

  Selleri S.; Angeli A. (2025). Malassezia spp. carbonic anhydrases. THE ENZYMES, vol. 57, pp. 65-89, ISSN:1874-6047 DOI  

  Akgul, Ozlem; Renzi, Gioele; Angeli, Andrea; Ferraroni, Marta; Carta, Fabrizio; Supuran, Claudiu T (2025). Novel Taurinamide-Based Compounds as Carbonic Anhydrase Inhibitors. ARCHIV DER PHARMAZIE, vol. 358, pp. 0-0, ISSN:1521-4184 DOI  

  Gazzaroli, Giorgia; Tavani, Camilla; Filiberti, Serena; Massardi, Maria Luisa; Turati, Marta; Garattini, Giulia; Peat, Thomas S; Pieraccini, Giuseppe; Angeli, Andrea; Supuran, Claudiu T; Carta, Fabrizio; Giacomini, Arianna; Ronca, Roberto (2025). An ureido-substituted benzenesulfonamide carbonic anhydrase inhibitor exerts a potent antitumor effect in vitro and in vivo. EXPERIMENTAL HEMATOLOGY & ONCOLOGY, vol. 14, pp. 0-0, ISSN:2162-3619 DOI  

  Al-Matarneh, Cristina M.; Simionescu, Natalia; Nicolescu, Alina; Silion, Mihaela; Angeli, Andrea; Paoletti, Niccolò; Bonardi, Alessandro; Gratteri, Paola; Pinteala, Mariana; Supuran, Claudiu T. (2025). Novel 3-Sulfonamide Dual-Tail Pyrrol-2-one Bridged Molecules as Potent Human Carbonic Anhydrase Isoform Inhibitors: Design, Synthesis, Molecular Modeling Investigation, and Anticancer Activity in MeWo, SK-BR-3, and MG-63 Cell Lines. JOURNAL OF MEDICINAL CHEMISTRY, vol. 68, pp. 1863-1882, ISSN:0022-2623 DOI  

  Bozdag M.; Mroweh N.; Raucci A.; Angeli A.; Peppicelli S.; Biagioni A.; Calorini L.; Trisciuoglio D.; Ragno R.; Astolfi R.; Giuliani L.; Zwergel C.; Valente S.; Andreucci E.; Carta F.; Mai A.; Supuran C.T. (2025). Discovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells. JOURNAL OF MEDICINAL CHEMISTRY, vol. 68, pp. 22874-22895, ISSN:0022-2623 DOI  

  Melfi F.; D'Agostino I.; Carradori S.; Carta F.; Angeli A.; Costa G.; Renzi G.; Cikos A.; Vullo D.; Resetar J.; Ferraroni M.; Baroni C.; Mancuso F.; Gitto R.; Ambrosio F.A.; Marchese E.; Torcasio R.; Amodio N.; Capasso C.; Alcaro S.; Supuran C.T. (2025). O-derivatization of natural tropolone and β-thujaplicin leading to effective inhibitors of human carbonic anhydrases IX and XII. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 290, pp. 0-0, ISSN:1768-3254 DOI  

  Angeli A.; Ferraroni M.; Capasso C.; Supuran C.T. (2025). Structural Studies of the Dopamine D4 Receptor Antagonist Sonepiprazole as an Inhibitor of Human Carbonic Anhydrases. ACS MEDICINAL CHEMISTRY LETTERS, vol. 16, pp. 483-486, ISSN:1948-5875 DOI  

  Vigiani, Erica; Bonardi, Alessandro; Catarzi, Daniela; Varano, Flavia; Calenda, Sara; Ceni, Costanza; Vagnoni, Giulia; Angeli, Andrea; Nocentini, Alessio; Gratteri, Paola; Supuran, Claudiu T.; Colotta, Vittoria (2025). Repurposing the amino-3,5-dicyanopyridine scaffold from adenosine receptor ligands to carbonic anhydrase activators. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 291, pp. 0-0, ISSN:0223-5234 DOI  

  Spadini, Costanza; Mezzasalma, Nicolo; Odigie, Amienwanlen Eugene; Angeli, Andrea; Carta, Fabrizio; Selleri, Silvia; Gandolfo, Emanuele; Taddei, Simone; Franceschi, Valentina; Minesso, Sergio; Supuran, Claudiu T.; Cabassi, Clotilde Silvia (2025). Comparative efficacy of selenoureido carbonic anhydrase inhibitors and azole antifungal drugs against clinical isolates of Malassezia pachydermatis. VETERINARY DERMATOLOGY (ONLINE), pp. 0-0, ISSN:1365-3164 DOI  

  Angeli A.; Chelli I.; Lucarini L.; Sgambellone S.; Marri S.; Villano S.; Ferraroni M.; De Luca V.; Capasso C.; Carta F.; Supuran C.T. (2024). Novel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy. JOURNAL OF MEDICINAL CHEMISTRY, vol. 67, pp. 3066-3089, ISSN:0022-2623 DOI  

  Lucarini, Elena; D'Antogiovanni, Vanessa; Antonioli, Luca; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Ferraroni, Marta; Locuoco, Maria; Capperucci, Antonella; Tanini, Damiano; Angeli, Andrea; Supuran, Claudiu T. (2024). Study of Chalcogen Aspirin Derivatives with Carbonic Anhydrase Inhibitory Properties for Treating Inflammatory Pain. ACS MEDICINAL CHEMISTRY LETTERS, pp. 0-0, ISSN:1948-5875 DOI  

  Marjan Sobati; Morteza Abdoli; Andrea Angeli; Alessandro Bonardi; Marta Ferraroni; Claudiu T Supuran; Raivis Žalubovskis (2024). Sulfonamide-incorporated bis(α-aminophosphonates) as promising carbonic anhydrase inhibitors: Design, synthesis, biological evaluation, and X-ray crystallographic studies. ARCHIV DER PHARMAZIE, pp. 1-11, ISSN:0365-6233 DOI  

  Marinacci B.; D'Agostino I.; Angeli A.; Carradori S.; Melfi F.; Grande R.; Corsiani M.; Ferraroni M.; Agamennone M.; Tondo A.R.; Zara S.; Puca V.; Pellegrini B.; Vagaggini C.; Dreassi E.; Patrauchan M.A.; Capasso C.; Nicolotti O.; Carta F.; Supuran C.T. (2024). Inhibition of Pseudomonas aeruginosa Carbonic Anhydrases, Exploring Ciprofloxacin Functionalization Toward New Antibacterial Agents: An In-Depth Multidisciplinary Study. JOURNAL OF MEDICINAL CHEMISTRY, vol. 67, pp. 19077-19102, ISSN:1520-4804 DOI   Accesso ONLINE all'editore

  Shaldam MA; Khalil AF; Almahli H; Jaballah MY; Angeli A; Khaleel EF; Badi RM; Elkaeed EB; Supuran CT; Eldehna WM; Tawfik HO (2024). Identification of 3-(5-cyano-6-oxo-pyridin-2-yl)benzenesulfonamides as novel anticancer agents endowed with EGFR inhibitory activity. ARCHIV DER PHARMAZIE, vol. 357, pp. 0-0, ISSN:1521-4184 DOI  

  Angeli A. (2024). Bacterial γ-carbonic anhydrases. THE ENZYMES, vol. 55, pp. 93-120, ISSN:1874-6047 DOI  

  Secci D.; Sanna E.; Distinto S.; Onali A.; Lupia A.; Demuru L.; Atzeni G.; Meleddu R.; Cottiglia F.; Angeli A.; Supuran C.T.; Maccioni E. (2024). Privileged Scaffold Hybridization in the Design of Carbonic Anhydrase Inhibitors. MOLECULES, vol. 29, pp. 0-0, ISSN:1420-3049 DOI  

  Trawally M.; Demir-Yazici K.; Angeli A.; Kaya K.; Akdemir A.; Supuran C.T.; Guzel-Akdemir O. (2024). Thiosemicarbazone-benzenesulfonamide Derivatives as Human Carbonic Anhydrases Inhibitors: Synthesis, Characterization, and In silico Studies. ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, vol. 24, pp. 649-667, ISSN:1871-5206 DOI  

  Angeli A.; De Luca V.; Capasso C.; Di Costanzo L.F.; Supuran C.T. (2024). Comparative CO2 and SiO2 hydratase activity of an enzyme from the siliceous demosponge Suberites domuncula. ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, vol. 758, pp. 0-0, ISSN:0003-9861 DOI  

  Angeli A.; De Luca V.; Huang X.; Winter D.L.; Capasso C.; Supuran C.T.; Donald W.A. (2024). Phosphorylation strongly affects the inhibition of human carbonic anhydrase I CO2 hydration activity. ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, vol. 761, pp. 0-0, ISSN:0003-9861 DOI  

  Angeli A.; Petrou A.; Kartsev V.G.; Zubenko A.; Divaeva L.N.; Chekrisheva V.; Iacopetta D.; Sinicropi M.S.; Sirakanyan S.; Geronikaki A.; Supuran C.T. (2024). Phthalazine Sulfonamide Derivatives as Carbonic Anhydrase Inhibitors. Synthesis, Biological and in silico Evaluation. CHEMMEDCHEM, vol. 19, pp. 0-0, ISSN:1860-7179 DOI  

  Secci D.; Distinto S.; Onali A.; Sanna E.; Lupia A.; Demuru L.; Atzeni G.; Cottiglia F.; Meleddu R.; Angeli A.; Supuran C.T.; Maccioni E. (2024). New Structural Features of Isatin Dihydrothiazole Hybrids for Selective Carbonic Anhydrase Inhibitors. ACS MEDICINAL CHEMISTRY LETTERS, vol. 15, pp. 1860-1865, ISSN:1948-5875 DOI  

  Supuran C.T.; Angeli A.; Tanini D. (2024). Advances in Prodrugs: Design and Therapeutic Applications. Elsevier, ISBN:9780443156359 DOI  

  Tanini D.; Angeli A.; Supuran C.T. (2024). Prodrugs: General concepts and prodrug design in medicinal chemistry. In: Claudiu T. Supuran, A. Angeli, D. Tanini. Advances in Prodrugs: Design and Therapeutic Applications, pp. 3-19 Elsevier, ISBN:9780443156359. DOI  

  Bernardoni B.L.; D'Agostino I.; La Motta C.; Angeli A. (2024). An insight into the last 5-year patents on Porphyromonas gingivalis and Streptococcus mutans, the pivotal pathogens in the oral cavity. EXPERT OPINION ON THERAPEUTIC PATENTS, vol. 34, pp. 433-463, ISSN:1354-3776 DOI  

  Swain B.; Marde V.S.; Singh P.; Angeli A.; Khan A.; Yaddanapudi V.M.; Ullah Q.; Supuran C.T.; Arifuddin M. (2024). Design, synthesis, and biological evaluation of 3-benzenesulfonamide-linked 3-hydrazinoisatin derivatives as carbonic anhydrase inhibitors. ARCHIV DER PHARMAZIE, vol. 357, pp. 0-0, ISSN:0365-6233 DOI  

  De Luca L.; Bucolo F.; Angeli A.; Mancuso F.; Crupi V.; Supuran C.T.; Gitto R. (2024). Synthesis, biochemical screening and in-silico investigations of arylsulfonamides bearing linear and cyclic tails. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 113, pp. 0-0, ISSN:0960-894X DOI  

  Moi D.; Vittorio S.; Angeli A.; Supuran C.T.; Onnis V. (2024). Discovery of a New Class of 1-(4-Sulfamoylbenzoyl)piperidine-4-carboxamides as Human Carbonic Anhydrase Inhibitors. ACS MEDICINAL CHEMISTRY LETTERS, vol. 15, pp. 470-477, ISSN:1948-5875 DOI  

  Singh P.; Nerella S.G.; Swain B.; Angeli A.; Ullah Q.; Supuran C.T.; Arifuddin M. (2024). Design, synthesis and in vitro evaluation of novel thiazole-coumarin hybrids as selective and potent human carbonic anhydrase IX and XII inhibitors. INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, vol. 268, pp. 0-0, ISSN:0141-8130 DOI  

  Palomba M.; Angeli A.; Galdini R.; Hughineata A.J.; Perin G.; Lenardao E.J.; Marini F.; Santi C.; Supuran C.T.; Bagnoli L. (2024). Iodine/Oxone® oxidative system for the synthesis of selenylindoles bearing a benzenesulfonamide moiety as carbonic anhydrase I, II, IX, and XII inhibitors. ORGANIC & BIOMOLECULAR CHEMISTRY, vol. 22, pp. 6532-6542, ISSN:1477-0520 DOI  

  Giampietro L.; Marinacci B.; Della Valle A.; D'Agostino I.; Lauro A.; Mori M.; Carradori S.; Ammazzalorso A.; De Filippis B.; Maccallini C.; Angeli A.; Capasso C.; Francati S.; Mollica A.; Grande R.; Supuran C.T. (2024). Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori: Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies. PHARMACEUTICALS, vol. 17, pp. 0-0, ISSN:1424-8247 DOI  

  Denner T.C.; Heise N.V.; Serbian I.; Angeli A.; Supuran C.T.; Csuk R. (2024). An asiatic acid derived trisulfamate acts as a nanomolar inhibitor of human carbonic anhydrase VA. STEROIDS, vol. 205, pp. 0-0, ISSN:0039-128X DOI  

  Maier S.S.; Pinteala M.; Angeli A.; Supuran C.T. (2024). Self-assembling prodrugs. In: Stelian S. Maier, Mariana Pinteala, Andrea Angeli, Claudiu T. Supuran. Advances in Prodrugs: Design and Therapeutic Applications, pp. 113-151 Elsevier. DOI  

  Angeli, Andrea; Tanini, Damiano (2024). Photoactivatable prodrugs. In: Claudiu T. Supuran, A. Angeli, D. Tanini. Advances in Prodrugs: Design and Therapeutic Applications, pp. 73-95 Elsevier, ISBN:9780443156359. DOI  

  Giovannuzzi, Simone; Tanini, Damiano; Angeli, Andrea (2024). Prodrugs for cancer therapy. In: Claudiu T. Supuran, A. Angeli, D. Tanini. Advances in Prodrugs: Design and Therapeutic Applications, pp. 233-263 Elsevier, ISBN:9780443156359. DOI  

  Angeli A.; Ferraroni M.; Capasso C.; Supuran C.T. (2024). The dopamine D2 receptors antagonist Veralipride inhibits carbonic anhydrases: solution and crystallographic insights on human isoforms. CHEMISTRY - AN ASIAN JOURNAL, vol. 19, pp. 0-0, ISSN:1861-471X DOI   Accesso ONLINE all'editore

  Angeli, A.; De Luca, V.; Huang, X.; Winter, D.L.; Capasso, C.; Supuran, C.T.; Donald, W.A. (2024). Phosphorylation Strongly Affects the Inhibition of Human Carbonic Anhydrase ICO2 Hydration Activity. ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, pp. 0-0, ISSN:0003-9861 DOI  

  Shaldam M.A.; Abdulla M.-H.; Angeli A.; Hefny S.M.; El-labbad E.M.; Obeed A.B.; Alhassan N.S.; Supuran C.T.; Eldehna W.M.; Tawfik H.O. (2024). Novel sulfonamide-tethered Schiff bases as anti-proliferative agents with VEGFR-2 inhibitory activity: Synthesis, biological assessment, and molecular dynamic simulations. JOURNAL OF MOLECULAR STRUCTURE, vol. 1309, pp. 0-0, ISSN:0022-2860 DOI  

  Al-Matarneh, Cristina M.; Pinteala, Mariana; Nicolescu, Alina; Silion, Mihaela; Mocci, Francesca; Puf, Razvan; Angeli, Andrea; Ferraroni, Marta; Supuran, Claudiu T.; Zara, Susi; Carradori, Simone; Paoletti, Niccolò; Bonardi, Alessandro; Gratteri, Paola (2024). Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety. JOURNAL OF MEDICINAL CHEMISTRY, vol. 67, pp. 3018-3038, ISSN:0022-2623 DOI  

  Karchuganova E.; Martynova S.; Kalinin S.; Angeli A.; Dar'in D.; Vullo D.; Supuran C.T.; Bakulina O. (2024). Direct assembly of N-sulfamoyl lactam scaffolds bearing a zinc-binding group for inhibiting metalloenzymes based on desymmetrization of sulfamide and the Castagnoli-Cushman reaction. TETRAHEDRON, vol. 154, pp. 0-0, ISSN:0040-4020 DOI  

  D'Agostino I.; Bonardi A.; Ferraroni M.; Gratteri P.; Angeli A.; Supuran C.T. (2024). Exploring the Polypharmacological Potential of PCI-27483: A Selective Inhibitor of Carbonic Anhydrases IX and XII. ACS MEDICINAL CHEMISTRY LETTERS, vol. 15, pp. 2042-2045, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Giovannuzzi S.; Nikitjuka A.; Angeli A.; Smietana M.; Massardi M.-L.; Turati M.; Ronca R.; Bonardi A.; Nocentini A.; Ferraroni M.; Supuran C.T.; Winum J.-Y. (2024). Benzoxaborinine, New Chemotype for Carbonic Anhydrase Inhibition: Ex Novo Synthesis, Crystallography, In Silico Studies, and Anti-Melanoma Cell Line Activity. JOURNAL OF MEDICINAL CHEMISTRY, vol. 67, pp. 18221-18234, ISSN:1520-4804 DOI   Accesso ONLINE all'editore

  Hefny S.M.; El-Moselhy T.F.; El-Din N.; Ammara A.; Angeli A.; Ferraroni M.; El-Dessouki A.M.; Shaldam M.A.; Yahya G.; Al-Karmalawy A.A.; Supuran C.T.; Tawfik H.O. (2024). A new framework for novel analogues of pazopanib as potent and selective human carbonic anhydrase inhibitors: Design, repurposing rational, synthesis, crystallographic, in vivo and in vitro biological assessments. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 274, pp. 116527-116527, ISSN:1768-3254 DOI  

  Hakan Aslan; Gioele Renzi; Andrea Angeli; Ilaria D'Agostino; Roberto Ronca; Maria Luisa Massardi; Camilla Tavani; Simone Carradori; Marta Ferraroni; Paolo Governa; Fabrizio Manetti; Fabrizio Carta; Claudiu T. Supuran (2024). Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity. RSC MEDICINAL CHEMISTRY, vol. 15, pp. 1929-1941, ISSN:2632-8682 DOI   Accesso ONLINE all'editore

  Angeli A.; Occhini A.; Renzi G.; Capperucci A.; Ferraroni M.; Tanini D.; Supuran C.T. (2024). Thia- and Seleno-Michael Reactions for the Synthesis of Carbonic Anhydrases Inhibitors. CHEMMEDCHEM, pp. 0-0, ISSN:1860-7187 DOI   Accesso ONLINE all'editore

  Gumus A.; D'Agostino I.; Puca V.; Crocetta V.; Carradori S.; Cutarella L.; Mori M.; Carta F.; Angeli A.; Capasso C.; Supuran C.T. (2024). Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α-carbonic anhydrase inhibitors. ARCHIV DER PHARMAZIE, pp. 0-0, ISSN:0365-6233 DOI  

  De Luca, Viviana; Angeli, Andrea; Nocentini, Alessio; Gratteri, Paola; Pratesi, Silvia; Tanini, Damiano; Carginale, Vincenzo; Capperucci, Antonella; Supuran, Claudiu T.; Capasso, Clemente (2024). Leveraging SARS-CoV-2 Main Protease (Mpro) for COVID-19 Mitigation with Selenium-Based Inhibitors. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 25, pp. 0-0, ISSN:1422-0067 DOI  

  El-Malah, Afaf; Taher, Ehab S; Angeli, Andrea; Elbaramawi, Samar S; Mahmoud, Zeinab; Moustafa, Nour; Supuran, Claudiu T; Ibrahim, Tarek S (2023). Schiff bases as linker in the development of quinoline-sulfonamide hybrids as selective cancer-associated carbonic anhydrase isoforms IX/XII inhibitors: A new regioisomerism tactic. BIOORGANIC CHEMISTRY, vol. 131, pp. 106309-106309, ISSN:0045-2068 DOI  

  Angeli A.; Ferraroni M.; Bonardi A.; Supuran C.T.; Nocentini A. (2023). Diversely N-substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N-nitrosulfonamides. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 38, pp. 2178430-2178430, ISSN:1475-6366 DOI  

  D'Agostino I.; Zara S.; Carradori S.; De Luca V.; Capasso C.; Kocken C.H.M.; Zeeman A.-M.; Angeli A.; Carta F.; Supuran C.T. (2023). Antimalarial Agents Targeting Plasmodium falciparum Carbonic Anhydrase: Towards Artesunate Hybrid Compounds with Dual Mechanism of Action. CHEMMEDCHEM, pp. 0-0, ISSN:1860-7179 DOI  

  Angeli A.; Micheli L.; Turnaturi R.; Pasquinucci L.; Parenti C.; Alterio V.; Di Fiore A.; De Simone G.; Monti S.M.; Carta F.; Di Cesare Mannelli L.; Ghelardini C.; Supuran C.T. (2023). Discovery of a novel series of potent carbonic anhydrase inhibitors with selective affinity for μ Opioid receptor for Safer and long-lasting analgesia. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 260, pp. 0-0, ISSN:0223-5234 DOI  

  Mahammad Ghouse S.; Bahatam K.; Angeli A.; Pawar G.; Chinchilli K.K.; Yaddanapudi V.M.; Mohammed A.; Supuran C.T.; Nanduri S. (2023). Synthesis and biological evaluation of new 3-substituted coumarin derivatives as selective inhibitors of human carbonic anhydrase IX and XII. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 38, pp. 2185760-2185760, ISSN:1475-6366 DOI  

  Vats, Lalit; Siwach, Kiran; Angeli, Andrea; Bikal, Prerna; Bhardwaj, Jitender Kumar; Supuran, Claudiu T; Sharma, Pawan K (2023). Tail approach synthesis of triazolylthiazolotriazole bearing benzenesulfonamides as carbonic anhydrase inhibitors capable of inducing apoptosis. ARCHIV DER PHARMAZIE, vol. 356, pp. 0-0, ISSN:0365-6233 DOI  

  Maria Giulia Davighi, Camilla Matassini, Andrea Goti, Marta Ferraroni, Andrea Angeli, Claudiu T. Supuran, Francesca Cardona (2023). Mono- and three-tailed sugar and iminosugar decorated benzenesulfonamide carbonic anhydrase inhibitors. ORGANIC & BIOMOLECULAR CHEMISTRY, vol. 2023, pp. 1-13, ISSN:1477-0520 DOI   Accesso ONLINE all'editore

  Haapanen S.; Angeli A.; Tolvanen M.; Emameh R.Z.; Supuran C.T.; Parkkila S. (2023). Cloning, characterization, and inhibition of the novel β-carbonic anhydrase from parasitic blood fluke, Schistosoma mansoni. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 38, pp. 2184299-2184299, ISSN:1475-6366 DOI  

  Zengin Kurt B.; Celebi G.; Ozturk Civelek D.; Angeli A.; Akdemir A.; Sonmez F.; Supuran C.T. (2023). Tail-Approach-Based Design and Synthesis of Coumarin-Monoterpenes as Carbonic Anhydrase Inhibitors and Anticancer Agents. ACS OMEGA, vol. 8, pp. 5787-5807, ISSN:2470-1343 DOI  

  Marialuigia Fantacuzzi; Ilaria D’Agostino; Simone Carradori; Francesco Liguori; Fabrizio Carta; Mariangela Agamennone; Andrea Angeli; Filomena Sannio; Jean-Denis Docquier; Clemente Capasso; Claudiu T. Supuran (2023). Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 38, pp. 0-0, ISSN:1475-6366 DOI  

  Astrain-Redin N.; Paoletti N.; Plano D.; Bonardi A.; Gratteri P.; Angeli A.; Sanmartin C.; Supuran C.T. (2023). Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 38, pp. 2191165-2191165, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  Sharma, Vikas; Kumar, Rajiv; Angeli, Andrea; Supuran, Claudiu T; Sharma, Pawan K (2023). Benzenesulfonamides with trisubstituted triazole motif as selective carbonic anhydrase I, II, IV, and IX inhibitors. ARCHIV DER PHARMAZIE, vol. 356, pp. 0-0, ISSN:0365-6233 DOI  

  Angeli A.; Micheli L.; Carta F.; Ferraroni M.; Pirali T.; Fernandez Carvajal A.; Ferrer Montiel A.; Di Cesare Mannelli L.; Ghelardini C.; Supuran C.T. (2023). First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy. JOURNAL OF MEDICINAL CHEMISTRY, vol. 66, pp. 1616-1633, ISSN:0022-2623 DOI  

  Angeli A.; Supuran C.T. (2023). Click chemistry approaches for developing carbonic anhydrase inhibitors and their applications. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 38, pp. 2166503-2166503, ISSN:1475-6366 DOI  

  andrea angeli; Niccolò Paoletti; Claudiu Supuran (2023). Five-Membered Heterocyclic Sulfonamides as Carbonic Anhydrase Inhibitors. MOLECULES, vol. 28, pp. 3220-3220, ISSN:1420-3049 DOI  

  Fabrizio Carta; Andrea Angeli; Claudiu T Supuran; Silvia Selleri (2023). CARBAMOSELENOYL DERIVATIVES AS ANTI-INFECTIVE AGENTS. Numero: WO2023/073634 A1 Fabrizio Carta; Andrea Angeli; Silvia Selleri; Claudiu T Supuran; Silvia Clotilde Cabassi; Costanza Spadini

  Chinchilli K.K.; Singh P.; Swain B.; Goud N.S.; Sigalapalli D.K.; Choli A.; Angeli A.; Nanduri S.; Yaddanapudi V.M.; Supuran C.T.; Arifuddin M. (2023). Development of Novel Indole-3-sulfonamide-heteroaryl Hybrids as Carbonic Anhydrase Inhibitors: Design, Synthesis and in-vitro Screening. ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, vol. 23, pp. 1225-1233, ISSN:1871-5206 DOI  

  Sequeira L.; Distinto S.; Meleddu R.; Gaspari M.; Angeli A.; Cottiglia F.; Secci D.; Onali A.; Sanna E.; Borges F.; Uriarte E.; Alcaro S.; Supuran C.T.; Maccioni E. (2023). 2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 38, pp. 0-0, ISSN:1475-6366 DOI  

  Shaldam M.A.; Almahli H.; Angeli A.; Badi R.M.; Khaleel E.F.; Zain-Alabdeen A.I.; Elsayed Z.M.; Elkaeed E.B.; Salem R.; Supuran C.T.; Eldehna W.M.; Tawfik H.O. (2023). Discovery of sulfonamide-tethered isatin derivatives as novel anticancer agents and VEGFR-2 inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 38, pp. 0-0, ISSN:1475-6366 DOI  

  Chinchilli K.K.; Akunuri R.; Ghouse S.M.; Soujanya D.; Angeli A.; Parupalli R.; Arifuddin M.; Yaddanapudi V.M.; Supuran C.T.; Nanduri S. (2023). Design, synthesis, and structure–activity studies of new rhodanine derivatives as carbonic anhydrase II, IX inhibitors. ARCHIV DER PHARMAZIE, vol. 356, pp. 0-0, ISSN:0365-6233 DOI  

  Ricci F.; Angeli A.; Mancuso F.; De Luca L.; Supuran C.T.; Gitto R. (2023). Screening Campaign and Docking Investigations in Identifying New Hit Compounds as Inhibitors of Human Carbonic Anhydrases Expressed In Tumour Cells. CHEMMEDCHEM, vol. 18, pp. 0-0, ISSN:1860-7179 DOI  

  Ismail R.S.M.; El Kerdawy A.M.; Soliman D.H.; Georgey H.H.; Abdel Gawad N.M.; Angeli A.; Supuran C.T. (2023). Discovery of a new potent oxindole multi-kinase inhibitor among a series of designed 3-alkenyl-oxindoles with ancillary carbonic anhydrase inhibitory activity as antiproliferative agents. BMC CHEMISTRY, vol. 17, pp. 0-0, ISSN:2661-801X DOI  

  Gazzaroli G.; Angeli A.; Giacomini A.; Ronca R. (2023). Proteasome inhibitors as anticancer agents. EXPERT OPINION ON THERAPEUTIC PATENTS, vol. 33, pp. 775-796, ISSN:1354-3776 DOI  

  Melfi F.; Carradori S.; Angeli A.; D'Agostino I. (2023). Nature as a source and inspiration for human monoamine oxidase B (hMAO-B) inhibition: A review of the recent advances in chemical modification of natural compounds. EXPERT OPINION ON DRUG DISCOVERY, vol. 18, pp. 851-879, ISSN:1746-0441 DOI  

  Angeli A.; Kartsev V.; Petrou A.; Lichitsky B.; Komogortsev A.; Geronikaki A.; Supuran C.T. (2023). Substituted furan sulfonamides as carbonic anhydrase inhibitors: Synthesis, biological and in silico studies. BIOORGANIC CHEMISTRY, vol. 138, pp. 0-0, ISSN:0045-2068 DOI  

  Tinivella, Annachiara; Nwachukwu, Jerome C; Angeli, Andrea; Foschi, Francesca; Benatti, Anna Laura; Pinzi, Luca; Izard, Tina; Ferraroni, Marta; Erumbi, Rangarajan; Christodoulou, Michael S; Passarella, Daniele; Supuran, Claudiu T; Nettles, Kendall W; Rastelli, Giulio (2023). Design, synthesis, biological evaluation and crystal structure determination of dual modulators of carbonic anhydrases and estrogen receptors. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 246, pp. 115011-115011, ISSN:0223-5234 DOI  

  Carradori, Simone; Angeli, Andrea; Sfragano, Patrick S.; Yzeiri, Xheila; Calamante, Massimo; Tanini, Damiano; Capperucci, Antonella; Kunstek, Hannah; Varbanov, Mihayl; Capasso, Clemente; Supuran, Claudiu T. (2023). Photoactivatable Heptamethine-Based Carbonic Anhydrase Inhibitors Leading to New Anti-Antibacterial Agents. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 24, pp. 0-0, ISSN:1422-0067 DOI  

  Angeli A. (2023). Reverse transcriptase. Metalloenzymes, pp. 23-34 DOI  

  Moi D.; Vittorio S.; Angeli A.; Balboni G.; Supuran C.T.; Onnis V. (2023). Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors. MOLECULES, vol. 28, pp. 91-91, ISSN:1420-3049 DOI  

  Combs J.; Bozdag M.; Cravey L.D.; Kota A.; McKenna R.; Angeli A.; Carta F.; Supuran C.T. (2023). New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors. MOLECULES, vol. 28, pp. 890-890, ISSN:1420-3049 DOI  

  Angeli A.; Petrou A.; Kartsev V.; Lichitsky B.; Komogortsev A.; Capasso C.; Geronikaki A.; Supuran C.T. (2023). Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 24, pp. 2802-2802, ISSN:1661-6596 DOI  

  Denner T.C.; Angeli A.; Ferraroni M.; Supuran C.T.; Csuk R. (2023). Ureidobenzenesulfonamides as Selective Carbonic Anhydrase I, IX, and XII Inhibitors. MOLECULES, vol. 28, pp. 0-0, ISSN:1420-3049 DOI   Accesso ONLINE all'editore

  Aboukhatwa S.M.; Sidhom P.A.; Angeli A.; Supuran C.T.; Tawfik H.O. (2023). Terminators or Guardians? Design, Synthesis, and Cytotoxicity Profiling of Chalcone-Sulfonamide Hybrids. ACS OMEGA, vol. 8, pp. 7666-7683, ISSN:2470-1343 DOI  

  Andrea Angeli; Marta Ferraroni; Carlotta Granchi; Filippo Minutolo; Xiaozhuo Chen; Pratik Shriwas; Emilio Russo; Antonio Leo; Silvia Selleri; Fabrizio Carta; Claudiu T. Supuran (2023). First-in-Class Dual Targeting Compounds for the Management of Seizures in Glucose Transporter Type 1 Deficiency Syndrome. JOURNAL OF MEDICINAL CHEMISTRY, pp. 0-0, ISSN:0022-2623 DOI  

  De Luca V.; Angeli A.; Mazzone V.; Adelfio C.; Carginale V.; Scaloni A.; Carta F.; Selleri S.; Supuran C.T.; Capasso C. (2022). Heterologous expression and biochemical characterisation of the recombinant β-carbonic anhydrase (MpaCA) from the warm-blooded vertebrate pathogen malassezia pachydermatis. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 37, pp. 62-68, ISSN:1475-6366 DOI  

  Sharonova, Tatiana; Zhmurov, Petr; Kalinin, Stanislav; Nocentini, Alessio; Angeli, Andrea; Ferraroni, Marta; Korsakov, Mikhail; Supuran, Claudiu T; Krasavin, Mikhail (2022). Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 37, pp. 857-865-865, ISSN:1475-6366 DOI  

  Thacker P.S.; Mohammed A.; Supuran C.T.; Tiwari P.L.; Goud N.S.; Srikanth D.; Angeli A. (2022). Synthesis and Biological Evaluation of Coumarin Carboxamides as Selective and Potent Inhibitors of Carbonic Anhydrases IX and XII. ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, vol. 22, pp. 2647-2654, ISSN:1871-5206 DOI  

  Gustavo Provensi, Alessia Costa, Barbara Rani, Maria Vittoria Becagli, Fabio Vaiano, Maria Beatrice Passani, Damiano Tanini, Antonella Capperucci, Simone Carradori, Jacobus P Petzer, Anél Petzer, Daniela Vullo, Gabriele Costantino, Patrizio Blandina, Andrea Angeli, Claudiu T Supuran (2022). New β-arylchalcogeno amines with procognitive properties targeting Carbonic Anhydrases and Monoamine Oxidases. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 244, pp. 1-11, ISSN:0223-5234 DOI  

  Carradori, Simone; Fantacuzzi, Marialuigia; Ammazzalorso, Alessandra; Angeli, Andrea; De Filippis, Barbara; Galati, Salvatore; Petzer, Anél; Petzer, Jacobus P; Poli, Giulio; Tuccinardi, Tiziano; Agamennone, Mariangela; Supuran, Claudiu T (2022). Resveratrol Analogues as Dual Inhibitors of Monoamine Oxidase B and Carbonic Anhydrase VII: A New Multi-Target Combination for Neurodegenerative Diseases?. MOLECULES, vol. 27, pp. 7816-7816, ISSN:1420-3049 DOI  

  Agamennone, Mariangela; Fantacuzzi, Marialuigia; Carradori, Simone; Petzer, Anél; Petzer, Jacobus P; Angeli, Andrea; Supuran, Claudiu T; Luisi, Grazia (2022). Coumarin-Based Dual Inhibitors of Human Carbonic Anhydrases and Monoamine Oxidases Featuring Amino Acyl and (Pseudo)-Dipeptidyl Appendages: In Vitro and Computational Studies. MOLECULES, vol. 27, pp. 0-0, ISSN:1420-3049 DOI  

  Francesconi, Oscar; Corzana, Francisco; Kontogianni, Georgia-Ioanna; Pesciullesi, Giorgio; Gualdani, Roberta; Supuran, Claudiu T; Angeli, Andrea; Kavasi, Rafaela Maria; Chatzinikolaidou, Maria; Nativi, Cristina (2022). Lipoyl-Based Antagonists of Transient Receptor Potential Cation A (TRPA1) Downregulate Osteosarcoma Cell Migration and Expression of Pro-Inflammatory Cytokines. ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE, vol. 5, pp. 0-0, ISSN:2575-9108 DOI  

  Kumar R.; Kumar A.; Ram S.; Angeli A.; Bonardi A.; Nocentini A.; Gratteri P.; Supuran C.T.; Sharma P.K. (2022). Novel benzenesulfonamide-bearing pyrazoles and 1,2,4-thiadiazoles as selective carbonic anhydrase inhibitors. ARCHIV DER PHARMAZIE, vol. 355, pp. e2100241-e2100241, ISSN:0365-6233 DOI   Accesso ONLINE all'editore

  Tanini D.; Capperucci A.; Locuoco M.; Ferraroni M.; Costantino G.; Angeli A.; Supuran C.T. (2022). Benzoselenoates: A novel class of carbonic anhydrase inhibitors. BIOORGANIC CHEMISTRY, vol. 122, pp. 0-0, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Manzoor, Shoaib; Angeli, Andrea; Zara, Susi; Carradori, Simone; Rahman, Md Ataur; Raza, Md Kausar; Supuran, Claudiu T; Hoda, Nasimul (2022). Development of benzene and benzothiazole-sulfonamide analogues as selective inhibitors of the tumor-associated carbonic anhydrase IX. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 243, pp. 0-0, ISSN:0223-5234 DOI  

  Bozdag M.; Cravey L.; Combs J.; Kota A.; McKenna R.; Angeli A.; Selleri S.; Carta F.; Supuran C.T. (2022). Small Molecule Alkoxy Oriented Selectiveness on Human Carbonic Anhydrase II and IX Inhibition. CHEMMEDCHEM, vol. 17, pp. 0-0, ISSN:1860-7179 DOI  

  Gantner M.E.; Prada Gori D.N.; Llanos M.A.; Talevi A.; Angeli A.; Vullo D.; Supuran C.T.; Gavernet L. (2022). Identification of New Carbonic Anhydrase VII Inhibitors by Structure-Based Virtual Screening. JOURNAL OF CHEMICAL INFORMATION AND MODELING, vol. 62, pp. 4760-4770, ISSN:1549-9596 DOI  

  Nada H.; Elkamhawy A.; Abdellattif M.H.; Angeli A.; Lee C.H.; Supuran C.T.; Lee K. (2022). 4-Anilinoquinazoline-based benzenesulfonamides as nanomolar inhibitors of carbonic anhydrase isoforms I, II, IX, and XII: design, synthesis, in-vitro, and in-silico biological studies. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 37, pp. 994-1004, ISSN:1475-6366 DOI  

  Ferraroni M; Angeli A; Carradori S; Supuran CT (2022). Inhibition of Schistosoma mansoni carbonic anhydrase by the antiparasitic drug clorsulon: X-ray crystallographic and in vitro studies. ACTA CRYSTALLOGRAPHICA. SECTION D, STRUCTURAL BIOLOGY, vol. 78, pp. 321-327, ISSN:2059-7983 DOI  

  Micheli L.; Testai L.; Angeli A.; Carrino D.; Pacini A.; Margiotta F.; Flori L.; Supuran C.T.; Calderone V.; Ghelardini C.; Mannelli L.D.C. (2022). Inhibitors of Mitochondrial Human Carbonic Anhydrases VA and VB as a Therapeutic Strategy against Paclitaxel-Induced Neuropathic Pain in Mice. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 23, pp. 6229-6229, ISSN:1422-0067 DOI  

  Jimenez, Lucia; Mayoral-Varo, Victor; Amenábar, Carlos; Ortega, Judit; Sequeira, João G N; Machuqueiro, Miguel; Mourato, Cristiana; Silvestri, Romano; Angeli, Andrea; Carta, Fabrizio; Supuran, Claudiu T; Megías, Diego; Ferreira, Bibiana I; Link, Wolfgang (2022). Multiplexed cellular profiling identifies an organoselenium compound as an inhibitor of CRM1-mediated nuclear export. TRAFFIC, vol. 23, pp. 0-0, ISSN:1398-9219 DOI  

  Urbanski L.J.; Angeli A.; Mykuliak V.V.; Azizi L.; Kuuslahti M.; Hytonen V.P.; Supuran C.T.; Parkkila S. (2022). Biochemical and structural characterization of beta-carbonic anhydrase from the parasite Trichomonas vaginalis. JOURNAL OF MOLECULAR MEDICINE, vol. 100, pp. 115-124, ISSN:0946-2716 DOI  

  Mancuso F.; Angeli A.; De Luca V.; Bucolo F.; De Luca L.; Capasso C.; Supuran C.T.; Gitto R. (2022). Synthesis and biological evaluation of sulfonamide-based compounds as inhibitors of carbonic anhydrase from Vibrio cholerae. ARCHIV DER PHARMAZIE, vol. 355, pp. 2200070-2200070, ISSN:0365-6233 DOI  

  Siwach K.; Kumar A.; Panchal H.; Kumar R.; Bhardwaj J.K.; Angeli A.; Supuran C.T.; Sharma P.K. (2022). Selective inhibition of carbonic anhydrase IX by sulphonylated 1,2,3-triazole incorporated benzenesulphonamides capable of inducing apoptosis. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 37, pp. 1454-1463, ISSN:1475-6366 DOI  

  Pontecorvi V.; Mori M.; Picarazzi F.; Zara S.; Carradori S.; Cataldi A.; Angeli A.; Berrino E.; Chimenti P.; Ciogli A.; Secci D.; Guglielmi P.; Supuran C.T. (2022). Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 23, pp. 7950-7950, ISSN:1661-6596 DOI  

  Angeli A.; Ferraroni M.; Capperucci A.; Tanini D.; Costantino G.; Supuran C.T. (2022). Selenocarbamates As a Prodrug-Based Approach to Carbonic Anhydrase Inhibition. CHEMMEDCHEM, vol. 17, pp. e2022000085-0, ISSN:1860-7179 DOI   Accesso ONLINE all'editore

  Tawfik, Haytham O; Belal, Amany; Abourehab, Mohammed A S; Angeli, Andrea; Bonardi, Alessandro; Supuran, Claudiu T; El-Hamamsy, Mervat H (2022). Dependence on linkers' flexibility designed for benzenesulfonamides targeting discovery of novel hCA IX inhibitors as potent anticancer agents. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 37, pp. 0-0, ISSN:1475-6366 DOI  

  Petreni, Andrea; Iacobescu, Alexandra; Simionescu, Natalia; Petrovici, Anca-Roxana; Angeli, Andrea; Fifere, Adrian; Pinteala, Mariana; Supuran, Claudiu T (2022). Carbonic Anhydrase inhibitors bearing organotelluride moieties as novel agents for antitumor therapy. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 244, pp. 0-0, ISSN:0223-5234 DOI  

  Akgul O.; Lucarini E.; Mannelli L.D.C.; Ghelardini C.; D'Ambrosio K.; Buonanno M.; Monti S.M.; De Simone G.; Angeli A.; Supuran C.T.; Carta F. (2022). Sultam based Carbonic Anhydrase VII inhibitors for the management of neuropathic pain. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 227, pp. 0-0, ISSN:0223-5234 DOI  

  Havrankova E.; Garaj V.; Mascaretti S.; Angeli A.; Soldanova Z.; Kemka M.; Motycka J.; Brazdova M.; Csollei J.; Jampilek J.; Supuran C.T. (2022). Novel 1,3,5-triazinyl aminobenzenesulfonamides incorporating aminoalcohol, aminochalcone and aminostilbene structural motifs as potent anti-vre agents, and carbonic anhydrases i, ii, vii, ix, and xii inhibitors. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 23, pp. 231-231, ISSN:1661-6596 DOI  

  Zain-Alabdeen, Abdelrahman I; El-Moselhy, Tarek F; Sharafeldin, Nabaweya; Angeli, Andrea; Supuran, Claudiu T; El-Hamamsy, Mervat H (2022). Synthesis and anticancer activity of new benzensulfonamides incorporating s-triazines as cyclic linkers for inhibition of carbonic anhydrase IX. SCIENTIFIC REPORTS, vol. 12, pp. 0-0, ISSN:2045-2322 DOI  

  Yamali C; Sakagami H; Satoh K; Bandow K; Uesawa Y; Bua S; Angeli A; Supuran CT; Gul HI (2022). Investigation of carbonic anhydrase inhibitory effects and cytotoxicities of pyrazole-based hybrids carrying hydrazone and zinc-binding benzenesulfonamide pharmacophores. BIOORGANIC CHEMISTRY, vol. 127, pp. 105969-105969, ISSN:0045-2068 DOI  

  Moi D.; Deplano A.; Angeli A.; Balboni G.; Supuran C.T.; Onnis V. (2022). Synthesis of Sulfonamides Incorporating Piperidinyl-Hydrazidoureido and Piperidinyl-Hydrazidothioureido Moieties and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity. MOLECULES, vol. 27, pp. 5370-5370, ISSN:1420-3049 DOI  

  D'Agostino I.; Mathew G.E.; Angelini P.; Venanzoni R.; Angeles Flores G.; Angeli A.; Carradori S.; Marinacci B.; Menghini L.; Abdelgawad M.A.; Ghoneim M.M.; Mathew B.; Supuran C.T. (2022). Biological investigation of N-methyl thiosemicarbazones as antimicrobial agents and bacterial carbonic anhydrases inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 37, pp. 986-993, ISSN:1475-6366 DOI  

  Angeli A.; Kartsev V.; Petrou A.; Lichitsky B.; Komogortsev A.; Pinteala M.; Geronikaki A.; Supuran C.T. (2022). Pyrazolo[4,3-c]pyridine Sulfonamides as Carbonic Anhydrase Inhibitors: Synthesis, Biological and In Silico Studies. PHARMACEUTICALS, vol. 15, pp. 316-316, ISSN:1424-8247 DOI  

  Chiaramonte N.; Gabellini A.; Angeli A.; Bartolucci G.; Braconi L.; Dei S.; Teodori E.; Supuran C.T.; Romanelli M.N. (2022). New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I Activators. MOLECULES, vol. 27, pp. 0-0, ISSN:1420-3049 DOI  

  Kumar A.; Siwach K.; Rom T.; Kumar R.; Angeli A.; Kumar Paul A.; Supuran C.T.; Sharma P.K. (2022). Tail-approach based design and synthesis of Arylthiazolylhydrazono-1,2,3-triazoles incorporating sulfanilamide and metanilamide as human carbonic anhydrase I, II, IV and IX inhibitors. BIOORGANIC CHEMISTRY, vol. 123, pp. 105764-105764, ISSN:0045-2068 DOI  

  Thacker P.S.; Newaskar V.; Angeli A.; Sigalapalli D.K.; Goud N.S.; Chirra H.; Shaik A.B.; Arifuddin M.; Supuran C.T. (2022). Synthesis and biological evaluation of coumarin-thiazole hybrids as selective carbonic anhydrase IX and XII inhibitors. ARCHIV DER PHARMAZIE, vol. 355, pp. 2200232-2200232, ISSN:0365-6233 DOI  

  Elkamhawy A.; Woo J.; Nada H.; Angeli A.; Bedair T.M.; Supuran C.T.; Lee K. (2022). Identification of Novel and Potent Indole-Based Benzenesulfonamides as Selective Human Carbonic Anhydrase II Inhibitors: Design, Synthesis, In Vitro, and In Silico Studies. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 23, pp. 2540-2540, ISSN:1661-6596 DOI  

  Singh P.; Sridhar Goud N.; Swain B.; Kumar Sahoo S.; Choli A.; Angeli A.; Singh Kushwah B.; Madhavi Yaddanapudi V.; Supuran C.T.; Arifuddin M. (2022). Synthesis of a new series of quinoline/pyridine indole-3-sulfonamide hybrids as selective carbonic anhydrase IX inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 70, pp. 128809-128809, ISSN:0960-894X DOI  

  Urbanski L.J.; Bua S.; Angeli A.; Emameh R.Z.; Barker H.R.; Kuuslahti M.; Hytonen V.P.; Parkkila S.; Supuran C.T. (2022). The production and biochemical characterization of α-carbonic anhydrase from Lactobacillus rhamnosus GG. APPLIED MICROBIOLOGY AND BIOTECHNOLOGY, vol. 106, pp. 4065-4074, ISSN:0175-7598 DOI  

  Swain B.; Sahoo S.K.; Singh P.; Angeli A.; Yaddanapudi V.M.; Supuran C.T.; Arifuddin M. (2022). Exploration of 2-phenylquinoline-4-carboxamide linked benzene sulfonamide derivatives as isoform selective inhibitors of transmembrane human carbonic anhydrases. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 234, pp. 114247-114247, ISSN:0223-5234 DOI  

  Singh P.; Choli A.; Swain B.; Angeli A.; Sahoo S.K.; Yaddanapudi V.M.; Supuran C.T.; Arifuddin M. (2022). Design and development of novel series of indole-3-sulfonamide ureido derivatives as selective carbonic anhydrase II inhibitors. ARCHIV DER PHARMAZIE, vol. 355, pp. 2100333-2100333, ISSN:0365-6233 DOI  

  Ferraroni M.; Angeli A.; Pinteala M.; Supuran C.T. (2022). Sulfonamide diuretic azosemide as an efficient carbonic anhydrase inhibitor. JOURNAL OF MOLECULAR STRUCTURE, vol. 1268, pp. 0-0, ISSN:0022-2860 DOI  

  Eysteinsson T.; Garcia-Llorca A.; Angeli A.; Supuran C.T.; Carta F. (2022). Vasodilation of Pre-contracted Porcine Retinal Arteries by Carbonic Anhydrase Inhibitors with Enhanced Lipophilicity. CURRENT EYE RESEARCH, vol. 47, pp. 1615-1621, ISSN:0271-3683 DOI  

  Angeli A.; Ferraroni M.; Carta F.; Haberli C.; Keiser J.; Costantino G.; Supuran C.T. (2022). Development of Praziquantel sulphonamide derivatives as antischistosomal drugs. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 37, pp. 1479-1494, ISSN:1475-6366 DOI  

  Angeli A.; Velluzzi A.; Selleri S.; Capasso C.; Spadini C.; Iannarelli M.; Cabassi C.S.; Carta F.; Supuran C.T. (2022). Seleno Containing Compounds as Potent and Selective Antifungal Agents. ACS INFECTIOUS DISEASES, vol. 8, pp. 1905-1919, ISSN:2373-8227 DOI  

  Chiaramonte N.; Angeli A.; Sgambellone S.; Bonardi A.; Nocentini A.; Bartolucci G.; Braconi L.; Dei S.; Lucarini L.; Teodori E.; Gratteri P.; Wunsch B.; Supuran C.T.; Romanelli M.N. (2022). 2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 228, pp. 0-0, ISSN:0223-5234 DOI  

  Angeli, Andrea; Urbański, Linda J; Capasso, Clemente; Parkkila, Seppo; Supuran, Claudiu T (2022). Activation studies with amino acids and amines of a β-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri previously annotated as Staphylococcus aureus (SauBCA) carbonic anhydrase. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 37, pp. 0-0, ISSN:1475-6366 DOI  

  Artasensi, Angelica; Angeli, Andrea; Lammi, Carmen; Bollati, Carlotta; Gervasoni, Silvia; Baron, Giovanna; Matucci, Rosanna; Supuran, Claudiu T; Vistoli, Giulio; Fumagalli, Laura (2022). Discovery of a Potent and Highly Selective Dipeptidyl Peptidase IV and Carbonic Anhydrase Inhibitor as "Antidiabesity" Agents Based on Repurposing and Morphing of WB-4101. JOURNAL OF MEDICINAL CHEMISTRY, vol. 65, pp. 0-0, ISSN:0022-2623 DOI  

  Gumus A.; Bozdag M.; Akdemir A.; Angeli A.; Selleri S.; Carta F.; Supuran C.T. (2022). Thiosemicarbazide-Substituted Coumarins as Selective Inhibitors of the Tumor Associated Human Carbonic Anhydrases IX and XII. MOLECULES, vol. 27, pp. 0-0, ISSN:1420-3049 DOI  

  Singh P.; Kumar Sigalapalli D.; Sridhar Goud N.; Swain B.; Kumar Sahoo S.; Angeli A.; Shaik A.B.; Madhavi Yaddanapudi V.; Supuran C.T.; Arifuddin M. (2022). Ureidosulfocoumarin Derivatives As Selective and Potent Carbonic Anhydrase IX and XII Inhibitors. CHEMMEDCHEM, vol. 17, pp. 202100725-202100725, ISSN:1860-7179 DOI  

  Pena L.; Jimenez C.; Arancibia R.; Angeli A.; Supuran C.T. (2022). Heterobimetallic complexes containing organometallic acylhydrazone ligands as potential inhibitors of human carbonic anhydrases. JOURNAL OF INORGANIC BIOCHEMISTRY, vol. 232, pp. 111814-111814, ISSN:0162-0134 DOI  

  Swain B.; Singh P.; Angeli A.; Sahoo S.K.; Yaddanapudi V.M.; Supuran C.T.; Arifuddin M. (2022). Efficient One-pot Synthesis of 3,3-di(indolyl)indolin-2-ones from Isatin and Indole Catalyzed by VOSO4 as Non-Sulfonamide Carbonic Anhydrase Inhibitors. ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, vol. 22, pp. 2358-2366, ISSN:1871-5206 DOI  

  Chinchilli K.K.; Royyala V.N.; Thacker P.S.; Angeli A.; Danaboina S.; Singh P.; Nanduri S.; Supuran C.T.; Arifuddin M. (2022). Design, synthesis, SAR, and biological evaluation of saccharin-based hybrids as carbonic anhydrase inhibitors. ARCHIV DER PHARMAZIE, vol. 355, pp. 2200019-2200019, ISSN:0365-6233 DOI  

  Paloukopoulou C.; Govari S.; Soulioti A.; Stefanis I.; Angeli A.; Matheeussen A.; Capasso C.; Cos P.; Supuran C.T.; Karioti A. (2022). Phenols from Origanum dictamnus L. and Thymus vulgaris L. and their activity against Malassezia globosa carbonic anhydrase. NATURAL PRODUCT RESEARCH, vol. 36, pp. 1558-1564, ISSN:1478-6419 DOI  

  Erigur E.C.; Altug C.; Angeli A.; Supuran C.T. (2022). Design, synthesis and human carbonic anhydrase I, II, IX and XII inhibitory properties of 1,3-thiazole sulfonamides. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 59, pp. 128581-128581, ISSN:0960-894X DOI  

  Sbravati D.; Bonardi A.; Bua S.; Angeli A.; Ferraroni M.; Nocentini A.; Casnati A.; Gratteri P.; Sansone F.; Supuran C.T. (2022). Calixarenes Incorporating Sulfonamide Moieties: Versatile Ligands for Carbonic Anhydrases Inhibition. CHEMISTRY-A EUROPEAN JOURNAL, vol. 28, pp. 1-8, ISSN:0947-6539 DOI   Accesso ONLINE all'editore

  Swain, Baijayantimala; Khan, Abrar; Singh, Priti; Marde, Vaibhav S; Angeli, Andrea; Chinchilli, Krishna Kartheek; Yaddanapudi, Venkata Madhavi; Carradori, Simone; Supuran, Claudiu T; Arifuddin, Mohammed (2022). Design, Synthesis and Biological Assessment of Rhodanine-Linked Benzenesulfonamide Derivatives as Selective and Potent Human Carbonic Anhydrase Inhibitors. MOLECULES, vol. 27, pp. 8028-8028, ISSN:1420-3049 DOI  

  Andrea Angeli; Marta Ferraroni; Akram A. Da’dara; Silvia Selleri; Mariana Pinteala; Fabrizio Carta; Patrick J. Skelly; Claudiu T. Supuran (2021). Structural Insights into Schistosoma mansoni Carbonic Anhydrase (SmCA) Inhibition by Selenoureido-Substituted Benzenesulfonamides. JOURNAL OF MEDICINAL CHEMISTRY, pp. 0-0, ISSN:0022-2623 DOI  

  Eldeeb A.H.; Abo-Ashour M.F.; Angeli A.; Bonardi A.; Lasheen D.S.; Elrazaz E.Z.; Nocentini A.; Gratteri P.; Abdel-Aziz H.A.; Supuran C.T. (2021). Novel benzenesulfonamides aryl and arylsulfone conjugates adopting tail/dual tail approaches: Synthesis, carbonic anhydrase inhibitory activity and molecular modeling studies. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 221, pp. 113486-113509, ISSN:0223-5234 DOI   Accesso ONLINE all'editore

  Plyasova A.A.; Berrino E.; Khan I.I.; Veselovsky A.V.; Pokrovsky V.S.; Angeli A.; Ferraroni M.; Supuran C.T.; Pokrovskaya M.V.; Alexandrova S.S.; Gladilina Y.A.; Sokolov N.N.; Hilal A.; Carta F.; Zhdanov D.D. (2021). Mechanisms of the Antiproliferative and Antitumor Activity of Novel Telomerase-Carbonic Anhydrase Dual-Hybrid Inhibitors. JOURNAL OF MEDICINAL CHEMISTRY, vol. 64, pp. 11432-11444, ISSN:0022-2623 DOI  

  Gumus A.; Bozdag M.; Angeli A.; Peat T.S.; Carta F.; Supuran C.T.; Selleri S. (2021). Privileged scaffolds in medicinal chemistry: Studies on pyrazolo[1,5-a]pyrimidines on sulfonamide containing Carbonic Anhydrase inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 49, pp. 0-0, ISSN:0960-894X DOI  

  Akgul O.; Angeli A.; Selleri S.; Capasso C.; Supuran C.T.; Carta F. (2021). Taurultams incorporating arylsulfonamide: First in vitro inhibition studies of α-, β- and γ-class Carbonic Anhydrases from Vibrio cholerae and Burkholderia pseudomallei. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 219, pp. 0-0, ISSN:0223-5234 DOI  

  Angeli A.; Pinteala M.; Maier S.S.; Toti A.; Di Cesare Mannelli L.; Ghelardini C.; Selleri S.; Carta F.; Supuran C.T. (2021). Tellurides bearing benzensulfonamide as carbonic anhydrase inhibitors with potent antitumor activity. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 45, pp. 0-0, ISSN:0960-894X DOI  

  Biagiotti G.; Angeli A.; Giacomini A.; Toniolo G.; Landini L.; Salerno G.; Di Cesare Mannelli L.; Ghelardini C.; Mello T.; Mussi S.; Ravelli C.; Marelli M.; Cicchi S.; Menna E.; Ronca R.; Supuran C.T.; Richichi B. (2021). Glyco-Coated CdSe/ZnS Quantum Dots as Nanoprobes for Carbonic Anhydrase IX Imaging in Cancer Cells. ACS APPLIED NANO MATERIALS, vol. 4, pp. 14153-14160, ISSN:2574-0970 DOI   Accesso ONLINE all'editore

  Yamali C.; Inci Gul H.; Ozli G.; Angeli A.; Ballar Kirmizibayrak P.; Erbaykent Tepedelen B.; Sakagami H.; Bua S.; Supuran C.T. (2021). Exploring of tumor-associated carbonic anhydrase isoenzyme IX and XII inhibitory effects and cytotoxicities of the novel N-aryl-1-(4-sulfamoylphenyl)-5-(thiophen-2-yl)-1H-pyrazole-3-carboxamides. BIOORGANIC CHEMISTRY, vol. 115, pp. 105194-105194, ISSN:0045-2068 DOI  

  Mancuso F.; De Luca L.; Bucolo F.; Vrabel M.; Angeli A.; Capasso C.; Supuran C.T.; Gitto R. (2021). 4-Sulfamoylphenylalkylamides as Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae. CHEMMEDCHEM, vol. 16, pp. 3787-3794, ISSN:1860-7179 DOI  

  Swain B.; Aashritha K.; Singh P.; Angeli A.; Kothari A.; Sigalapalli D.K.; Yaddanapudi V.M.; Supuran C.T.; Arifuddin M. (2021). Design and synthesis of benzenesulfonamide-linked imidazo[2,1-b][1,3,4]thiadiazole derivatives as carbonic anhydrase I and II inhibitors. ARCHIV DER PHARMAZIE, vol. 354, pp. 2100028-2100028, ISSN:0365-6233 DOI  

  Berrino E.; Carradori S.; Angeli A.; Carta F.; Supuran C.T.; Guglielmi P.; Coletti C.; Paciotti R.; Schweikl H.; Maestrelli F.; Cerbai E.; Gallorini M. (2021). Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages. ANTIOXIDANTS, vol. 10, pp. 1-24, ISSN:2076-3921 DOI  

  Angeli A.; Carta F.; Nocentini A.; Winum J.-Y.; Zalubovskis R.; Onnis V.; Eldehna W.M.; Capasso C.; Carradori S.; Donald W.A.; Dedhar S.; Supuran C.T. (2021). Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors. BIOPHYSICAL JOURNAL, vol. 120, pp. 178-181, ISSN:0006-3495 DOI  

  Lenci E.; Angeli A.; Calugi L.; Innocenti R.; Carta F.; Supuran C.T.; Trabocchi A. (2021). Multitargeting application of proline-derived peptidomimetics addressing cancer-related human matrix metalloproteinase 9 and carbonic anhydrase II. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 214, pp. 0-0, ISSN:0223-5234 DOI  

  Angeli A.; Berrino E.; Carradori S.; Supuran C.T.; Cirri M.; Carta F.; Costantino G. (2021). Amine-and amino acid-based compounds as carbonic anhydrase activators. MOLECULES, vol. 26, pp. 0-0, ISSN:1420-3049 DOI  

  Angeli A.; Kartsev V.; Petrou A.; Pinteala M.; Vydzhak R.M.; Panchishin S.Y.; Brovarets V.; De Luca V.; Capasso C.; Geronikaki A.; Supuran C.T. (2021). New sulfanilamide derivatives incorporating heterocyclic carboxamide moieties as carbonic anhydrase inhibitors. PHARMACEUTICALS, vol. 14, pp. 828-828, ISSN:1424-8247 DOI  

  Chandra K.M.; Goud N.S.; Arifuddin M.; Alvala M.; Alvala R.; Angeli A.; Supuran C.T. (2021). Synthesis and biological evaluation of novel 4,7-disubstituted coumarins as selective tumor-associated carbonic anhydrase IX and XII inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 39, pp. 127877-127877, ISSN:0960-894X DOI  

  Singh P.; Purnachander Yadav P.; Swain B.; Thacker P.S.; Angeli A.; Supuran C.T.; Arifuddin M. (2021). Discovery of a novel series of indolylchalcone-benzenesulfonamide hybrids acting as selective carbonic anhydrase II inhibitors. BIOORGANIC CHEMISTRY, vol. 108, pp. 104647-104647, ISSN:0045-2068 DOI  

  Angeli A.; Kartsev V.; Petrou A.; Pinteala M.; Brovarets V.; Slyvchuk S.; Pilyo S.; Geronikaki A.; Supuran C.T. (2021). Chromene-containing aromatic sulfonamides with carbonic anhydrase inhibitory properties. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 22, pp. 5082-5082, ISSN:1661-6596 DOI  

  Cakmak E.B.; Zengin Kurt B.; Ozturk Civelek D.; Angeli A.; Akdemir A.; Sonmez F.; Supuran C.T.; Kucukislamoglu M. (2021). Quinoline-sulfamoyl carbamates/sulfamide derivatives: Synthesis, cytotoxicity, carbonic anhydrase activity, and molecular modelling studies. BIOORGANIC CHEMISTRY, vol. 110, pp. 104778-104778, ISSN:0045-2068 DOI  

  Mishra C.B.; Kumari S.; Angeli A.; Bua S.; Mongre R.K.; Tiwari M.; Supuran C.T. (2021). Discovery of Potent Carbonic Anhydrase Inhibitors as Effective Anticonvulsant Agents: Drug Design, Synthesis, and in Vitro and in Vivo Investigations. JOURNAL OF MEDICINAL CHEMISTRY, vol. 64, pp. 3100-3114, ISSN:0022-2623 DOI  

  Swain B.; Abhay; Singh P.; Angeli A.; Aashritha K.; Nagesh N.; Supuran C.T.; Arifuddin M. (2021). 3-Functionalised benzenesulphonamide based 1,3,4-oxadiazoles as selective carbonic anhydrase XIII inhibitors: Design, synthesis and biological evaluation. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 37, pp. 127856-127856, ISSN:0960-894X DOI  

  Angeli A.; Kartsev V.; Petrou A.; Pinteala M.; Brovarets V.; Vydzhak R.; Panchishin S.; Geronikaki A.; Supuran C.T. (2021). Carbonic anhydrase inhibition with sulfonamides incorporating pyrazole-and pyridazinecarboxamide moieties provides examples of isoform-selective inhibitors. MOLECULES, vol. 26, pp. 7023-7023, ISSN:1420-3049 DOI  

  Urbanski L.J.; Angeli A.; Hytonen V.P.; Di Fiore A.; De Simone G.; Parkkila S.; Supuran C.T. (2021). Inhibition of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with sulphonamides. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 36, pp. 329-334, ISSN:1475-6366 DOI  

  Meleddu R.; Deplano S.; Maccioni E.; Ortuso F.; Cottiglia F.; Secci D.; Onali A.; Sanna E.; Angeli A.; Angius R.; Alcaro S.; Supuran C.T.; Distinto S. (2021). Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 36, pp. 685-692, ISSN:1475-6366 DOI  

  Thacker P.S.; Tiwari P.L.; Angeli A.; Srikanth D.; Swain B.; Arifuddin M.; Supuran C.T. (2021). Synthesis and biological evaluation of coumarin-linked 4-anilinomethyl-1,2,3-triazoles as potent inhibitors of carbonic anhydrases ix and xiii involved in tumorigenesis. METABOLITES, vol. 11, pp. 225-225, ISSN:2218-1989 DOI  

  Grande R.; Carradori S.; Puca V.; Vitale I.; Angeli A.; Nocentini A.; Bonardi A.; Gratteri P.; Lanuti P.; Bologna G.; Simeone P.; Capasso C.; De Luca V.; Supuran C.T. (2021). Selective inhibition of helicobacter pylori carbonic anhydrases by carvacrol and thymol could impair biofilm production and the release of outer membrane vesicles. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 22, pp. 11583-11603, ISSN:1422-0067 DOI   Accesso ONLINE all'editore

  De Luca V.; Angeli A.; Mazzone V.; Adelfio C.; Carta F.; Selleri S.; Carginale V.; Scaloni A.; Supuran C.T.; Capasso C. (2021). Inhibitory effects of sulfonamide derivatives on the β‐carbonic anhydrase (Mpaca) from malassezia pachydermatis, a commensal, pathogenic fungus present in domestic animals. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 22, pp. 0-0, ISSN:1422-0067 DOI  

  Vannozzi G.; Vullo D.; Angeli A.; Ferraroni M.; Combs J.; Lomelino C.; Andring J.; Mckenna R.; Bartolucci G.; Pallecchi M.; Lucarini L.; Sgambellone S.; Masini E.; Carta F.; Supuran C.T. (2021). One-Pot Procedure for the Synthesis of Asymmetric Substituted Ureido Benzene Sulfonamides as Effective Inhibitors of Carbonic Anhydrase Enzymes. JOURNAL OF MEDICINAL CHEMISTRY, vol. 65, pp. 824-837, ISSN:0022-2623 DOI  

  Mancuso F.; Di Fiore A.; De Luca L.; Angeli A.; De Simone G.; Supuran C.T.; Gitto R. (2021). Design, synthesis and biochemical evaluation of novel carbonic anhydrase inhibitors triggered by structural knowledge on hCA VII. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 44, pp. 116279-116279, ISSN:0968-0896 DOI  

  Barresi E.; Ravichandran R.; Germelli L.; Angeli A.; Baglini E.; Salerno S.; Marini A.M.; Costa B.; Da Pozzo E.; Martini C.; Da Settimo F.; Supuran C.; Cosconati S.; Taliani S. (2021). Carbonic anhydrase activation profile of indole-based derivatives. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 36, pp. 1783-1797, ISSN:1475-6366 DOI  

  Angeli A.; Urbanski L.J.; Hytonen V.P.; Parkkila S.; Supuran C.T. (2021). Activation of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with amines and amino acids. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 36, pp. 758-763, ISSN:1475-6366 DOI  

  Yamali C.; Sakagami H.; Uesawa Y.; Kurosaki K.; Satoh K.; Masuda Y.; Yokose S.; Ece A.; Bua S.; Angeli A.; Supuran C.T.; Gul H.I. (2021). Comprehensive study on potent and selective carbonic anhydrase inhibitors: Synthesis, bioactivities and molecular modelling studies of 4-(3-(2-arylidenehydrazine-1-carbonyl)-5-(thiophen-2-yl)-1H-pyrazole-1-yl) benzenesulfonamides. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 217, pp. 113351-113351, ISSN:0223-5234 DOI  

  Salerno S.; Amendola G.; Angeli A.; Baglini E.; Barresi E.; Marini A.M.; Ravichandran R.; Viviano M.; Castellano S.; Novellino E.; Da Settimo F.; Supuran C.T.; Cosconati S.; Taliani S. (2021). Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 220, pp. 113490-113490, ISSN:0223-5234 DOI  

  Thacker P.S.; Srikanth D.; Angeli A.; Singh P.; Chinchilli K.K.; Arifuddin M.; Supuran C.T. (2021). Coumarin-Thiourea Hybrids Show Potent Carbonic Anhydrase IX and XIII Inhibitory Action. CHEMMEDCHEM, vol. 16, pp. 1252-1256, ISSN:1860-7179 DOI  

  Tanini D.; Carradori S.; Capperucci A.; Lupori L.; Zara S.; Ferraroni M.; Ghelardini C.; Mannelli L.D.C.; Micheli L.; Lucarini E.; Carta F.; Angeli A.; Supuran C.T. (2021). Chalcogenides-incorporating carbonic anhydrase inhibitors concomitantly reverted oxaliplatin-induced neuropathy and enhanced antiproliferative action. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 225, pp. 0-0, ISSN:0223-5234 DOI  

  Debora Pratesi, Andrea Sodini, Camilla Matassini, Francesca Cardona, Andrea Angeli, Fabrizio Carta, Marta Ferraroni, Claudiu T. Supuran, Andrea Goti (2021). Synthesis of Azasugar–Sulfonamide conjugates and their Evaluation as Inhibitors of Carbonic Anhydrases: the Azasugar Approach to Selectivity. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. 2021, pp. 2604-2614, ISSN:1099-0690 DOI  

  Nocentini, Alessio; Angeli, Andrea; Carta, Fabrizio; Winum, Jean-Yves; Zalubovskis, Raivis; Carradori, Simone; Capasso, Clemente; Donald, William A; Supuran, Claudiu T (2021). Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 36, pp. 561-580, ISSN:1475-6366 DOI  

  Kucukbay H.; Gonul Z.; Kucukbay F.Z.; Tekin Z.; Angeli A.; Bartolucci G.; Supuran C.T.; Tatlici E.; Apohan E.; Yesilada O. (2021). Synthesis of new 7-amino-3,4-dihydroquinolin-2(1H)-one-peptide derivatives and their carbonic anhydrase enzyme inhibition, antioxidant, and cytotoxic activities. ARCHIV DER PHARMAZIE, vol. 354, pp. 0-0, ISSN:0365-6233 DOI  

  Akgul O.; Angeli A.; Vullo D.; Carta F.; Supuran C.T. (2020). Unconventional amino acids in medicinal chemistry: First report on taurine merged within carbonic anhydrase inhibitors. BIOORGANIC CHEMISTRY, vol. 103, pp. 0-0, ISSN:0045-2068 DOI  

  Bozdag M.; Supuran C.T.; Esposito D.; Angeli A.; Carta F.; Monti S.M.; De Simone G.; Alterio V. (2020). 2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site. CHEMICAL COMMUNICATIONS, vol. 56, pp. 8297-8300, ISSN:1359-7345 DOI  

  Angeli A.; Carta F.; Supuran C.T. (2020). Carbonic anhydrases: Versatile and useful biocatalysts in chemistry and biochemistry. CATALYSTS, vol. 10, pp. 1-11, ISSN:2073-4344 DOI  

  Clima L.; Craciun B.F.; Angeli A.; Petreni A.; Bonardi A.; Nocentini A.; Carta F.; Gratteri P.; Pinteala M.; Supuran C.T. (2020). Synthesis, Computational Studies and Assessment of in Vitro Activity of Squalene Derivatives as Carbonic Anhydrase Inhibitors. CHEMMEDCHEM, vol. 15, pp. 2052-2057, ISSN:1860-7179 DOI  

  Del Prete, Sonia; Angeli, Andrea; Ghobril, Cynthia; Hitce, Julien; Clavaud, Cécile; Marat, Xavier; Supuran, Claudiu T; Capasso, Clemente (2020). Sulfonamide Inhibition Profile of the β-Carbonic Anhydrase from Malassezia restricta, An Opportunistic Pathogen Triggering Scalp Conditions. METABOLITES, vol. 10, pp. 39-39, ISSN:2218-1989 DOI  

  Fois, Benedetta; Distinto, Simona; Meleddu, Rita; Deplano, Serenella; Maccioni, Elias; Floris, Costantino; Rosa, Antonella; Nieddu, Mariella; Caboni, Pierluigi; Sissi, Claudia; Angeli, Andrea; Supuran, Claudiu T; Cottiglia, Filippo (2020). Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 539-548-548, ISSN:1475-6366 DOI  

  Angeli, Andrea; Pinteala, Mariana; Maier, Stelian S; Simionescu, Bogdan C; Milaneschi, Andrea; Abbas, Ghulam; Del Prete, Sonia; Capasso, Clemente; Capperucci, Antonella; Tanini, Damiano; Carta, Fabrizio; Supuran, Claudiu T (2020). Evaluation of Thio- and Seleno-Acetamides Bearing Benzenesulfonamide as Inhibitor of Carbonic Anhydrases from Different Pathogenic Bacteria. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 21, pp. 598-598, ISSN:1422-0067 DOI  

  Angeli A.; Pinteala M.; Maier S.S.; Simionescu B.C.; Da'dara A.A.; Skelly P.J.; Supuran C.T. (2020). Sulfonamide inhibition studies of an α-carbonic anhydrase from Schistosoma mansoni, a platyhelminth parasite responsible for schistosomiasis. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 21, pp. 1842-1850, ISSN:1661-6596 DOI  

  Krasavin M.; Kalinin S.; Zozulya S.; Gryniukova A.; Borysko P.; Angeli A.; Supuran C.T. (2020). Screening of benzenesulfonamide in combination with chemically diverse fragments against carbonic anhydrase by differential scanning fluorimetry. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 306-310, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  Genah S.; Angeli A.; Supuran C.T.; Morbidelli L. (2020). Effect of Carbonic Anhydrase IX inhibitors on human endothelial cell survival. PHARMACOLOGICAL RESEARCH, vol. 159, pp. 104964-104964, ISSN:1043-6618 DOI  

  Angeli, Andrea; Etxebeste-Mitxeltorena, Mikel; Sanmartín, Carmen; Espuelas, Socorro; Moreno, Esther; Azqueta, Amaya; Parkkila, Seppo; Carta, Fabrizio; Supuran, Claudiu T (2020). Tellurides Bearing Sulfonamides as Novel Inhibitors of Leishmanial Carbonic Anhydrase with Potent Antileishmanial Activity. JOURNAL OF MEDICINAL CHEMISTRY, vol. 63, pp. 4306-4314, ISSN:0022-2623 DOI  

  Angeli A.; Ferraroni M.; Pinteala M.; Maier S.S.; Simionescu B.C.; Carta F.; Del Prete S.; Capasso C.; Supuran C.T. (2020). Crystal structure of a tetrameric type II β-carbonic anhydrase from the pathogenic bacterium burkholderia pseudomallei. MOLECULES, vol. 25, pp. 2269-2278, ISSN:1420-3049 DOI  

  Berrino E.; Angeli A.; Zhdanov D.D.; Kiryukhina A.P.; Milaneschi A.; De Luca A.; Bozdag M.; Carradori S.; Selleri S.; Bartolucci G.; Peat T.S.; Ferraroni M.; Supuran C.T.; Carta F. (2020). Azidothymidine "clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors. JOURNAL OF MEDICINAL CHEMISTRY, vol. 63, pp. 7392-7409, ISSN:0022-2623 DOI  

  Angeli A.; Peat T.S.; Selleri S.; Saleh Alfawaz Altamimi A.; Supuran C.T.; Carta F. (2020). X-ray crystallography of Epacadostat in adduct with Carbonic Anhydrase IX. BIOORGANIC CHEMISTRY, vol. 97, pp. 103669-103669, ISSN:0045-2068 DOI  

  Sharma V.; Kumar R.; Angeli A.; Supuran C.T.; Sharma P.K. (2020). Tail approach synthesis of novel benzenesulfonamides incorporating 1,3,4-oxadiazole hybrids as potent inhibitor of carbonic anhydrase I, II, IX, and XII isoenzymes. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 193, pp. 112219-112219, ISSN:0223-5234 DOI  

  Angeli, Andrea; Carta, Fabrizio; Donnini, Selene; Capperucci, Antonella; Ferraroni, Marta; Tanini, Damiano; Supuran, Claudiu T (2020). Selenolesterase enzyme activity of carbonic anhydrases. CHEMICAL COMMUNICATIONS, pp. 0-0, ISSN:1359-7345 DOI  

  Manasa, Kesari Lakshmi; Pujitha, Sravya; Sethi, Aaftaab; Mohammed, Arifuddin; Alvala, Mallika; Angeli, Andrea; Supuran, Claudiu T (2020). Synthesis and Biological Evaluation of Imidazo[2 ,1-b]Thiazole based Sulfonyl Piperazines as Novel Carbonic Anhydrase II Inhibitors. METABOLITES, vol. 10, pp. 136-136, ISSN:2218-1989 DOI  

  Vistoli, Giulio; Aldini, Giancarlo; Fumagalli, Laura; Dallanoce, Clelia; Angeli, Andrea; Supuran, Claudiu T. (2020). Activation Effects of Carnosine- and Histidine-Containing Dipeptides on Human Carbonic Anhydrases: A Comprehensive Study. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 21, pp. 1761-1761, ISSN:1422-0067 DOI  

  Meleddu R.; Distinto S.; Cottiglia F.; Angius R.; Caboni P.; Angeli A.; Melis C.; Deplano S.; Alcaro S.; Ortuso F.; Supuran C.T.; Maccioni E. (2020). New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII. ACS MEDICINAL CHEMISTRY LETTERS, pp. 0-0, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Nguyen, Giang T H; Nocentini, Alessio; Angeli, Andrea; Gratteri, Paola; Supuran, Claudiu T; Donald, William A (2020). Perfluoroalkyl Substances of Significant Environmental Concern Can Strongly Inhibit Human Carbonic Anhydrase Isozymes. ANALYTICAL CHEMISTRY, vol. 92, pp. 4614-4622, ISSN:0003-2700 DOI  

  Niccolò Chiaramonte, Soumia Maach, Caterina Biliotti, Andrea Angeli, Gian luca Bartolucci, Laura Braconi, Silvia Dei, Elisabetta Teodori, Claudiu T. Supuran, Maria Novella Romanelli (2020). Synthesis and carbonic anhydrase activating properties of a series of 2-amino-imidazolines structurally related to clonidine. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 1003-1010, ISSN:1475-6366 DOI  

  Urbanski L.J.; Angeli A.; Hytonen V.P.; Di Fiore A.; Parkkila S.; De Simone G.; Supuran C.T. (2020). Inhibition of the newly discovered β‑carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with inorganic anions and small molecules. JOURNAL OF INORGANIC BIOCHEMISTRY, vol. 213, pp. 111274-111274, ISSN:0162-0134 DOI  

  Thacker P.S.; Sridhar Goud N.; Argulwar O.S.; Soman J.; Angeli A.; Alvala M.; Arifuddin M.; Supuran C.T. (2020). Synthesis and biological evaluation of some coumarin hybrids as selective carbonic anhydrase IX and XII inhibitors. BIOORGANIC CHEMISTRY, vol. 104, pp. 104272-104272, ISSN:0045-2068 DOI  

  Felipe Raposo Passos Mansoldo; Fabrizio Carta; Andrea Angeli; Veronica da Silva Cardoso; Claudiu T. Supuran; Alane Beatriz Vermelho (2020). Chagas Disease: Perspectives on the Past and Present and Challenges in Drug Discovery. MOLECULES, vol. 25, pp. 0-0, ISSN:1420-3049 DOI  

  Kucukbay H.; Gonul Z.; Kucukbay F.Z.; Angeli A.; Bartolucci G.; Supuran C.T. (2020). Preparation, carbonic anhydrase enzyme inhibition and antioxidant activity of novel 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives incorporating mono or dipeptide moiety. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 1021-1026, ISSN:1475-6366 DOI  

  Chinchilli K.K.; Angeli A.; Thacker P.S.; Korra L.N.; Biswas R.; Arifuddin M.; Supuran C.T. (2020). Design, synthesis, and biological evaluation of 1,2,3-triazole-linked triazino[5,6-b]indole-benzene sulfonamide conjugates as potent carbonic anhydrase I, II, IX, and XIII inhibitors. METABOLITES, vol. 10, pp. 200-200, ISSN:2218-1989 DOI  

  Guzel-Akdemir O.; Carradori S.; Grande R.; Demir-Yazici K.; Angeli A.; Supuran C.T.; Akdemir A. (2020). Development of thiazolidinones as fungal carbonic anhydrase inhibitors. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 21, pp. 2960-2960, ISSN:1661-6596 DOI  

  Mancuso F.; De Luca L.; Angeli A.; Del Prete S.; Capasso C.; Supuran C.T.; Gitto R. (2020). Synthesis, computational studies and assessment of in vitro inhibitory activity of umbelliferon-based compounds against tumour-associated carbonic anhydrase isoforms IX and XII. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 1442-1449, ISSN:1475-6366 DOI  

  Singh P.; Swain B.; Thacker P.S.; Sigalapalli D.K.; Purnachander Yadav P.; Angeli A.; Supuran C.T.; Arifuddin M. (2020). Synthesis and carbonic anhydrase inhibition studies of sulfonamide based indole-1,2,3-triazole chalcone hybrids. BIOORGANIC CHEMISTRY, vol. 99, pp. 103839-103839, ISSN:0045-2068 DOI  

  Elzahhar P.A.; Abd El Wahab S.M.; Elagawany M.; Daabees H.; Belal A.S.F.; EL-Yazbi A.F.; Eid A.H.; Alaaeddine R.; Hegazy R.R.; Allam R.M.; Helmy M.W.; Bahaa Elgendy; Angeli A.; El-Hawash S.A.; Supuran C.T. (2020). Expanding the anticancer potential of 1,2,3-triazoles via simultaneously targeting Cyclooxygenase-2, 15-lipoxygenase and tumor-associated carbonic anhydrases. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 200, pp. 112439-112439, ISSN:0223-5234 DOI  

  Urbanski L.J.; Fiore A.D.; Azizi L.; Hytonen V.P.; Kuuslahti M.; Buonanno M.; Monti S.M.; Angeli A.; Emameh R.Z.; Supuran C.T.; De Simone G.; Parkkila S. (2020). Biochemical and structural characterisation of a protozoan beta-carbonic anhydrase from trichomonas vaginalis. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 1292-1299, ISSN:1475-6366 DOI  

  Mancuso F.; De Luca L.; Angeli A.; Berrino E.; Del Prete S.; Capasso C.; Supuran C.T.; Gitto R. (2020). In Silico-Guided Identification of New Potent Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae. ACS MEDICINAL CHEMISTRY LETTERS, vol. 11, pp. 2294-2299, ISSN:1948-5875 DOI  

  D'Ambrosio K.; Carradori S.; Cesa S.; Angeli A.; Monti S.M.; Supuran C.T.; De Simone G. (2020). Catechols: A new class of carbonic anhydrase inhibitors. CHEMICAL COMMUNICATIONS, vol. 56, pp. 13033-13036, ISSN:1359-7345 DOI  

  Angeli A.; Carta F.; Nocentini A.; Winum J.-Y.; Zalubovskis R.; Akdemir A.; Onnis V.; Eldehna W.M.; Capasso C.; Simone G.D.; Monti S.M.; Carradori S.; Donald W.A.; Dedhar S.; Supuran C.T. (2020). Carbonic anhydrase inhibitors targeting metabolism and tumor microenvironment. METABOLITES, vol. 10, pp. 1-21, ISSN:2218-1989 DOI  

  D'Ascenzio M.; Secci D.; Carradori S.; Zara S.; Guglielmi P.; Cirilli R.; Pierini M.; Poli G.; Tuccinardi T.; Angeli A.; Supuran C.T. (2020). 1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors. JOURNAL OF MEDICINAL CHEMISTRY, vol. 63, pp. 2470-2488, ISSN:0022-2623 DOI  

  Poli G.; Bozdag M.; Berrino E.; Angeli A.; Tuccinardi T.; Carta F.; Supuran C.T. (2020). N-aryl-N′-ureido-O-sulfamates as potent and selective inhibitors of hCA VB over hCA VA: Deciphering the binding mode of new potential agents in mitochondrial dysfunctions. BIOORGANIC CHEMISTRY, vol. 100, pp. 0-0, ISSN:0045-2068 DOI  

  Kaproń, Barbara; Czarnomysy, Robert; Wysokiński, Mariusz; Andrys, Rudolf; Musilek, Kamil; Angeli, Andrea; Supuran, Claudiu T; Plech, Tomasz (2020). 1,2,4-Triazole-based anticonvulsant agents with additional ROS scavenging activity are effective in a model of pharmacoresistant epilepsy. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 993-1002, ISSN:1475-6366 DOI  

  Andring J.T.; Fouch M.; Akocak S.; Angeli A.; Supuran C.T.; Ilies M.A.; McKenna R. (2020). Structural Basis of Nanomolar Inhibition of Tumor-Associated Carbonic Anhydrase IX: X-Ray Crystallographic and Inhibition Study of Lipophilic Inhibitors with Acetazolamide Backbone. JOURNAL OF MEDICINAL CHEMISTRY, vol. 63, pp. 13064-13075, ISSN:0022-2623 DOI  

  Urbanski L.J.; Bua S.; Angeli A.; Kuuslahti M.; Hytonen V.P.; Supuran C.T.; Parkkila S. (2020). Sulphonamide inhibition profile of Staphylococcus aureus β-carbonic anhydrase. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 1834-1839, ISSN:1475-6366 DOI  

  Angeli A.; Prete S.D.; Ghobril C.; Hitce J.; Clavaud C.; Marrat X.; Donald W.A.; Capasso C.; Supuran C.T. (2020). Activation studies of the β-carbonic anhydrases from Malassezia restricta with amines and amino acids. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 824-830, ISSN:1475-6366 DOI  

  Mancuso F.; Di Fiore A.; De Luca L.; Angeli A.; Monti S.M.; De Simone G.; Supuran C.T.; Gitto R. (2020). Looking toward the Rim of the Active Site Cavity of Druggable Human Carbonic Anhydrase Isoforms. ACS MEDICINAL CHEMISTRY LETTERS, pp. 0-0, ISSN:1948-5875 DOI  

  Ali, Majid; Bozdag, Murat; Farooq, Umar; Angeli, Andrea; Carta, Fabrizio; Berto, Paola; Zanotti, Giuseppe; Supuran, Claudiu T (2020). Benzylaminoethyureido-Tailed Benzenesulfonamides: Design, Synthesis, Kinetic and X-ray Investigations on Human Carbonic Anhydrases. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 21, pp. 2560-2560, ISSN:1422-0067 DOI  

  Thacker P.S.; Angeli A.; Argulwar O.S.; Tiwari P.L.; Arifuddin M.; Supuran C.T. (2020). Design, synthesis and biological evaluation of coumarin linked 1,2,4-oxadiazoles as selective carbonic anhydrase IX and XII inhibitors. BIOORGANIC CHEMISTRY, vol. 98, pp. 103739-103739, ISSN:0045-2068 DOI  

  Demir-Yazici K.; Guzel-Akdemir O.; Angeli A.; Supuran C.T.; Akdemir A. (2020). Novel indole-based hydrazones as potent inhibitors of the α-class carbonic anhydrase from pathogenic bacterium vibrio cholerae. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 21, pp. 3131-3131, ISSN:1422-0067 DOI  

  Carta F.; Vullo D.; Angeli A. (2020). Design, synthesis, and biological evaluation of selective hCA IX inhibitors. pH-Interfering Agents as Chemosensitizers in Cancer Therapy, pp. 63-78 DOI  

  Tanini, Damiano; Capperucci, Antonella; Ferraroni, Marta; Carta, Fabrizio; Angeli, Andrea; Supuran, Claudiu T. (2020). Direct and Straightforward access to substituted alkyl selenols as novel carbonic anhydrase inhibitors. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 185, pp. 111811-111817, ISSN:0223-5234 DOI  

  Pratesi, Debora; Matassini, Camilla; Goti, Andrea; Angeli, Andrea; Carta, Fabrizio; Supuran, Claudiu T.; Spanevello, Rolando; Cardona, Francesca (2020). Glycomimetic Based Approach toward Selective Carbonic Anhydrase Inhibitors. ACS MEDICINAL CHEMISTRY LETTERS, vol. 11, pp. 727-731, ISSN:1948-5875 DOI  

  Ciccone V.; Filippelli A.; Angeli A.; Supuran C.T.; Morbidelli L. (2020). Pharmacological inhibition of CA-IX impairs tumor cell proliferation, migration and invasiveness. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, vol. 21, pp. 2983-2983, ISSN:1661-6596 DOI  

  Llanos M.A.; Sbaraglini M.L.; Villalba M.L.; Ruiz M.D.; Carrillo C.; Soto C.A.; Talevi A.; Angeli A.; Parkkila S.; Supuran C.T.; Gavernet L. (2020). A structure-based approach towards the identification of novel antichagasic compounds: Trypanosoma cruzi carbonic anhydrase inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 21-30, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  Krasavin M.; Kalinin S.; Zozulya S.; Griniukova A.; Borysko P.; Angeli A.; Supuran C.T. (2020). Further validation of strecker-type α-aminonitriles as a new class of potent human carbonic anhydrase II inhibitors: hit expansion within the public domain using differential scanning fluorimetry leads to chemotype refinement. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 165-171, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  Swain B.; Angeli A.; Singh P.; Supuran C.T.; Arifuddin M. (2020). New coumarin/sulfocoumarin linked phenylacrylamides as selective transmembrane carbonic anhydrase inhibitors: Synthesis and in-vitro biological evaluation. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 28, pp. 115586-115586, ISSN:0968-0896 DOI  

  Guglielmi P.; Rotondi G.; Secci D.; Angeli A.; Chimenti P.; Nocentini A.; Bonardi A.; Gratteri P.; Carradori S.; Supuran C.T. (2020). Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 35, pp. 1891-1905, ISSN:1475-6366 DOI  

  Ali M.; Angeli A.; Bozdag M.; Carta F.; Capasso C.; Farooq U.; Supuran C.T. (2020). Benzylaminoethylureido-Tailed Benzenesulfonamides Show Potent Inhibitory Activity against Bacterial Carbonic Anhydrases. CHEMMEDCHEM, pp. 0-0, ISSN:1860-7179 DOI  

  Angeli A.; Ferraroni M.; Nocentini A.; Selleri S.; Gratteri P.; Supuran C.T.; Carta F. (2019). Polypharmacology of epacadostat: A potent and selective inhibitor of the tumor associated carbonic anhydrases IX and XII. CHEMICAL COMMUNICATIONS, vol. 55, pp. 5720-5723, ISSN:1359-7345 DOI   Accesso ONLINE all'editore

  Ammazzalorso A.; Carradori S.; Angeli A.; Akdemir A.; De Filippis B.; Fantacuzzi M.; Giampietro L.; Maccallini C.; Amoroso R.; Supuran C.T. (2019). Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 34, pp. 1051-1061, ISSN:1475-6366 DOI  

  Damiano Tanini, Antonella Capperucci, Claudiu T. Supuran, Andrea Angeli (2019). Sulfur, selenium and tellurium containing amines act as effective carbonic anhydrase activators. BIOORGANIC CHEMISTRY, vol. 87, pp. 516-523, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Angeli A.; Del Prete S.; Pinteala M.; Maier S.S.; Donald W.A.; Simionescu B.C.; Capasso C.; Supuran C.T. (2019). The first activation study of the β-carbonic anhydrases from the pathogenic bacteria Brucella suis and Francisella tularensis with amines and amino acids. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 34, pp. 1178-1185, ISSN:1475-6366 DOI  

  Thacker P.S.; Alvala M.; Arifuddin M.; Angeli A.; Supuran C.T. (2019). Design, synthesis and biological evaluation of coumarin-3-carboxamides as selective carbonic anhydrase IX and XII inhibitors. BIOORGANIC CHEMISTRY, vol. 86, pp. 386-392, ISSN:0045-2068 DOI  

  Angeli A.; Pinteala M.; Maier S.S.; Del Prete S.; Capasso C.; Simionescu B.C.; Supuran C.T. (2019). Inhibition of bacterial α-, β- and γ-class carbonic anhydrases with selenazoles incorporating benzenesulfonamide moieties. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 34, pp. 0-0, ISSN:1475-6374 DOI   Accesso ONLINE all'editore

  Angeli A.; Pinteala M.; Maier S.S.; Del Prete S.; Capasso C.; Simionescu B.C.; Supuran C.T. (2019). Inhibition of bacterial α-, β- and γ-class carbonic anhydrases with selenazoles incorporating benzenesulfonamide moieties. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 34, pp. 244-249, ISSN:1475-6366 DOI  

  Yamali C.; Gul H.I.; Ece A.; Bua S.; Angeli A.; Sakagami H.; Sahin E.; Supuran C.T. (2019). Synthesis, biological evaluation and in silico modelling studies of 1,3,5-trisubstituted pyrazoles carrying benzenesulfonamide as potential anticancer agents and selective cancer-associated hCA IX isoenzyme inhibitors. BIOORGANIC CHEMISTRY, vol. 92, pp. 103222-103222, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Narella S.G.; Shaik M.G.; Mohammed A.; Alvala M.; Angeli A.; Supuran C.T. (2019). Synthesis and biological evaluation of coumarin-1,3,4-oxadiazole hybrids as selective carbonic anhydrase IX and XII inhibitors. BIOORGANIC CHEMISTRY, vol. 87, pp. 765-772, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Angeli A.; Supuran C.T. (2019). Prostaglandin receptor agonists as antiglaucoma agents (a patent review 2013–2018). EXPERT OPINION ON THERAPEUTIC PATENTS, vol. 29, pp. 793-803, ISSN:1354-3776 DOI   Accesso ONLINE all'editore

  Buemi M.R.; Di Fiore A.; De Luca L.; Angeli A.; Mancuso F.; Ferro S.; Monti S.M.; Buonanno M.; Russo E.; De Sarro G.; De Simone G.; Supuran C.T.; Gitto R. (2019). Exploring structural properties of potent human carbonic anhydrase inhibitors bearing a 4-(cycloalkylamino-1-carbonyl)benzenesulfonamide moiety. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 163, pp. 443-452, ISSN:1768-3254 DOI   Accesso ONLINE all'editore

  Rotondi G.; Guglielmi P.; Carradori S.; Secci D.; De Monte C.; De Filippis B.; Maccallini C.; Amoroso R.; Cirilli R.; Akdemir A.; Angeli A.; Supuran C.T. (2019). Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 34, pp. 1400-1413, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  Swain B.; Singh Digwal C.; Angeli A.; Alvala M.; Singh P.; Supuran C.T.; Arifuddin M. (2019). Synthesis and exploration of 2-morpholino-4-phenylthiazol-5-yl acrylamide derivatives for their effects against carbonic anhydrase I, II, IX and XII isoforms as a non-sulfonamide class of inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 27, pp. 115090-115090, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Da'dara A.A.; Angeli A.; Ferraroni M.; Supuran C.T.; Skelly P.J. (2019). Crystal structure and chemical inhibition of essential schistosome host-interactive virulence factor carbonic anhydrase SmCA. COMMUNICATIONS BIOLOGY, vol. 2, pp. 333-333, ISSN:2399-3642 DOI   Accesso ONLINE all'editore

  Distinto S.; Meleddu R.; Ortuso F.; Cottiglia F.; Deplano S.; Sequeira L.; Melis C.; Fois B.; Angeli A.; Capasso C.; Angius R.; Alcaro S.; Supuran C.T.; Maccioni E. (2019). Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 34, pp. 1526-1533, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  Angeli A.; Pinteala M.; Maier S.S.; Del Prete S.; Capasso C.; Simionescu B.C.; Supuran C.T. (2019). Inhibition of α-, β-, γ-, δ-, ζ- and η-class carbonic anhydrases from bacteria, fungi, algae, diatoms and protozoans with famotidine. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 34, pp. 644-650, ISSN:1475-6366 DOI  

  Kurt B.Z.; Dag A.; Dogan B.; Durdagi S.; Angeli A.; Nocentini A.; Supuran C.T.; Sonmez F. (2019). Synthesis, biological activity and multiscale molecular modeling studies of bis-coumarins as selective carbonic anhydrase IX and XII inhibitors with effective cytotoxicity against hepatocellular carcinoma. BIOORGANIC CHEMISTRY, vol. 87, pp. 838-850, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Del Prete S.; Angeli A.; Ghobril C.; Hitce J.; Clavaud C.; Marat X.; Supuran C.T.; Capasso C. (2019). Anion inhibition profile of the β-carbonic anhydrase from the opportunist pathogenic fungus malassezia restricta involved in dandruff and seborrheic dermatitis. METABOLITES, vol. 9, pp. 147-147, ISSN:2218-1989 DOI   Accesso ONLINE all'editore

  Bozdag M.; Poli G.; Angeli A.; Lucarini E.; Tuccinardi T.; Di Cesare Mannelli L.; Selleri S.; Ghelardini C.; Winum J.-Y.; Carta F.; Supuran C.T. (2019). N-aryl-N’-ureido-O-sulfamates: Potent and selective inhibitors of the human Carbonic Anhydrase VII isoform with neuropathic pain relieving properties. BIOORGANIC CHEMISTRY, vol. 89, pp. 103033-103043, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Mustafa G.; Angeli A.; Zia-ur-Rehman M.; Akbar N.; Ishtiaq S.; Supuran C.T. (2019). An efficient method for the synthesis of novel derivatives 4-5-[4-(4-amino-5-mercapto-4H-[1,2,4]triazol-3-yl)-phenyl]-3-trifluoromethyl-pyrazol-1-yl-benzenesulfonamide and their anti-inflammatory potential. BIOORGANIC CHEMISTRY, vol. 91, pp. 103110-103110, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Zengin Kurt B.; Sonmez F.; Ozturk D.; Akdemir A.; Angeli A.; Supuran C.T. (2019). Synthesis of coumarin-sulfonamide derivatives and determination of their cytotoxicity, carbonic anhydrase inhibitory and molecular docking studies. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 183, pp. 111702-111702, ISSN:1768-3254 DOI   Accesso ONLINE all'editore

  Somers K.; Wen V.W.; Middlemiss S.M.C.; Osborne B.; Forgham H.; Jung M.S.; Karsa M.; Clifton M.; Bongers A.; Gao J.; Mayoh C.; Raoufi-Rad N.; Kusnadi E.P.; Hannan K.M.; Scott D.A.; Kwek A.; Liu B.; Flemming C.; Chudakova D.A.; Pandher R.; Failes T.W.; Lim J.; Angeli A.; Osterman A.L.; Imamura T.; Kees U.R.; Supuran C.T.; Pearson R.B.; Hannan R.D.; Davis T.P.; McCarroll J.; Kavallaris M.; Turner N.; Gudkov A.V.; Haber M.; Norris M.D.; Henderson M.J. (2019). A novel small molecule that kills a subset of MLL-rearranged leukemia cells by inducing mitochondrial dysfunction. ONCOGENE, vol. 38, pp. 3824-3842, ISSN:0950-9232 DOI   Accesso ONLINE all'editore

  Angeli A.; Di Cesare Mannelli L.; Ghelardini C.; Peat T.S.; Bartolucci G.; Menicatti M.; Carta F.; Supuran C.T. (2019). Benzensulfonamides bearing spyrohydantoin moieties act as potent inhibitors of human carbonic anhydrases II and VII and show neuropathic pain attenuating effects. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 177, pp. 188-197, ISSN:1768-3254 DOI   Accesso ONLINE all'editore

  Al-Tamimi A.-M.S.; Etxebeste-Mitxeltorena M.; Sanmartin C.; Jimenez-Ruiz A.; Syrjanen L.; Parkkila S.; Selleri S.; Carta F.; Angeli A.; Supuran C.T. (2019). Discovery of new organoselenium compounds as antileishmanial agents. BIOORGANIC CHEMISTRY, vol. 86, pp. 339-345, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Berrino E.; Milazzo L.; Micheli L.; Vullo D.; Angeli A.; Bozdag M.; Nocentini A.; Menicatti M.; Bartolucci G.; Di Cesare Mannelli L.; Ghelardini C.; Supuran C.T.; Carta F. (2019). Synthesis and evaluation of carbonic anhydrase inhibitors with carbon monoxide releasing properties for the management of rheumatoid arthritis. JOURNAL OF MEDICINAL CHEMISTRY, vol. 62, pp. 7233-7249, ISSN:1520-4804 DOI  

  Niccolò Chiaramontea, Silvia Bua, Andrea Angeli, Marta Ferraroni, Ilaria Picchioni, Gianluca Bartolucci, Laura Braconi, Silvia Dei, Elisabetta Teodori, Claudiu T. Supuran, Maria Novella Romanelli (2019). Sulfonamides incorporating piperazine bioisosteres as potent human carbonic anhydrase I, II, IV and IX inhibitors. BIOORGANIC CHEMISTRY, vol. 91, pp. 1-11, ISSN:0045-2068 DOI  

  Andrea Angeli; Lorenzo Di Cesare Mannelli; Carla Ghelardini; Thomas S. Peat; Gianluca Bartolucci; Marta Menicatti; Fabrizio Carta; Claudiu T. Supuran (2019). Benzensulfonamides bearing spyrohydantoin moieties act as potent inhibitors of human carbonic anhydrases {II} and {VII} and show neuropathic pain attenuating effects. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 177, pp. 188-197, ISSN:1768-3254 DOI  

  Angeli A.; Del Prete S.; Osman S.M.; AlOthman Z.; Donald W.A.; Capasso C.; Supuran C.T. (2019). Activation studies of the γ-carbonic anhydrases from the antarctic marine bacteria pseudoalteromonas haloplanktis and colwellia psychrerythraea with amino acids and amines. MARINE DRUGS, vol. 17, pp. 238-247, ISSN:1660-3397 DOI  

  Akdemir A.; Angeli A.; Goktas F.; Eraslan Elma P.; Karali N.; Supuran C.T. (2019). Novel 2-indolinones containing a sulfonamide moiety as selective inhibitors of candida β-carbonic anhydrase enzyme. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 34, pp. 528-531, ISSN:1475-6366 DOI  

  Payaz D.U.; Kucukbay F.Z.; Kucukbay H.; Angeli A.; Supuran C.T. (2019). Synthesis carbonic anhydrase enzyme inhibition and antioxidant activity of novel benzothiazole derivatives incorporating glycine, methionine, alanine, and phenylalanine moieties. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 34, pp. 343-349, ISSN:1475-6366 DOI  

  Swain B.; Angeli A.; Angapelly S.; Thacker P.S.; Singh P.; Supuran C.T.; Arifuddin M. (2019). Synthesis of a new series of 3-functionalised-1-phenyl-1,2,3-triazole sulfamoylbenzamides as carbonic anhydrase I, II, IV and IX inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 34, pp. 1199-1209, ISSN:1475-6366 DOI  

  Bozdag M.; Angeli A.; Tanc M. (2019). Mechanisms of action of carbonic anhydrase inhibitors: Compounds that anchor to the zinc-bound nucleophile. Carbonic Anhydrases Biochemistry and Pharmacology of an Evergreen Pharmaceutical Target, pp. 223-243 DOI  

  Tanini, Damiano; Ricci, Lorenzo; Capperucci, Antonella; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Peat, Thomas S; Carta, Fabrizio; Angeli, Andrea; Supuran, Claudiu T (2019). Synthesis of novel tellurides bearing benzensulfonamide moiety as carbonic anhydrase inhibitors with antitumor activity. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 181, pp. 111586-111594, ISSN:1768-3254 DOI  

  Andrea Angeli; Claudiu T Supuran (2019). Therapeutic Use of Carbonic Anhydrase Inhibitors and Their Multiple Drug Interactions. Pharmaceutical Biocatalysis, pp. 0-0

  Angeli, Andrea; Tanini, Damiano; Nocentini, Alessio; Capperucci, Antonella; Ferraroni, Marta; Gratteri, Paola; Supuran, Claudiu T.* (2019). Selenols: a new class of carbonic anhydrase inhibitors. CHEMICAL COMMUNICATIONS, vol. 55, pp. 648-651, ISSN:1359-7345 DOI   Accesso ONLINE all'editore

  angeli andrea (2019). Synthesis, characterization, biological assays and development of new enzyme modulators for the treatment of human pathologies. (Tutor: Claudiu T. Supuran)

  Kalinin, Stanislav; Nocentini, Alessio; Kovalenko, Alexander; Sharoyko, Vladimir; Bonardi, Alessandro; Angeli, Andrea; Gratteri, Paola; Tennikova, Tatiana B.; Supuran, Claudiu T.; Krasavin, Mikhail (2019). From random to rational: A discovery approach to selective subnanomolar inhibitors of human carbonic anhydrase IV based on the Castagnoli-Cushman multicomponent reaction. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 182, pp. 111642-111660, ISSN:1768-3254 DOI  

  Kalisha Vali Y.; Gundla R.; Singh O.V.; Tamboli Y.; Di Cesare Manelli L.; Ghelardini C.; Al-Tamimi A.-M.S.; Carta F.; Angeli A.; Supuran C.T. (2019). Spirocyclic sulfonamides with carbonic anhydrase inhibitory and anti-neuropathic pain activity. BIOORGANIC CHEMISTRY, vol. 92, pp. 103210-103220, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Bozdag, Murat; Ferraroni, Marta; Ward, Carol; Carta, Fabrizio; Bua, Silvia; Angeli, Andrea; Langdon, Simon P; Kunkler, Ian H; Al-Tamimi, Abdul-Malek S; Supuran, Claudiu T (2019). Carbonic anhydrase inhibitors based on sorafenib scaffold: Design, synthesis, crystallographic investigation and effects on primary breast cancer cells. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 182, pp. 111600-111611, ISSN:1768-3254 DOI  

  Thacker P.S.; Shaikh P.; Angeli A.; Arifuddin M.; Supuran C.T. (2019). Synthesis and biological evaluation of novel 8-substituted quinoline-2-carboxamides as carbonic anhydrase inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 34, pp. 1172-1177, ISSN:1475-6366 DOI  

  Abdel-Aziz A.A.-M.; Angeli A.; El-Azab A.S.; Hammouda M.E.A.; El-Sherbeny M.A.; Supuran C.T. (2019). Synthesis and anti-inflammatory activity of sulfonamides and carboxylates incorporating trimellitimides: Dual cyclooxygenase/carbonic anhydrase inhibitory actions. BIOORGANIC CHEMISTRY, vol. 84, pp. 260-268, ISSN:0045-2068 DOI  

  Tanini D.; Capperucci A.; Scopelliti M.; Milaneschi A.; Angeli A.; Supuran C.T. (2019). Syntesis of thio- and seleno-acetamides bearing benzenesulfonamide as potent inhibitors of human carbonic anhydrase II and XII. BIOORGANIC CHEMISTRY, vol. 89, pp. 102984-102984, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Angapelly, Srinivas; Ramya, P. V. Sri; Sodhi, Rohini; Angeli, Andrea; Rangan, Krishnan; Nagesh, Narayana; Supuran, Claudiu T.; Arifuddin, Mohammed* (2018). Iodine-mediated one-pot intramolecular decarboxylation domino reaction for accessing functionalised 2-(1,3,4-oxadiazol-2-yl)anilines with carbonic anhydrase inhibitory action. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 615-628, ISSN:1475-6366 DOI  

  Angeli, Andrea; Del Prete, Sonia; Osman, Sameh M; Alasmary, Fatmah A S; Alothman, Zeid; Donald, William A; Capasso, Clemente; Supuran, Claudiu T (2018). Activation studies of the α- and β-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae with amines and amino acids. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 227-233, ISSN:1475-6366 DOI  

  De Simone G.; Angeli A.; Bozdag M.; Supuran C.T.; Winum J.-Y.; Monti S.M.; Alterio V. (2018). Inhibition of carbonic anhydrases by a substrate analog: benzyl carbamate directly coordinates the catalytic zinc ion mimicking bicarbonate binding. CHEMICAL COMMUNICATIONS, vol. 54, pp. 10312-10315, ISSN:1359-7345 DOI   Accesso ONLINE all'editore

  Abdoli M.; Bozdag M.; Angeli A.; Supuran C.T. (2018). Benzamide-4-sulfonamides are effective human carbonic anhydrase I, II, VII, and IX inhibitors. METABOLITES, vol. 8, pp. 37-48, ISSN:2218-1989 DOI  

  Guzel-Akdemir O.; Angeli A.; Demir K.; Supuran C.T.; Akdemir A. (2018). Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 1299-1308, ISSN:1475-6366 DOI  

  Bonardi, Alessandro; Falsini, Matteo; Catarzi, Daniela; Varano, Flavia; Di Cesare Mannelli, Lorenzo; Tenci, Barbara; Ghelardini, Carla; Angeli, Andrea; Supuran, Claudiu T.; Colotta, Vittoria* (2018). Structural investigations on coumarins leading to chromeno[4,3-c]pyrazol-4-ones and pyrano[4,3-c]pyrazol-4-ones: New scaffolds for the design of the tumor-associated carbonic anhydrase isoforms IX and XII. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 146, pp. 47-59, ISSN:0223-5234 DOI   Accesso ONLINE all'editore

  Meleddu R.; Distinto S.; Cottiglia F.; Angius R.; Gaspari M.; Taverna D.; Melis C.; Angeli A.; Bianco G.; Deplano S.; Fois B.; Del Prete S.; Capasso C.; Alcaro S.; Ortuso F.; Yanez M.; Supuran C.T.; Maccioni E. (2018). Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides. ACS MEDICINAL CHEMISTRY LETTERS, vol. 9, pp. 1045-1050, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Angeli A.; Kuuslahti M.; Parkkila S.; Supuran C.T. (2018). Activation studies with amines and amino acids of the α-carbonic anhydrase from the pathogenic protozoan Trypanosoma cruzi. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 26, pp. 4187-4190, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Angeli A.; Buonanno M.; Donald W.A.; Monti S.M.; Supuran C.T. (2018). The zinc – but not cadmium – containing ζ-carbonic from the diatom Thalassiosira weissflogii is potently activated by amines and amino acids. BIOORGANIC CHEMISTRY, vol. 80, pp. 261-265, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Gul H.I.; Yamali C.; Sakagami H.; Angeli A.; Leitans J.; Kazaks A.; Tars K.; Ozgun D.O.; Supuran C.T. (2018). New anticancer drug candidates sulfonamides as selective hCA IX or hCA XII inhibitors. BIOORGANIC CHEMISTRY, vol. 77, pp. 411-419, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Angeli A.; Supuran C.T. (2018). Treatment of sleep apnea with a combination of a carbonic anhydrase inhibitor and an aldosterone antagonist: a patent evaluation of CA2958110 and IN6616DEN2012. EXPERT OPINION ON THERAPEUTIC PATENTS, vol. 28, pp. 723-727, ISSN:1354-3776 DOI   Accesso ONLINE all'editore

  Stefanucci A.; Angeli A.; Dimmito M.P.; Luisi G.; Del Prete S.; Capasso C.; Donald W.A.; Mollica A.; Supuran C.T. (2018). Activation of β- and γ-carbonic anhydrases from pathogenic bacteria with tripeptides. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 945-950, ISSN:1475-6366 DOI  

  Annunziato G.; Giovati L.; Angeli A.; Pavone M.; Del Prete S.; Pieroni M.; Capasso C.; Bruno A.; Conti S.; Magliani W.; Supuran C.T.; Costantino G. (2018). Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 1537-1544, ISSN:1475-6366 DOI   Accesso ONLINE all'editore

  Angeli A.; Del Prete S.; Alasmary F.A.S.; Alqahtani L.S.; AlOthman Z.; Donald W.A.; Capasso C.; Supuran C.T. (2018). The first activation studies of the η-carbonic anhydrase from the malaria parasite Plasmodium falciparum with amines and amino acids. BIOORGANIC CHEMISTRY, vol. 80, pp. 94-98, ISSN:0045-2068 DOI  

  Angeli A.; Abbas G.; del Prete S.; Capasso C.; Supuran C.T. (2018). Selenides bearing benzenesulfonamide show potent inhibition activity against carbonic anhydrases from pathogenic bacteria Vibrio cholerae and Burkholderia pseudomallei. BIOORGANIC CHEMISTRY, vol. 79, pp. 319-322, ISSN:0045-2068 DOI  

  Bozdag M.; Carta F.; Angeli A.; Osman S.M.; Alasmary F.A.S.; AlOthman Z.; Supuran C.T. (2018). Synthesis of N′-phenyl-N-hydroxyureas and investigation of their inhibitory activities on human carbonic anhydrases. BIOORGANIC CHEMISTRY, vol. 78, pp. 1-6, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Zolnowska B.; Slawinski J.; Szafranski K.; Angeli A.; Supuran C.T.; Kawiak A.; Wieczor M.; Zielinska J.; Baczek T.; Bartoszewska S. (2018). Novel 2-(2-arylmethylthio-4-chloro-5-methylbenzenesulfonyl)-1-(1,3,5-triazin-2-ylamino)guanidine derivatives: Inhibition of human carbonic anhydrase cytosolic isozymes I and II and the transmembrane tumor-associated isozymes IX and XII, anticancer activity, and molecular modeling studies. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 143, pp. 1931-1941, ISSN:1768-3254 DOI   Accesso ONLINE all'editore

  Mocan A.; Carradori S.; Locatelli M.; Secci D.; Cesa S.; Mollica A.; Riga S.; Angeli A.; Supuran C.T.; Celia C.; Di Marzio L. (2018). Bioactive isoflavones from Pueraria lobata root and starch: Different extraction techniques and carbonic anhydrase inhibition. FOOD AND CHEMICAL TOXICOLOGY, vol. 112, pp. 441-447, ISSN:0278-6915 DOI   Accesso ONLINE all'editore

  Mishra C.B.; Kumari S.; Angeli A.; Bua S.; Buonanno M.; Monti S.M.; Tiwari M.; Supuran C.T. (2018). Discovery of potent anti-convulsant carbonic anhydrase inhibitors: Design, synthesis, in vitro and in vivo appraisal. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 156, pp. 430-443, ISSN:0223-5234 DOI  

  Angeli, Andrea; Di Cesare Mannelli, Lorenzo; Trallori, Elena; Peat, Thomas S.; Ghelardini, Carla; Carta, Fabrizio; Supuran, Claudiu T.* (2018). Design, Synthesis, and X-ray of Selenides as New Class of Agents for Prevention of Diabetic Cerebrovascular Pathology. ACS MEDICINAL CHEMISTRY LETTERS, vol. 9, pp. 462-467, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Tanini, Damiano; Capperucci, Antonella; Malevolti, Gianni; Turco, Francesca; Ferraroni, Marta; Supuran, Claudiu T.* (2018). Synthesis of different thio-scaffolds bearing sulfonamide with subnanomolar carbonic anhydrase II and IX inhibitory properties and X-ray investigations for their inhibitory mechanism. BIOORGANIC CHEMISTRY, vol. 81, pp. 642-648, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Ferraroni, Marta; Supuran, Claudiu T.* (2018). Famotidine, an Antiulcer Agent, Strongly Inhibits Helicobacter pylori and Human Carbonic Anhydrases. ACS MEDICINAL CHEMISTRY LETTERS, vol. 9, pp. 1035-1038, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Chiaramonte, Niccolò; Manetti, Dina; Romanelli, Maria Novella; Supuran, Claudiu T (2018). Investigation of piperazines as human carbonic anhydrase I, II, IV and VII activators. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 303-308, ISSN:1475-6366 DOI  

  Angeli, Andrea; Donald, William A.; Parkkila, Seppo; Supuran, Claudiu T. (2018). Activation studies with amines and amino acids of the β-carbonic anhydrase from the pathogenic protozoan Leishmania donovani chagasi. BIOORGANIC CHEMISTRY, vol. 78, pp. 406-410, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Métayer, Benoit; Angeli, Andrea; Mingot, Agnès; Jouvin, Kévin; Evano, Gwilherm; Supuran, Claudiu T.; Thibaudeau, Sébastien* (2018). Fluoroenesulphonamides: N-sulphonylurea isosteres showing nanomolar selective cancer-related transmembrane human carbonic anhydrase inhibition. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 804-808, ISSN:1475-6366 DOI  

  Mishra, Chandra Bhushan; Kumari, Shikha; Angeli, Andrea; Bua, Silvia; Tiwari, Manisha*; Supuran, Claudiu T. (2018). Discovery of benzenesulfonamide derivatives as carbonic anhydrase inhibitors with effective anticonvulsant action: Design, synthesis, and pharmacological evaluation. JOURNAL OF MEDICINAL CHEMISTRY, vol. 61, pp. 3151-3165, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Alasmary, Fatmah A. S.; Del Prete, Sonia; Osman, Sameh M.; AlOthman, Zeid; Donald, William A.; Capasso, Clemente; Supuran, Claudiu T. (2018). The first activation study of a δ-carbonic anhydrase: TweCAδ from the diatom Thalassiosira weissflogii is effectively activated by amines and amino acids. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 680-685, ISSN:1475-6366 DOI  

  Vats, Lalit; Sharma, Vikas; Angeli, Andrea; Kumar, Rajiv; Supuran, Claudiu T.; Sharma, Pawan K.* (2018). Synthesis of novel 4-functionalized 1,5-diaryl-1,2,3-triazoles containing benzenesulfonamide moiety as carbonic anhydrase I, II, IV and IX inhibitors. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 150, pp. 678-686, ISSN:0223-5234 DOI   Accesso ONLINE all'editore

  Akgul, Ozlem; Di Cesare Mannelli, Lorenzo; Vullo, Daniela; Angeli, Andrea; Ghelardini, Carla; Bartolucci, Gianluca; Altamimi, Abdulmalik Saleh Alfawaz; Scozzafava, Andrea; Supuran, Claudiu T; Carta, Fabrizio (2018). Discovery of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Management of Rheumatoid Arthritis. JOURNAL OF MEDICINAL CHEMISTRY, pp. 1-60, ISSN:0022-2623 DOI  

  Angapelly, Srinivas; Angeli, Andrea; Jabbar Khan, Arbaj; SriRamya, Posa Venkata; Supuran, Claudiu Trandafir; Arifuddin, Mohammed (2018). Synthesis and Biological Evaluation of 4-sulfamoylphenyl/sulfocoumarin carboxamides as selective inhibitors of carbonic anhydrase isoforms hCA II, IX and XII. CHEMMEDCHEM, pp. 1-9, ISSN:1860-7179 DOI  

  Gul, Halise Inci*; Yamali, Cem; Bulbuller, Merve; Kirmizibayrak, Petek Ballar; Gul, Mustafa; Angeli, Andrea; Bua, Silvia; Supuran, Claudiu T. (2018). Anticancer effects of new dibenzenesulfonamides by inducing apoptosis and autophagy pathways and their carbonic anhydrase inhibitory effects on hCA I, hCA II, hCA IX, hCA XII isoenzymes. BIOORGANIC CHEMISTRY, vol. 78, pp. 290-297, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Trallori, Elena; Ferraroni, Marta; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Supuran, Claudiu T.* (2018). Discovery of new 2, 5-disubstituted 1,3-selenazoles as selective human carbonic anhydrase IX inhibitors with potent anti-tumor activity. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 157, pp. 1214-1222, ISSN:0223-5234 DOI   Accesso ONLINE all'editore

  Angeli A, di Cesare Mannelli L, Lucarini E, Peat TS, Ghelardini C, Supuran CT (2018). Design, synthesis and X-ray crystallography of selenides bearing benzenesulfonamide moiety with neuropathic pain modulating effects.. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, pp. 210-219, ISSN:0223-5234 DOI  

  Angeli, Andrea; Trallori, Elena; Carta, Fabrizio; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Supuran, Claudiu T.* (2018). Heterocoumarins Are Selective Carbonic Anhydrase IX and XII Inhibitors with Cytotoxic Effects against Cancer Cells Lines. ACS MEDICINAL CHEMISTRY LETTERS, vol. 9, pp. 947-951, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Melis C.; Distinto S.; Bianco G.; Meleddu R.; Cottiglia F.; Fois B.; Taverna D.; Angius R.; Alcaro S.; Ortuso F.; Gaspari M.; Angeli A.; Del Prete S.; Capasso C.; Supuran C.T.; Maccioni E. (2018). Targeting Tumor Associated Carbonic Anhydrases IX and XII: Highly Isozyme Selective Coumarin and Psoralen Inhibitors. ACS MEDICINAL CHEMISTRY LETTERS, vol. 9, pp. 725-729, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Tanini, Damiano; Capperucci, Antonella; Supuran, Claudiu T. (2018). First evaluation of organotellurium derivatives as carbonic anhydrase I, II, IV, VII and IX inhibitors. BIOORGANIC CHEMISTRY, vol. 76, pp. 268-272, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  De Luca, Laura; Mancuso, Francesca; Ferro, Stefania; Buemi, Maria Rosa; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T.; Gitto, Rosaria (2018). Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 143, pp. 276-282, ISSN:0223-5234 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Del Prete, Sonia; Donald, William A.; Capasso, Clemente; Supuran, Claudiu T. (2018). The γ-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae is potently activated by amines and amino acids. BIOORGANIC CHEMISTRY, vol. 77, pp. 1-5, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Del Prete, Sonia; Osman, Sameh M; Alasmary, Fatmah A S; Alothman, Zeid; Donald, William A; Capasso, Clemente; Supuran, Claudiu T (2018). Activation studies with amines and amino acids of the β-carbonic anhydrase encoded by the Rv3273 gene from the pathogenic bacterium Mycobacterium tuberculosis. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 33, pp. 364-369, ISSN:1475-6366 DOI  

  Mikus P.; Krajciova D.; Mikulova M.; Horvath B.; Pecher D.; Garaj V.; Bua S.; Angeli A.; Supuran C.T. (2018). Novel sulfonamides incorporating 1,3,5-triazine and amino acid structural motifs as inhibitors of the physiological carbonic anhydrase isozymes I, II and IV and tumor-associated isozyme IX. BIOORGANIC CHEMISTRY, vol. 81, pp. 241-252, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Vaiano, Fabio; Mari, Francesco; Bertol, Elisabetta; Supuran, Claudiu T (2017). Psychoactive substances belonging to the amphetamine class potently activate brain carbonic anhydrase isoforms VA, VB, VII, and XII. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 32, pp. 1253-1259-1259, ISSN:1475-6366 DOI  

  Angapelly, Srinivas; Sri Ramya, P. V.; Angeli, Andrea; Supuran, Claudiu T.; Arifuddin, Mohammed (2017). Sulfocoumarin-, Coumarin-, 4-Sulfamoylphenyl-Bearing Indazole-3-carboxamide Hybrids: Synthesis and Selective Inhibition of Tumor-Associated Carbonic Anhydrase Isozymes IX and XII. CHEMMEDCHEM, vol. 12, pp. 1578-1584, ISSN:1860-7179 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Abbas, Ghulam; Del Prete, Sonia; Carta, Fabrizio; Capasso, Clemente; Supuran, Claudiu T. (2017). Acyl selenoureido benzensulfonamides show potent inhibitory activity against carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. BIOORGANIC CHEMISTRY, vol. 75, pp. 170-172, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Mishra, Chandra Bhushan; Kumari, Shikha; Angeli, Andrea; Monti, Simona Maria; Buonanno, Martina; Tiwari, Manisha; Supuran, Claudiu T (2017). Discovery of Benzenesulfonamides with Potent Human Carbonic Anhydrase Inhibitory and Effective Anticonvulsant Action: Design, Synthesis, and Pharmacological Assessment. JOURNAL OF MEDICINAL CHEMISTRY, vol. 60, pp. 2456-2469, ISSN:0022-2623 DOI  

  Melis, Claudia; Meleddu, Rita; Angeli, Andrea; Distinto, Simona; Bianco, Giulia; Capasso, Clemente; Cottiglia, Filippo; Angius, Rossella; Supuran, CLAUDIU TRANDAFIR; Maccioni, Elias (2017). Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 32, pp. 68-73, ISSN:1475-6366 DOI  

  Angeli, Andrea; Tanini, Damiano; Viglianisi, Caterina; Panzella, Lucia; Capperucci, Antonella; Menichetti, Stefano; Supuran, Claudiu T (2017). Evaluation of selenide, diselenide and selenoheterocycle derivatives as carbonic anhydrase I, II, IV, VII and IX inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 25, pp. 2518-2523, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Abdel-Aziz, Alaa A. -. M.; Nocentini, Alessio; El-Azab, Adel S.; Gratteri, Paola; Supuran, Claudiu T. (2017). Synthesis and carbonic anhydrase inhibition of polycyclic imides incorporating N-benzenesulfonamide moieties. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 25, pp. 5373-5379, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Bruno E.; Buemi M.R.; Di Fiore A.; De Luca L.; Ferro S.; Angeli A.; Cirilli R.; Sadutto D.; Alterio V.; Monti S.M.; Supuran C.T.; De Simone G.; Gitto R. (2017). Probing Molecular Interactions between Human Carbonic Anhydrases (hCAs) and a Novel Class of Benzenesulfonamides. JOURNAL OF MEDICINAL CHEMISTRY, vol. 60, pp. 4316-4326, ISSN:0022-2623 DOI  

  Abdoli M.; Angeli A.; Bozdag M.; Carta F.; Kakanejadifard A.; Saeidian H.; Supuran C.T. (2017). Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo[d]thiazole-5- and 6-sulfonamides. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 32, pp. 1071-1078, ISSN:1475-6366 DOI  

  Bianco G, Meleddu R, Distinto S, Cottiglia F, Gaspari M, Melis C, Corona A, Angius R, Angeli A, Taverna D, Alcaro S, Leitans J, Kazaks A, Tars K, Supuran CT, Maccioni E. (2017). N-Acylbenzenesulfonamide Dihydro-1,3,4-oxadiazole Hybrids: Seeking Selectivity toward Carbonic Anhydrase Isoforms. ACS MEDICINAL CHEMISTRY LETTERS, pp. 792-796, ISSN:1948-5875 DOI  

  Karali N.; Akdemir A.; Goktas F.; Eraslan Elma P.; Angeli A.; Kizilirmak M.; Supuran C.T. (2017). Novel sulfonamide-containing 2-indolinones that selectively inhibit tumor-associated alpha carbonic anhydrases. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 25, pp. 3714-3718, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Zengin Kurt B.; Sonmez F.; Durdagi S.; Aksoydan B.; Ekhteiari Salmas R.; Angeli A.; Kucukislamoglu M.; Supuran C.T. (2017). Synthesis, biological activity and multiscale molecular modeling studies for coumaryl-carboxamide derivatives as selective carbonic anhydrase IX inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 32, pp. 1042-1052, ISSN:1475-6366 DOI  

  De Vita D.; Angeli A.; Pandolfi F.; Bortolami M.; Costi R.; Di Santo R.; Suffredini E.; Ceruso M.; Del Prete S.; Capasso C.; Scipione L.; Supuran C.T. (2017). Inhibition of the α-carbonic anhydrase from Vibrio cholerae with amides and sulfonamides incorporating imidazole moieties. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 32, pp. 798-804, ISSN:1475-6366 DOI  

  Krasavin, Mikhail; Shetnev, Anton; Sharonova, Tatyana; Baykov, Sergey; Tuccinardi, Tiziano; Kalinin, Stanislav; Angeli, Andrea; Supuran, Claudiu T. (2017). Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1,2,4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic hCA II and membrane-bound hCA IX isoforms. BIOORGANIC CHEMISTRY, vol. 76, pp. 88-97, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Kalinin, Stanislav; Kopylov, Stanislav; Tuccinardi, Tiziano; Sapegin, Alexander; Dar'In, Dmitry; Angeli, Andrea; Supuran, Claudiu T.; Krasavin, Mikhail (2017). Lucky Switcheroo: Dramatic Potency and Selectivity Improvement of Imidazoline Inhibitors of Human Carbonic Anhydrase VII. ACS MEDICINAL CHEMISTRY LETTERS, vol. 8, pp. 1105-1109, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Angapelly S.; Ramya P.V.S.; Angeli A.; Del Prete S.; Capasso C.; Arifuddin M.; Supuran C.T. (2017). Development of sulfonamides incorporating phenylacrylamido functionalities as carbonic anhydrase isoforms I, II, IX and XII inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 25, pp. 5726-5732, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Tanini, Damiano; Capperucci, Antonella; Supuran, Claudiu T. (2017). Synthesis of Novel Selenides Bearing Benzenesulfonamide Moieties as Carbonic Anhydrase I, II, IV, VII, and IX Inhibitors. ACS MEDICINAL CHEMISTRY LETTERS, vol. 8, pp. 1213-1217, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Angeli, Andrea; Carta, Fabrizio; Bartolucci, Gian Luca; Supuran, Claudiu T.* (2017). Synthesis of novel acyl selenoureido benzensulfonamides as carbonic anhydrase I, II, VII and IX inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 25, pp. 3567-3573, ISSN:0968-0896 DOI   Accesso ONLINE all'editore

  Mollica, Adriano; Macedonio, Giorgia; Stefanucci, Azzurra; Carradori, Simone; Akdemir, Atilla; Angeli, Andrea; Supuran, Claudiu T (2017). Five- and Six-Membered Nitrogen-Containing Compounds as Selective Carbonic Anhydrase Activators. MOLECULES, vol. 22, pp. 1-13, ISSN:1420-3049 DOI  

  Bruno E.; Buemi M.R.; Di Fiore A.; De Luca L.; Ferro S.; Angeli A.; Cirilli R.; Sadutto D.; Alterio V.; Monti S.M.; Supuran C.T.; De Simone G.; Gitto R. (2017). Probing Molecular Interactions between Human Carbonic Anhydrases (hCAs) and a Novel Class of Benzenesulfonamides. JOURNAL OF MEDICINAL CHEMISTRY, vol. 60, pp. 4316-4326, ISSN:0022-2623 DOI  

  Angeli, Andrea; Tanini, Damiano; Peat, Thomas S. ; Di Cesare Mannelli,Lorenzo; Bartolucci, Gian Luca; Capperucci, Antonella; Ghelardini, Carla; Supuran, Claudiu T.; and Carta, Fabrizio (2017). Discovery of New Selenoureido Analogues of 4-(4-Fluorophenylureido)benzenesulfonamide as Carbonic Anhydrase Inhibitors. ACS MEDICINAL CHEMISTRY LETTERS, vol. 8, pp. 963-968, ISSN:1948-5875 DOI   Accesso ONLINE all'editore

  Fragai, Marco; Comito, Giuseppina; Di Cesare Mannelli, Lorenzo; Gualdani, Roberta; Calderone, Vito; Louka, Alexandra; Richichi, Barbara; Francesconi, Oscar; Angeli, Andrea; Nocentini, Alessio; Gratteri, Paola; Chiarugi, Paola; Ghelardini, Carla; Tadini-Buoninsegni, Francesco; Supuran, Claudiu T; Nativi, Cristina (2017). Lipoyl-Homotaurine Derivative (ADM_12) Reverts Oxaliplatin-Induced Neuropathy and Reduces Cancer Cells Malignancy by Inhibiting Carbonic Anhydrase IX (CAIX). JOURNAL OF MEDICINAL CHEMISTRY, vol. 60, pp. 9003-9011, ISSN:1520-4804 DOI  

  Sapegin, Alexander; Kalinin, Stanislav; Angeli, Andrea; Supuran, Claudiu T.; Krasavin, Mikhail (2017). Unprotected primary sulfonamide group facilitates ring-forming cascade en route to polycyclic [1,4]oxazepine-based carbonic anhydrase inhibitors. BIOORGANIC CHEMISTRY, vol. 76, pp. 140-146, ISSN:0045-2068 DOI   Accesso ONLINE all'editore

  Ramya, P. V. Sri; Angapelly, Srinivas; Angeli, Andrea; Digwal, Chander Singh; Arifuddin, Mohammed; Babu, Bathini Nagendra; Supuran, Claudiu T; Kamal, Ahmed (2017). Discovery of curcumin inspired sulfonamide derivatives as a new class of carbonic anhydrase isoforms I, II, IX, and XII inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 32, pp. 1274-1281, ISSN:1475-6366 DOI  

  Abdel-Aziz, Aa; Angeli, A; El-Azab, As; Abu El-Enin, Ma; Supuran, Ct (2017). Synthesis and biological evaluation of cyclic imides incorporating benzenesulfonamide moieties as carbonic anhydrase I, II, IV and IX inhibitors.. BIOORGANIC & MEDICINAL CHEMISTRY, pp. 31418-31423, ISSN:0968-0896 DOI  

  Falsini, Matteo; Squarcialupi, Lucia; Catarzi, Daniela; Varano, Flavia; Betti, Marco; Di Cesare Mannelli, Lorenzo; Tenci, Barbara; Ghelardini, Carla; Tanc, Muhammet; Angeli, Andrea; Supuran, Claudiu T.; Colotta, Vittoria (2017). 3-Hydroxy-1H-quinazoline-2,4-dione as a New Scaffold to Develop Potent and Selective Inhibitors of the Tumor-Associated Carbonic Anhydrases IX and XII. JOURNAL OF MEDICINAL CHEMISTRY, vol. 60, pp. 6428-6439, ISSN:0022-2623 DOI   Accesso ONLINE all'editore

  Mollica, Adriano; Locatelli, Marcello; Macedonio, Giorgia; Carradori, Simone; Sobolev, Anatoly P.; De Salvador, Roberto F.; Monti, Simona M.; Buonanno, Martina; Zengin, Gokhan; Angeli, Andrea; Supuran, Claudiu T. (2016). Microwave-assisted extraction, HPLC analysis, and inhibitory effects on carbonic anhydrase I, II, VA, and VII isoforms of 14 blueberry Italian cultivars. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 31, pp. 1-6, ISSN:1475-6366 DOI  

  Annunziato, Giannamaria; Angeli, Andrea; D'Alba, Francesca; Bruno, Agostino; Pieroni, Marco; Vullo, Daniela; De Luca, Viviana; Capasso, Clemente; Supuran, Claudiu T.; Costantino, Gabriele (2016). Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches. CHEMMEDCHEM, vol. 11, pp. 1904-1914, ISSN:1860-7179 DOI   Accesso ONLINE all'editore

  Mishra, Chandra Bhushan; Kumari, Shikha; Angeli, Andrea; Monti, Simona Maria; Buonanno, Martina; Prakash, Amresh; Tiwari, Manisha; Supuran, Claudiu T. (2016). Design, synthesis and biological evaluation of N-(5-methyl-isoxazol-3-yl/1,3,4-thiadiazol-2-yl)-4-(3-substitutedphenylureido) benzenesulfonamides as human carbonic anhydrase isoenzymes I, II, VII and XII inhibitors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, vol. 31, pp. 174-179, ISSN:1475-6366 DOI  

  Tanini, Damiano; Angeli, Andrea; Capperucci, Antonella (2016). Ionic liquids as an alternative reaction medium for HMDST based synthesis of thioaldehydes. PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, vol. 191, pp. 156-158, ISSN:1042-6507 DOI   Accesso ONLINE all'editore

  Angeli, A; Peat, T.S.; Bartolucci, G.; Nocentini, A.; Supuran, C.T.; Carta, F. (2016). Intramolecular oxidative deselenization of acylselenoureas: a facile synthesis of benzoxazole amides and carbonic anhydrase inhibitors. ORGANIC & BIOMOLECULAR CHEMISTRY, vol. 14, pp. 11353-11356, ISSN:1477-0520 DOI   Accesso ONLINE all'editore

  Annunziato G.; Angeli A.; D'Alba F.; Bruno A.; Pieroni M.; Vullo D.; De Luca V.; Capasso C.; Supuran C.T.; Costantino G. (2016). Cover Picture: Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches (ChemMedChem 17/2016). CHEMMEDCHEM, vol. 11, pp. 1876-1876, ISSN:1860-7179 DOI   Accesso ONLINE all'editore

  Abdel Gawad, Nagwa M.; Amin, Noha H.; Elsaadi, Mohammed T.; Mohamed, Fatma M.M.; Angeli, Andrea; De Luca, Viviana; Capasso, Clemente; Supuran, Claudiu T (2016). Synthesis of 4-(thiazol-2-ylamino)-benzenesulfonamides with carbonic anhydrase I, II and IX inhibitory activity and cytotoxic effects against breast cancer cell lines. BIOORGANIC & MEDICINAL CHEMISTRY, vol. 24, pp. 3043-3051, ISSN:0968-0896 DOI   Accesso ONLINE all'editore